日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Direct Selection of Functional De Novo Macrocycles for Activation of On-Cellulo Insulin Receptor

直接筛选功能性从头合成大环化合物以激活细胞内胰岛素受体

Kuo, Yun-Hsuan; Mihara, Emiko; Takagi, Junichi; Suga, Hiroaki

Ribosomal Synthesis of Topologically Defined Thioisoindole-Bridged Bicyclic Peptides

拓扑结构明确的硫代异吲哚桥联双环肽的核糖体合成

Zhang, Yue; Vinogradov, Alexander A; Sun, Yin; Suga, Hiroaki

A Nonviral Neo-Nucleocapsid for Cell-Specific RNA Delivery Developed by Pseudo-Cyclic Peptide Grafting and Directed Evolution

利用伪环肽嫁接和定向进化技术开发了一种用于细胞特异性RNA递送的非病毒新核衣壳

Kanayama, Daiki; Terasaka, Naohiro; Kato, Kazuki; Okazaki, Sae; Suga, Hiroaki

Discovery of Ultrapotent Heterodimeric Peptide Ligands Using Library-vs-Library RaPID Selections

利用文库对文库快速筛选发现超强异二聚肽配体

Ohno, Yuto; Vinogradov, Alexander A; Suga, Hiroaki

Discovery of Supra-Bivalent GSK3β Inhibitory Peptides Containing an ATP-Mimetic Amino Acid

发现含有ATP模拟氨基酸的超二价GSK3β抑制肽

Haslböck, Sara; Vinogradov, Alexander A; Okada, Chikako; Fujimura, Naoakusa; Aikawa, Haruo; Sengoku, Toru; Suga, Hiroaki

A reprogrammed genetic code consisting of 32 distinct amino acids

由32种不同氨基酸组成的重新编程的遗传密码

Katoh, Takayuki; Suga, Hiroaki

Engineering of tRNAPro1E2 anticodon stem enhances multiple/consecutive ribosomal incorporation of N-methyl-l-α-amino acids and d-α-amino acids

tRNAPro1E2反密码子茎的工程改造增强了N-甲基-L-α-氨基酸和D-α-氨基酸的多次/连续核糖体掺入

Hirashima, Ryoichi; Katoh, Takayuki; Suga, Hiroaki

The Alteromonas macleodii ribosome enables consecutive incorporation of bulky D-amino acids into peptides

麦克劳德氏交替单胞菌核糖体能够将体积较大的D-氨基酸连续掺入肽链中。

Katoh, Takayuki; Takada, Hiraku; Sigal, Maxwell; Suga, Hiroaki

De novo discovery of bicyclic cysteine-rich peptides targeting gasdermin D

从头发现靶向 gasdermin D 的富含半胱氨酸的双环肽

Li, Choi Yi; Sun, Yin; Vinogradov, Alexander A; Suga, Hiroaki

High-affinity, structure-validated and selective macrocyclic peptide tools for chemical biology studies of Huntingtin

用于亨廷顿蛋白化学生物学研究的高亲和力、结构验证和选择性大环肽工具

Fanti, Rebeka; Wolf, Esther; Ikenoue, Tatsuya; Deme, Justin C; Balakrishnan, Swati; Keith, Brandon A; Alteen, Matthew G; Chandrasekaran, Renu; Yadav, Manisha; Bhajiawala, Ritika; Ackloo, Suzanne; Feng, Jia; Pouladi, Mahmoud A; Edwards, Aled M; Wilson, Derek J; Lea, Susan M; Suga, Hiroaki; Harding, Rachel J