日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Lead optimization of 5jc21 (CG13250), a quinolin-2(1H)-one-based inhibitor of the BRD4 member of the bromodomain and extraterminal (BET) family of proteins

对 5jc21 (CG13250) 进行先导化合物优化,5jc21 是一种基于喹啉-2(1H)-酮的 BRD4 抑制剂,属于溴结构域和末端外结构域 (BET) 蛋白家族。

Chauhan, Jay; Pogash, Sarah; Yoshioka, Makoto; Raje, Mithun; Van Eker, Daniel; Strovel, Jeffrey W; Fletcher, Steven

A phase 1 study of the amino acid modulator pegcrisantaspase and venetoclax for relapsed or refractory acute myeloid leukemia

一项针对复发或难治性急性髓系白血病的氨基酸调节剂pegcrisantaspase和venetoclax的I期研究

Liu, Yuchen; Bollino, Dominique R; Bah, Osman M; Strovel, Erin T; Le, Tien V; Zarrabi, Jinoos; Philip, Sunita; Lapidus, Rena G; Baer, Maria R; Niyongere, Sandrine; Duong, Vu H; Dougherty, Christine C; Beumer, Jan H; Caprinolo, Katherine D; Kamangar, Farin; Emadi, Ashkan

Clinical and biochemical footprints of inherited metabolic diseases: XVII. Dysmorphisms

遗传性代谢疾病的临床和生化特征:十七、畸形

Greene, Carol L; Saenz-Ayala, Sofia; Strovel, Erin T; Rossignol, Francis; Ferreira, Carlos R; Blau, Nenad

Long-acting Erwinia chrysanthemi, Pegcrisantaspase, induces alternate amino acid biosynthetic pathways in a preclinical model of pancreatic ductal adenocarcinoma

长效菊欧文氏菌 Pegcrisantaspase 在胰腺导管腺癌的临床前模型中诱导替代氨基酸生物合成途径

Dominique Bollino, Kanwal Hameed, Anusha Bhat, Arveen Zarrabi, Andrea Casildo, Xinrong Ma, Kayla M Tighe, Brandon Carter-Cooper, Erin T Strovel, Rena G Lapidus, Ashkan Emadi

Venetoclax and pegcrisantaspase for complex karyotype acute myeloid leukemia

维奈克拉和聚乙二醇化物蛋白酶治疗复杂核型急性髓系白血病

Ashkan Emadi, Bandish Kapadia, Dominique Bollino, Binny Bhandary, Maria R Baer, Sandrine Niyongere, Erin T Strovel, Hannah Kaizer, Elizabeth Chang, Eun Yong Choi, Xinrong Ma, Kayla M Tighe, Brandon Carter-Cooper, Blake S Moses, Curt I Civin, Anup Mahurkar, Amol C Shetty, Ronald B Gartenhaus, Farin K

Predicting Novel Therapies and Targets: Regulation of Notch3 by the Bromodomain Protein BRD4

预测新型疗法和靶点:溴结构域蛋白 BRD4 对 Notch3 的调控

Alejandro Villar-Prados,Sherry Y Wu,Karem A Court,Shaolin Ma,Christopher LaFargue,Mamur A Chowdhury,Margaret I Engelhardt,Cristina Ivan,Prahlad T Ram,Ying Wang,Keith Baggerly,Cristian Rodriguez-Aguayo,Gabriel Lopez-Berestein,Shyh Ming-Yang,David J Maloney,Makoto Yoshioka,Jeffrey W Strovel,Jason Roszik #,Anil K Sood #

Newborn Screening Long Term Follow-Up in the Medical Home

新生儿筛查长期随访在医疗之家进行

Badawi, Deborah; Bisordi, Katharine; Timmel, Marilyn J; Sorongon, Scott; Strovel, Erin

Lead optimization and efficacy evaluation of quinazoline-based BET family inhibitors for potential treatment of cancer and inflammatory diseases

喹唑啉类BET家族抑制剂的先导化合物优化和疗效评价,用于治疗癌症和炎症性疾病

Yang, Shyh-Ming; Yoshioka, Makoto; Strovel, Jeffrey W; Urban, Daniel J; Hu, Xin; Hall, Matthew D; Jadhav, Ajit; Maloney, David J

Identification of a Small Molecule That Selectively Inhibits ERG-Positive Cancer Cell Growth

鉴定出一种选择性抑制 ERG 阳性癌细胞生长的小分子

Ahmed A Mohamed #, Charles P Xavier #, Gauthaman Sukumar, Shyh-Han Tan, Lakshmi Ravindranath, Nishat Seraj, Vineet Kumar, Taduru Sreenath, David G McLeod, Gyorgy Petrovics, Inger L Rosner, Meera Srivastava, Jeffrey Strovel, Sanjay V Malhotra, Nicole A LaRonde, Albert Dobi, Clifton L Dalgard, Shiv Sr

Discovery and lead identification of quinazoline-based BRD4 inhibitors

基于喹唑啉的BRD4抑制剂的发现和先导化合物鉴定

Yang, Shyh-Ming; Urban, Daniel J; Yoshioka, Makoto; Strovel, Jeffrey W; Fletcher, Steven; Wang, Amy Q; Xu, Xin; Shah, Pranav; Hu, Xin; Hall, Matthew D; Jadhav, Ajit; Maloney, David J