Methyl substitution of a rexinoid agonist improves potency and reveals site of lipid toxicity
类雷昔洛韦激动剂的甲基取代可提高药效并揭示脂质毒性的部位
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm5004792
Venkatram R Atigadda, Gang Xia, Anil Desphande, LeeAnn J Boerma, Susan Lobo-Ruppert, Clinton J Grubbs, Craig D Smith, Wayne J Brouillette, Donald D Muccio