Identification and characterization of an atypical Gαs-biased β(2)AR agonist that fails to evoke airway smooth muscle cell tachyphylaxis
鉴定和表征一种非典型Gαs偏向性β(2)肾上腺素能受体激动剂,该激动剂无法诱发气道平滑肌细胞快速耐受性
期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2026668118
Kim, Donghwa; Tokmakova, Alina; Lujan, Lauren K; Strzelinski, Hannah R; Kim, Nicholas; Najari Beidokhti, Maliheh; Giulianotti, Marc A; Mafi, Amirhossein; Woo, Jung-A A; An, Steven S; Goddard, William A 3rd; Liggett, Stephen B