日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: FragGen: towards 3D geometry reliable fragment-based molecular generation

更正:FragGen:面向可靠的基于片段的三维几何分子生成

Zhang, Odin; Huang, Yufei; Chen, Shicheng; Yu, Mengyao; Zhang, Xujun; Lin, Haitao; Zeng, Yundian; Wang, Mingyang; Wu, Zhenxing; Zhao, Huifeng; Zhang, Zaixi; Hua, Chenqing; Kang, Yu; Cui, Sunliang; Pan, Peichen; Hsieh, Chang-Yu; Hou, Tingjun

A multicomponent reaction for modular assembly of indole-fused heterocycles

用于模块化组装吲哚稠合杂环的多组分反应

Li, Jiaming; Ni, Hao; Zhang, Weiwei; Lai, Zhencheng; Jin, Huimin; Zeng, Linwei; Cui, Sunliang

FragGen: towards 3D geometry reliable fragment-based molecular generation.

FragGen:面向可靠的基于片段的 3D 几何分子生成

Zhang Odin, Huang Yufei, Cheng Shichen, Yu Mengyao, Zhang Xujun, Lin Haitao, Zeng Yundian, Wang Mingyang, Wu Zhenxing, Zhao Huifeng, Zhang Zaixi, Hua Chenqing, Kang Yu, Cui Sunliang, Pan Peichen, Hsieh Chang-Yu, Hou Tingjun

Chemical Evolution and Biological Evaluation of Natural Products for Efficient Therapy of Acute Lung Injury

有效治疗急性肺损伤的天然产物的化学进化和生物学评价

Chengcheng Fan, Zeyi Zhang, Zhencheng Lai, Yanzi Yang, Jiaming Li, Lei Liu, Siyu Chen, Xueping Hu, Huajun Zhao, Sunliang Cui

Modular assembly of indole alkaloids enabled by multicomponent reaction

多组分反应实现吲哚生物碱的模块化组装

Li, Jiaming; Lai, Zhencheng; Zhang, Weiwei; Zeng, Linwei; Cui, Sunliang

Multicomponent double Mannich alkylamination involving C(sp(2))-H and benzylic C(sp(3))-H bonds

涉及 C(sp(2))-H 和苄基 C(sp(3))-H 键的多组分双曼尼希烷基胺化反应

Lai, Zhencheng; Wu, Rongkai; Li, Jiaming; Chen, Xing; Zeng, Linwei; Wang, Xi; Guo, Jingjing; Zhao, Zujin; Sajiki, Hironao; Cui, Sunliang

Discovery and Optimization of N-Acyl-6-sulfonamide-tetrahydroquinoline Derivatives as Novel Non-Steroidal Selective Glucocorticoid Receptor Modulators

发现和优化 N-酰基-6-磺酰胺-四氢喹啉衍生物作为新型非甾体选择性糖皮质激素受体调节剂

Dan Li, Xiaodong Bao, Jinping Pang, Xueping Hu, Longling Wang, Jiajia Wang, Zhaoxu Yang, Lei Xu, Siyu Wang, Qinjie Weng, Sunliang Cui, Tingjun Hou

Discovery of novel non-steroidal selective glucocorticoid receptor modulators by structure- and IGN-based virtual screening, structural optimization, and biological evaluation

通过基于结构和 IGN 的虚拟筛选、结构优化和生物学评价发现新型非甾体选择性糖皮质激素受体调节剂

Xueping Hu, Jinping Pang, Changwei Chen, Dejun Jiang, Chao Shen, Xin Chai, Liu Yang, Xujun Zhang, Lei Xu, Sunliang Cui, Tingjun Hou, Dan Li

Discovery of a small molecule inhibitor of cullin neddylation that triggers ER stress to induce autophagy

发现一种抑制 cullin neddylation 的小分子抑制剂,可引发内质网应激,从而诱导自噬

Yanan Li, Chaorong Wang, Tiantian Xu, Peichen Pan, Qing Yu, Lei Xu, Xiufang Xiong, Tingjun Hou, Sunliang Cui, Yi Sun

Subicular Caspase-1 Contributes to Pharmacoresistance in Temporal Lobe Epilepsy

下部 Caspase-1 导致颞叶癫痫产生药物耐药性

Cenglin Xu #, Shuo Zhang #, Yiwei Gong, Jiazhen Nao, Yujia Shen, Bei Tan, Shuheng Xu, Sunliang Cui, Yeping Ruan, Shuang Wang, Yi Wang, Zhong Chen