日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site

通过靶向正位点的不同亚区来控制阿片受体功能选择性

Rajendra Uprety #, Tao Che #, Saheem A Zaidi #, Steven G Grinnell, Balázs R Varga, Abdelfattah Faouzi, Samuel T Slocum, Abdullah Allaoa, András Varadi, Melissa Nelson, Sarah M Bernhard, Elizaveta Kulko, Valerie Le Rouzic, Shainnel O Eans, Chloe A Simons, Amanda Hunkele, Joan Subrath, Ying Xian Pan, 

Mitragynine/Corynantheidine Pseudoindoxyls As Opioid Analgesics with Mu Agonism and Delta Antagonism, Which Do Not Recruit β-Arrestin-2

美沙酮/柯南西定伪吲哚作为具有 Mu 激动作用和 Delta 拮抗作用的阿片类镇痛药,不会募集 β-Arrestin-2

András Váradi, Gina F Marrone, Travis C Palmer, Ankita Narayan, Márton R Szabó, Valerie Le Rouzic, Steven G Grinnell, Joan J Subrath, Evelyn Warner, Sanjay Kalra, Amanda Hunkele, Jeremy Pagirsky, Shainnel O Eans, Jessica M Medina, Jin Xu, Ying-Xian Pan, Attila Borics, Gavril W Pasternak, Jay P McLau

Synthesis and characterization of a dual kappa-delta opioid receptor agonist analgesic blocking cocaine reward behavior

双 kappa-delta 阿片受体激动剂镇痛药的合成与表征及阻断可卡因奖励行为

András Váradi, Gina F Marrone, Shainnel O Eans, Michelle L Ganno, Joan J Subrath, Valerie Le Rouzic, Amanda Hunkele, Gavril W Pasternak, Jay P McLaughlin, Susruta Majumdar

Synthesis of Carfentanil Amide Opioids Using the Ugi Multicomponent Reaction

采用 Ugi 多组分反应合成卡芬太尼酰胺阿片类药物

András Váradi, Travis C Palmer, Nathan Haselton, Daniel Afonin, Joan J Subrath, Valerie Le Rouzic, Amanda Hunkele, Gavril W Pasternak, Gina F Marrone, Attila Borics, Susruta Majumdar

Three-component coupling approach for the synthesis of diverse heterocycles utilizing reactive nitrilium trapping

利用反应性腈正离子捕获的三组分偶联方法合成多种杂环化合物

Váradi, András; Palmer, Travis C; Notis, Paula R; Redel-Traub, Gabriel N; Afonin, Daniel; Subrath, Joan J; Pasternak, Gavril W; Hu, Chunhua; Sharma, Indrajeet; Majumdar, Susruta