日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vivo efficacy of the boron-pleuromutilin AN11251 against Wolbachia of the rodent filarial nematode Litomosoides sigmodontis

硼-截短侧耳素AN11251对啮齿类丝状线虫Litomosoides sigmodontis沃尔巴克氏体的体内疗效

Ehrens, Alexandra; Lunde, Christopher S; Jacobs, Robert T; Struever, Dominique; Koschel, Marianne; Frohberger, Stefan J; Lenz, Franziska; Fendler, Martina; Turner, Joseph D; Ward, Stephen A; Taylor, Mark J; Freund, Yvonne R; Stefanakis, Rianna; Easom, Eric; Li, Xianfeng; Plattner, Jacob J; Hoerauf, Achim; Hübner, Marc P

Oxfendazole mediates macrofilaricidal efficacy against the filarial nematode Litomosoides sigmodontis in vivo and inhibits Onchocerca spec. motility in vitro

奥芬达唑在体内介导对丝虫线虫 Litomosoides sigmodontis 的杀大丝虫作用,并在体外抑制盘尾丝虫的活力

Marc P Hübner, Coralie Martin, Sabine Specht, Marianne Koschel, Bettina Dubben, Stefan J Frohberger, Alexandra Ehrens, Martina Fendler, Dominique Struever, Edward Mitre, Nathaly Vallarino-Lhermitte, Suzanne Gokool, Sara Lustigman, Manfred Schneider, Simon Townson, Achim Hoerauf, Ivan Scandale

Discovery of ABBV-4083, a novel analog of Tylosin A that has potent anti-Wolbachia and anti-filarial activity

发现新型泰乐菌素A类似物ABBV-4083,该类似物具有强效的抗沃尔巴克氏体和抗丝虫活性。

von Geldern, Thomas W; Morton, Howard E; Clark, Rick F; Brown, Brian S; Johnston, Kelly L; Ford, Louise; Specht, Sabine; Carr, Robert A; Stolarik, Deanne F; Ma, Junli; Rieser, Matthew J; Struever, Dominique; Frohberger, Stefan J; Koschel, Marianne; Ehrens, Alexandra; Turner, Joseph D; Hübner, Marc P; Hoerauf, Achim; Taylor, Mark J; Ward, Stephen A; Marsh, Kennan; Kempf, Dale J

In vivo kinetics of Wolbachia depletion by ABBV-4083 in L. sigmodontis adult worms and microfilariae

ABBV-4083 对 L. sigmodontis 成虫和微丝蚴中沃尔巴克氏体耗竭的体内动力学

Hübner, Marc P; Koschel, Marianne; Struever, Dominique; Nikolov, Venelin; Frohberger, Stefan J; Ehrens, Alexandra; Fendler, Martina; Johannes, Iliana; von Geldern, Thomas W; Marsh, Kennan; Turner, Joseph D; Taylor, Mark J; Ward, Stephen A; Pfarr, Kenneth; Kempf, Dale J; Hoerauf, Achim