日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mitochondrial KMT9 methylates DLAT to control pyruvate dehydrogenase activity and prostate cancer growth

线粒体KMT9通过甲基化DLAT来控制丙酮酸脱氢酶活性和前列腺癌生长。

Jia, Yanhan; Wang, Sheng; Urban, Sylvia; Müller, Judith M; Sum, Manuela; Wang, Qing; Bauer, Helena; Schulte, Uwe; Rampelt, Heike; Pfanner, Nikolaus; Schüle, Katrin M; Imhof, Axel; Forné, Ignasi; Berlin, Christopher; Sigle, August; Gratzke, Christian; Greschik, Holger; Metzger, Eric; Schüle, Roland

Structure-Guided Design of a KMT9 Inhibitor Prodrug with Cellular Activity.

基于结构的KMT9抑制剂前药设计及其细胞活性

Wang Sheng, Barthes Nicolas P F, Urban Sylvia, Hazai Viktor I, Klein Sebastian O, Pappert Tabea, Kümmel Paul, Heller Nicolas, Bacher Johannes, Staudt Maximilian, Ruprecht Jan, Peng Ling, Sum Manuela, Berlin Christopher, Sarraf Daad, Regenass Pierre, Warstat Robin, Walz Johannes, Mishra Pankaj, Zhang Lin, Einsle Oliver, Günther Stefan, Breit Bernhard, Metzger Eric, Jung Manfred, Schüle Roland