日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hybridization Approach Applied to Umbelliferon and Vanilloids toward New Inhibitors of Carbonic Anhydrases IX and XII with In Vitro Antiproliferative and Anti-inflammatory Activities

利用杂交方法筛选伞形酮和香草醛类化合物,以期获得具有体外抗增殖和抗炎活性的碳酸酐酶IX和XII新型抑制剂。

Melfi, Francesco; Mencarelli, Noemi; Carradori, Simone; Gallorini, Marialucia; Angeli, Andrea; Poli, Giulio; Cataldi, Amelia; D'Agostino, Ilaria; Di Credico, Andrea; Di Baldassarre, Angela; Tuccinardi, Tiziano; Supuran, Claudiu T

First-in-Class Dual PDGFR/Carbonic Anhydrase IX/XII Inhibitors: 6,7-Dimethoxyquinoline-Sulfonamides as Promising Antileukemic Agents

首创的双重PDGFR/碳酸酐酶IX/XII抑制剂:6,7-二甲氧基喹啉磺酰胺类药物作为有前景的抗白血病药物

Roshdy, Eslam; Řezníčková, Eva; Elbadawi, Mostafa M; Celik, Ismail; Giovannuzzi, Simone; Veselá, Denisa; Vojáčková, Veronika; Krňávková, Petra; Nocentini, Alessio; Supuran, Claudiu T; Kryštof, Vladimír; Eldehna, Wagdy M; Abe, Manabu

Hyaluronic Acid-Palmitate Nanoparticle Delivery of Carbonic Anhydrase Inhibitors Impairs Growth and Early Metabolism in Escherichia coli Through β- and γ-Carbonic Anhydrase-Associated Processes

透明质酸-棕榈酸酯纳米颗粒递送碳酸酐酶抑制剂通过β-和γ-碳酸酐酶相关过程损害大肠杆菌的生长和早期代谢

De Luca, Viviana; Verdoliva, Valentina; Supuran, Claudiu T; De Luca, Stefania; Capasso, Clemente

Investigation on N-Aryl-2-(4-sulfamoylphenyl)hydrazine-1-carbothioamide as Human Carbonic Anhydrases Inhibitors

对 N-芳基-2-(4-氨磺酰基苯基)肼-1-硫代甲酰胺作为人碳酸酐酶抑制剂的研究

Abdoli, Morteza; Angeli, Andrea; Bonardi, Alessandro; Gratteri, Paola; Jackevica, Ludmila; Sizovs, Antons; Supuran, Claudiu T; Žalubovskis, Raivis

Synthesis of Hydrazidoureidobenzensulfonamides Incorporating a Nicotinoyl Tail and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity

合成含烟酰尾的酰肼脲基苯磺酰胺及其对碳酸酐酶I、II、IX和XII的抑制活性

Deplano, Alberto; Moi, Davide; Vittorio, Serena; Angeli, Andrea; Supuran, Claudiu T; Onnis, Valentina

Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in Enterococcus faecium Septicemic Peritonitis Mouse Model While Sparing the Microbiome

细菌碳酸酐酶抑制剂 CAI0019 在粪肠球菌败血性腹膜炎小鼠模型中显示出疗效,同时不影响肠道菌群。

Abutaleb, Nader S; Holly, Katrina J; Metcalfe, Carolyn K; Abouelkhair, Ahmed A; Tharra, Prabhakara R; Shrinidhi, Annadka; Abdelsattar, Abdallah S; Burgo, Victoria; Melotte, Glory; Akin-Olabiyi, Tomi; Knoblauch, Sean; Ramaswamy, Ramanujam; Woodson, Che; Thirumalaikumar, Venkatesh P; Rodriguez, J Alejandra; Yeo, Franklin J; Snell, Olivia C; Nocentini, Alessio; Sundararajan, Anitha; Olson, Matthew R; Supuran, Claudiu T; Seleem, Mohamed N; Flaherty, Daniel P

Harnessing oligonucleotide architecture for potent multivalent inhibition of human carbonic anhydrases

利用寡核苷酸结构实现对人类碳酸酐酶的强效多价抑制

Abbass, Eslam M; Ladu, Federico; Mansot, Justine; Noël, Mathieu; Nocentini, Alessio; Sechi, Mario; Supuran, Claudiu T; Smietana, Michael; Winum, Jean-Yves

Chromones as Nonclassical Inhibitors of Carbonic Anhydrase IX and XII Isoforms: Probing Chromone-Based Derivatives

色酮类化合物作为碳酸酐酶IX和XII同工酶的非经典抑制剂:探索基于色酮的衍生物

Sequeira, Lisa; Distinto, Simona; Fernandes, Carlos; Sanna, Erica; Meleddu, Rita; Gaspari, Marco; Cottiglia, Filippo; Onali, Alessia; Angeli, Andrea; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T; Maccioni, Elias

Benzoxaboroles Are Inhibitors of the η-Class Carbonic Anhydrase From Plasmodium falciparum

苯并硼氧杂环己烷是恶性疟原虫η类碳酸酐酶的抑制剂

Bonardi, Alessandro; Wein, Sharon; Mustafa, Muhamad; Cerdan, Rachel; de Luca, Viviana; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T; Nocentini, Alessio; Winum, Jean-Yves

4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein

4-(5-氯-3-(3,4,5-三甲氧基苯甲酰基)-1H-吲哚-1-基)苯磺酰胺:一种新型多靶点药物,可选择性地靶向碳酸酐酶IX和XII、Wnt/β-catenin信号通路以及P-糖蛋白。

Puxeddu, Michela; Bordone, Rosa; Colla, Claudia; Rotili, Gabriele; Coluccia, Antonio; Sciò, Pietro; Cuřínová, Petra; Nocentini, Alessio; Supuran, Claudiu T; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Barba, Martina; Canettieri, Gianluca; Silvestri, Romano; La Regina, Giuseppe