日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Transition-Metal-Catalyzed C–H/N–H Annulation Reactions between Imidazoles and Alkynes for the Synthesis of Fluorescent Benzimidazo[2,1‑a]Isoquinolines

过渡金属催化咪唑与炔烃的C–H/N–H环化反应合成荧光苯并咪唑并[2,1-a]异喹啉

Aishwarya, S; Torres, Gabriela C; Lopez-Saenz, Jose A; Gutierrez, Denisse A; Kumar, Sujeet; Madarakhandi, Ashok; Metikurki, Basavaraj; Teraiya, Nishith; Aguilera, Renato J; Karki, Subhas S; Dias, Gleiston G

Design, synthesis and anticancer evaluation of novel hydrazide-2-oxindole analogues as GSK-3β kinase inhibitors.

设计、合成和评价新型酰肼-2-吲哚酮类似物作为GSK-3β激酶抑制剂的抗癌活性

Madarakhandi Ashok, Kumar Sujeet, Teraiya Nishith, Schols Dominique, Vastrad Soujanya J, Shyamjith P, Choudhary Bibha, Rai Arzoo, Karki Subhas S

Does Ortho-Substitution Enhance Cytotoxic Potencies in a Series of 3,5-Bis(benzylidene)-4-piperidones?

邻位取代是否能增强一系列 3,5-双(亚苄基)-4-哌啶酮的细胞毒性?

Karki, Subhas S; Das, Umashankar; Balzarini, Jan; De Clercq, Erik; Sakagami, Hiroshi; Uesawa, Yoshihiro; Roayapalley, Praveen K; Dimmock, Jonathan R

A Coumarin-Imidazothiadiazole Derivative, SP11 Abrogates Tumor Growth by Targeting HSP90 and Its Client Proteins

香豆素-咪唑噻二唑衍生物 SP11 通过靶向 HSP90 及其客户蛋白来抑制肿瘤生长

Snehal Nirgude, Shahana M V, Febina Ravindran, Sujeet Kumar, Shivangi Sharma, Raghunandan Mahadeva, Anisha Mhatre, Subhas S Karki, Bibha Choudhary

Synthesis of Novel Pyrazole-Oxindole Conjugates with Cytotoxicity in Human Cancer Cells via Apoptosis

通过诱导细胞凋亡,合成对人癌细胞具有细胞毒性的新型吡唑-吲哚酮缀合物

Jain, Pravesh M; Gutierrez, Denisse A; Kumar, Sujeet; Aguilera, Renato J; Karki, Subhas S

Three novel piperidones exhibit tumor-selective cytotoxicity on leukemia cells via protein degradation and stress-mediated mechanisms

三种新型哌啶酮通过蛋白质降解和应激介导机制对白血病细胞表现出肿瘤选择性细胞毒性

Lisett Contreras, Stephanie Medina, Austre Y Schiaffino Bustamante, Edgar A Borrego, Carlos A Valenzuela, Umashankar Das, Subhas S Karki, Jonathan R Dimmock, Renato J Aguilera

Synthesis, Molecular Docking and Preliminary Antileukemic Activity of 4-Methoxybenzyl Derivatives Bearing Imidazo[2,1-b][1,3,4]thiadiazole

含咪唑并[2,1-b][1,3,4]噻二唑的4-甲氧基苄基衍生物的合成、分子对接及初步抗白血病活性

Choodamani, B; Cano Hernandez, Karla G; Kumar, Sujeet; Tony, Ann Maria; Schiaffino Bustamante, Austre Y; Aguilera, Renato J; Schols, Dominique; Gopi Mohan, C; Karki, Subhas S

ST09, A Novel Curcumin Derivative, Blocks Cell Migration by Inhibiting Matrix Metalloproteases in Breast Cancer Cells and Inhibits Tumor Progression in EAC Mouse Tumor Models

ST09 是一种新型姜黄素衍生物,可通过抑制乳腺癌细胞中的基质金属蛋白酶来阻止细胞迁移,并抑制 EAC 小鼠肿瘤模型中的肿瘤进展

Snehal Nirgude, Raghunandan Mahadeva, Jinsha Koroth, Sujeet Kumar, Kothanahally S Sharath Kumar, Vidya Gopalakrishnan, Subhas S S Karki, Bibha Choudhary

Effects of green synthesised silver nanoparticles (ST06-AgNPs) using curcumin derivative (ST06) on human cervical cancer cells (HeLa) in vitro and EAC tumor bearing mice models

利用姜黄素衍生物 (ST06) 绿色合成的银纳米粒子 (ST06-AgNPs) 对体外培养的人宫颈癌细胞 (HeLa) 和 EAC 荷瘤小鼠模型的影响

Murugesan, Kalaimathi; Koroth, Jinsha; Srinivasan, Padma Priya; Singh, Amrita; Mukundan, Sanjana; Karki, Subhas S; Choudhary, Bibha; Gupta, Chhitar M

Synthesis of thiocarbohydrazide and carbohydrazide derivatives as possible biologically active agents

硫代碳酰肼和碳酰肼衍生物的合成及其作为潜在生物活性剂的研究

Gangarapu, Kiran; Manda, Sarangapani; Jallapally, Anvesh; Thota, Sreekanth; Karki, Subhas S; Balzarini, Jan; De Clercq, Erik; Tokuda, Harukuni