日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

METTL16-mediated inhibition of MXD4 promotes leukemia through activation of the MYC-MAX axis.

METTL16 介导的 MXD4 抑制通过激活 MYC-MAX 轴促进白血病。

Bove Guglielmo, Babaei Mehrad, Bueno-Costa Alberto, Amin Sajid, Simonelli Nicla, Benedetti Rosaria, Dell'Aversana Carmela, Conte Mariarosaria, Montella Liliana, Summa Vincenzo, Brindisi Margherita, Del Sorbo Maria Rosaria, Crepaldi Marco, Favale Gregorio, Profitos-Peleja Nuria, Carafa Vincenzo, Roué Gaël, Ciardiello Fortunato, Capuano Annalisa, Stunnenberg Hendrik G, Megchelenbrink Wouter L, Nebbioso Angela, Esteller Manel, Altucci Lucia, Del Gaudio Nunzio

Sustainable Joullié-Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors.

可持续的 Joullié-Ugi 和连续流实施产生了新型的受卡托普利启发的广谱金属β-内酰胺酶抑制剂

Alfano Antonella Ilenia, Pelliccia Sveva, Barone Simona, Cutarella Luigi, Cancade Sacha Michèle Idriss, Baia Valerio, Cassese Emilia, Russomanno Pasquale, Messano Nicolò, Frank Denia, Weizel Lilia, Rotter Marco J, Brunst Steffen, Wichelhaus Thomas A, Proschak Ewgenij, Tedesco Daniele, Mori Mattia, Docquier Jean Denis, Summa Vincenzo, Brindisi Margherita

Fixed combination of palmitoylethanolamide and melatonin in preventive therapy of migraine: results from a randomized clinical trial

棕榈酰乙醇胺和褪黑素固定组合用于偏头痛预防治疗:一项随机临床试验的结果

Piccolo, Vincenzo; Marzocchi, Adua; Maisto, Maria; Summa, Vincenzo; Tenore, Gian Carlo; Amoresano, Angela

Integrating Surface Plasmon Resonance and Docking Analysis for Mechanistic Insights of Tryptase Inhibitors

整合表面等离子体共振和分子对接分析以深入了解类胰蛋白酶抑制剂的作用机制

Porta, Alessia; Manelfi, Candida; Talarico, Carmine; Beccari, Andrea Rosario; Brindisi, Margherita; Summa, Vincenzo; Iaconis, Daniela; Gobbi, Marco; Beeg, Marten

Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2.

硫醇反应性或氧化还原活性:修改重新定位筛选导致新的无效化流程,并鉴定出针对 SARS-CoV-2 木瓜蛋白酶样蛋白酶的真正非共价抑制剂

Kuzikov Maria, Morasso Stefano, Reinshagen Jeanette, Wolf Markus, Monaco Vittoria, Cozzolino Flora, Golič Grdadolnik Simona, Šket Primož, Plavec Janez, Iaconis Daniela, Summa Vincenzo, Corona Angela, Paulis Annalaura, Esposito Francesca, Tramontano Enzo, Monti Maria, Beccari Andrea R, Manelfi Candida, Windshügel Björn, Gribbon Philip, Storici Paola, Zaliani Andrea

Agri-Food Waste Recycling for Healthy Remedies: Biomedical Potential of Nutraceuticals from Unripe Tomatoes (Solanum lycopersicum L.)

利用农产品废弃物回收利用,开发健康疗法:未成熟番茄(Solanum lycopersicum L.)营养保健品的生物医学潜力

Piccolo, Vincenzo; Pastore, Arianna; Maisto, Maria; Keivani, Niloufar; Tenore, Gian Carlo; Stornaiuolo, Mariano; Summa, Vincenzo

Unveiling the modulation of Pseudomonas aeruginosa virulence and biofilm formation by selective histone deacetylase 6 inhibitors

揭示选择性组蛋白去乙酰化酶6抑制剂对铜绿假单胞菌毒力和生物膜形成的调控作用

Barone, Simona; Mateu, Baptiste; Turco, Luigia; Pelliccia, Sveva; Lembo, Francesca; Summa, Vincenzo; Buommino, Elisabetta; Brindisi, Margherita

A Rapid and Reliable Spectrofluorimetric Method to Measure the Urinary Lactulose/Mannitol Ratio for Dysbiosis Assessment

快速可靠的光谱荧光法测定尿乳果糖/甘露醇比值用于评估肠道菌群失调

Marino Cerrato, Lorenzo; Schiano, Elisabetta; Iannuzzo, Fortuna; Tenore, Gian Carlo; Summa, Vincenzo; Daglia, Maria; Novellino, Ettore; Stornaiuolo, Mariano

Natural Chalcones for the Management of Obesity Disease

天然查尔酮用于肥胖症的治疗

Maisto, Maria; Marzocchi, Adua; Keivani, Niloufar; Piccolo, Vincenzo; Summa, Vincenzo; Tenore, Gian Carlo

Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds

光流化学重排技术:生成具有药用价值化合物的强大工具

Alfano, Antonella Ilenia; Pelliccia, Sveva; Rossino, Giacomo; Chianese, Orazio; Summa, Vincenzo; Collina, Simona; Brindisi, Margherita