日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of SD-965 as a Potent, Selective, and Efficacious STAT3 PROTAC Degrader

发现 SD-965 是一种高效、选择性强且有效的 STAT3 PROTAC 降解剂

Wu, Dimin; Zhou, Haibin; Bai, Longchuan; Acharyya, Ranjan Kumar; Metwally, Hoda; McEachern, Donna; Wang, Mi; Tošović, Jelena; Rej, Rohan Kalyan; Wang, Meilin; Wen, Bo; Sun, Duxin; Wang, Shaomeng

Investigation of Renal Tissue Deposition of the Calcineurin Inhibitors Voclosporin, Cyclosporine and Tacrolimus Using MALDI-MSI Imaging

利用MALDI-MSI成像技术研究钙调磷酸酶抑制剂沃克洛孢素、环孢素和他克莫司在肾脏组织中的沉积

Zhou, Simon; Rajanayake, Krishani Kumari; He, Miao; Wen, Bo; Lkhagva, Ankhbayar; Yap, Ernie; Sun, Duxin; Cross, Jennifer; Engelke, Kory; Huizinga, Robert B

SARS-CoV-2 B Epitope-Guided Neoantigen NanoVaccines Enhance Tumor-Specific CD4/CD8 T Cell Immunity through B Cell Antigen Presentation

SARS-CoV-2 B 表位引导的新抗原纳米疫苗通过 B 细胞抗原呈递增强肿瘤特异性 CD4/CD8 T 细胞免疫。

Li, Chengyi; Ke, Fang; Mao, Shuai; Montemayor, Zera; Traore, Mohamed Dit Mady; Balsa, Alejandra Duran; Djibo, Mahamadou; Karekar, Neha; Hu, Hongxiang; Wen, Hanning; Gao, Wei; Sun, Duxin

IDOL Deficiency Inhibits Cholesterol-Rich Diet-Induced Atherosclerosis in Rabbits

IDOL缺乏抑制高胆固醇饮食诱导的兔动脉粥样硬化

Koike, Tomonari; Koike, Yui; Niimi, Manabu; Guo, Yanhong; Yang, Dongshan; Song, Jun; Xu, Jie; Tang, Xiangming; Ren, Zhuoying; Kong, Xiangbo; Liu, Hongyu; Zhao, Xiangjie; Zhu, Tianqing; Li, Ruiting; Wen, Bo; Sun, Duxin; Rom, Oren; Han, Renzhi; Fan, Jianglin; Garcia-Barrio, Minerva T; Zhang, Jifeng; Chen, Y Eugene

MD-4251: A First-in-Class Oral MDM2 Degrader Inducing Complete Tumor Regression with Single-Dose Administration

MD-4251:一种首创的口服MDM2降解剂,单次给药即可诱导肿瘤完全消退

Acharyya, Ranjan Kumar; Huang, Liyue; Aguilar, Angelo; Hu, Biao; Bai, Longchuan; Metwally, Hoda; McEachern, Donna; Jiang, Wei; Wang, Yu; Li, Qiuxia; Wen, Bo; Sun, Duxin; Wang, Shaomeng

An ingestible device for automated sampling and location tracing in gastrointestinal tract

一种用于胃肠道自动采样和定位追踪的可摄入式装置

Li, Tao; Felton, Jeremy; Lewis, Johnathan; Cheng, Qisen; Meredith, Ryan; Lu, Hsueh-Tsung; Benken, Alexander; Dutta, Partha P; Liao, Jinhui; Zhao, Xiangyu D; Matvekas, Aleksas; Baker, Jason; Hasler, William L; Babiskin, Andrew; Walenga, Ross; Fang, Lanyan Lucy; Lionberger, Robert; Pai, Manjunath P; Sun, Duxin; Gianchandani, Yogesh B

Examining the Impact of Diet-and-Exercise-Induced Weight Loss on Drug Metabolism and Gastric Emptying in Patients with Obesity

研究饮食和运动引起的体重减轻对肥胖患者药物代谢和胃排空的影响

Liu, Shuhan; Wang, Lu; Miller, Nicole; Waltje, Andrea; Abdelnabi, Mohamed; Zhu, Hao-Jie; Sun, Duxin; Rothberg, Amy E; Pai, Manjunath P

Adaptive nuclear GTP synthesis promotes glioblastoma treatment resistance and is a targetable vulnerability in patients

适应性核GTP合成促进胶质母细胞瘤的治疗耐药性,并且是患者治疗中一个可靶向的脆弱点。

Scott, Andrew J; Liang, Ningning; Al-Holou, Wajd N; Xu, Jie; O'Brien, Alexandra; Lin, Angelica; Pareek, Vidhi; Sha, Zhou; Zhao, Zitong; Yang, John Z; Yang, Annabel; Kothari, Ayesha U; Wilder-Romans, Kari; Wu, Zhe; Feng, Jiane; Korimerla, Navyateja; Elaimy, Ameer; Palavalasa, Sravya; Chen, Jiali; Wang, Lu; Zhang, Li; Andren, Anthony C; Sajjakulnukit, Peter; Marini, Bernard; Heth, Jason A; Morgan, Meredith A; Lawrence, Theodore S; Benkovic, Stephen J; Nagrath, Deepak; Chandrasekaran, Sriram; Qi, Nathan R; Sun, Duxin; Wen, Bo; Pai, Manjunath P; Clarke, Nathan; Suresh, Krithika; Umemura, Yoshie; Lyssiotis, Costas A; Zhou, Weihua; Wahl, Daniel R

Discovery of ERD-1233 as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader for the Treatment of ER+ Human Breast Cancer

发现 ERD-1233 是一种强效且口服有效的雌激素受体 PROTAC 降解剂,可用于治疗 ER+ 人类乳腺癌

Acharyya, Ranjan Kumar; Rej, Rohan Kalyan; Hu, Biao; Chen, Zhixiang; Wu, Dimin; Lu, Jianfeng; Metwally, Hoda; McEachern, Donna; Wang, Yu; Jiang, Wei; Bai, Longchuan; Tošović, Jelena; Gersch, Christina L; Xu, Guozhang; Zhang, Weihong; Wu, WenXue; Priestley, E Scott; Sui, Zhihua; Sarkari, Farzad; Wen, Bo; Sun, Duxin; Rae, James M; Wang, Shaomeng

Discovery of SD-436: A Potent, Highly Selective and Efficacious STAT3 PROTAC Degrader Capable of Achieving Complete and Long-Lasting Tumor Regression

SD-436 的发现:一种强效、高选择性和高效的 STAT3 PROTAC 降解剂,能够实现完全且持久的肿瘤消退

Xu, Renqi; Zhou, Haibin; Bai, Longchuan; McEachern, Donna; Wu, Dimin; Acharyya, Ranjan Kumar; Wang, Mi; Tošović, Jelena; Yang, Chao-Yie; Chinnaswamy, Krishnapriya; Meagher, Jennifer L; Stuckey, Jeanne A; Liu, Cai; Wang, Meilin; Wen, Bo; Sun, Duxin; Wang, Shaomeng