日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mutation-specific dual potentiators maximize rescue of CFTR gating mutants

突变特异性双重增强剂可最大限度地挽救 CFTR 门控突变体

Veit, Guido; Da Fonte, Dillon F; Avramescu, Radu G; Premchandar, Aiswarya; Bagdany, Miklos; Xu, Haijin; Bensinger, Dennis; Stubba, Daniel; Schmidt, Boris; Matouk, Elias; Lukacs, Gergely L

Virtual Screening Identifies Irreversible FMS-like Tyrosine Kinase 3 Inhibitors with Activity toward Resistance-Conferring Mutations

虚拟筛选可鉴定出具有抗药性突变活性的不可逆 FMS 样酪氨酸激酶 3 抑制剂

Dennis Bensinger, Daniel Stubba, Anjali Cremer, Vanessa Kohl, Theresa Waßmer, Johanna Stuckert, Victoria Engemann, Kimberly Stegmaier, Katja Schmitz, Boris Schmidt

Cell-Based Optimization of Covalent Reversible Ketoamide Inhibitors Bridging the Unprimed to the Primed Site of the Proteasome β5 Subunit

基于细胞的共价可逆酮酰胺抑制剂优化,该抑制剂连接蛋白酶体β5亚基的非激活位点和激活位点

Stubba, Daniel; Bensinger, Dennis; Steinbacher, Janika; Proskurjakov, Lilia; Salcedo Gómez, Álvaro; Schmidt, Uwe; Roth, Stefan; Schmitz, Katja; Schmidt, Boris