日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Guided Optimization of 4-Chloro-Pyrazolopyridine Analogs for Covalent PREP Inhibition

基于结构的4-氯吡唑并吡啶类似物优化用于共价PREP抑制

Thakur, Kalyani; Fucci, Ian; Pandian, Joshua; Suazo, Kiall F; Monteiro, Diana C F; Yoo, Euna

Potent β-lactam-based tyrosyl-DNA phosphodiesterase 1 inhibitors identified by a virtual screen.

通过虚拟筛选鉴定出强效β-内酰胺类酪氨酰-DNA磷酸二酯酶1抑制剂

Zhao Xue Zhi, Wang Wenjie, Suazo Kiall F, Al Mahmud Md Rasel, Agama Keli, Lountos George T, Andresson Thorkell, Pommier Yves, Burke Terrence R Jr

Hierarchical small molecule inhibition of MYST acetyltransferases

MYST乙酰转移酶的分级小分子抑制

Chen, Xuemin; Castroverde, Alexandra; Perez, Minervo; Holewinski, Ronald; Suazo, Kiall F; Karki, Rashmi; Andressen, Thorkell; Garcia, Benjamin A; Meier, Jordan L

Paralogue-Selective Degradation of the Lysine Acetyltransferase EP300

赖氨酸乙酰转移酶EP300的旁系同源选择性降解

Chen, Xuemin; Crawford, McKenna C; Xiong, Ying; Shaik, Anver Basha; Suazo, Kiall F; Bauer, Ludwig G; Penikalapati, Manini S; Williams, Joycelyn H; Huber, Kilian V M; Andressen, Thorkell; Swenson, Rolf E; Meier, Jordan L

Improved synthesis and application of an alkyne-functionalized isoprenoid analogue to study the prenylomes of motor neurons, astrocytes and their stem cell progenitors.

改进炔烃官能化异戊二烯类似物的合成和应用,以研究运动神经元、星形胶质细胞及其干细胞祖细胞的异戊二烯体

Suazo Kiall F, Mishra Vartika, Maity Sanjay, Auger Shelby A, Justyna Katarzyna, Petre Alexandru M, Ottoboni Linda, Ongaro Jessica, Corti Stefania P, Lotti Francesco, Przedborski Serge, Distefano Mark D

Discovery of a Tunable Heterocyclic Electrophile 4-Chloro-pyrazolopyridine That Defines a Unique Subset of Ligandable Cysteines

发现一种可调控的杂环亲电试剂 4-氯吡唑并吡啶,它定义了可配位半胱氨酸的一个独特子集

Kim, Hong-Rae; Byun, David P; Thakur, Kalyani; Ritchie, Jennifer; Xie, Yixin; Holewinski, Ronald; Suazo, Kiall F; Stevens, Mckayla; Liechty, Hope; Tagirasa, Ravichandra; Jing, Yihang; Andresson, Thorkell; Johnson, Steven M; Yoo, Euna

Orthogonal Enzyme-Substrate Design Strategy for Discovery of Human Protein Palmitoyltransferase Substrates

正交酶-底物设计策略在人类蛋白质棕榈酰转移酶底物发现中的应用

Puthenveetil, Robbins; Auger, Shelby A; Gómez-Navarro, Natalia; Rana, Mitra Shumsher; Das, Riki; Healy, Liam Brendan; Suazo, Kiall F; Shi, Zhen-Dan; Swenson, Rolf E; Distefano, Mark D; Banerjee, Anirban

A Not-So-Ancient Grease History: Click Chemistry and Protein Lipid Modifications

油脂的古老历史:点击化学与蛋白质脂质修饰

Suazo, Kiall F; Park, Keun-Young; Distefano, Mark D

Neuronal Protein Farnesylation Regulates Hippocampal Synaptic Plasticity and Cognitive Function

神经元蛋白法尼基化调节海马突触可塑性和认知功能

Qu, Wenhui; Suazo, Kiall F; Liu, Wenfeng; Cheng, Shaowu; Jeong, Angela; Hottman, David; Yuan, Li-Lian; Distefano, Mark D; Li, Ling

Splice switching an oncogenic ratio of SmgGDS isoforms as a strategy to diminish malignancy

剪接转换和SmgGDS亚型致癌比例作为降低恶性肿瘤的策略

Brandt, Anthony C; McNally, Lisa; Lorimer, Ellen L; Unger, Bethany; Koehn, Olivia J; Suazo, Kiall F; Rein, Lisa; Szabo, Aniko; Tsaih, Shirng-Wern; Distefano, Mark D; Flister, Michael J; Rigo, Frank; McNally, Mark T; Williams, Carol L