日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a small molecule modulator of the Kv1.1/Kvβ1 channel complex that reduces neuronal excitability and in vitro epileptiform activity

发现一种Kv1.1/Kvβ1通道复合物的小分子调节剂,该调节剂可降低神经元兴奋性和体外癫痫样活动。

Niespodziany, Isabelle; Mullier, Brice; André, Véronique Marie; Ghisdal, Philippe; Jnoff, Eric; Moreno-Delgado, David; Swinnen, Dominique; Sands, Zara; Wood, Martyn; Wolff, Christian

Synthesis and Evaluation of Bicyclic Hydroxypyridones as Inhibitors of Catechol O-Methyltransferase

双环羟基吡啶酮类化合物的合成及作为儿茶酚O-甲基转移酶抑制剂的评价

Ernst, Glen; Akuma, Daniel; Au, Vinh; Buchler, Ingrid P; Byers, Spencer; Carr, Gregory V; Defays, Sabine; de León, Pablo; Demaude, Thierry; DePasquale, Michael; Durieu, Véronique; Huang, Yifang; Jigorel, Emilie; Kimos, Martha; Kolobova, Anna; Montel, Florian; Moureau, Florence; Poslusney, Michael; Swinnen, Dominique; Vandergeten, Marie-Christine; Van Houtvin, Nathalie; Wei, Huijun; White, Noelle; Wood, Martyn; Barrow, James C

GLEPP1/protein-tyrosine phosphatase phi inhibitors block chemotaxis in vitro and in vivo and improve murine ulcerative colitis.

GLEPP1/蛋白酪氨酸磷酸酶phi抑制剂在体外和体内均可阻断趋化作用,并改善小鼠溃疡性结肠炎

Gobert Rosanna Pescini, van den Eijnden Monique, Szyndralewiez Cedric, Jorand-Lebrun Catherine, Swinnen Dominique, Chen Linfeng, Gillieron Corine, Pixley Fiona, Juillard Pierre, Gerber Patrick, Johnson-Léger Caroline, Halazy Serge, Camps Montserrat, Bombrun Agnes, Shipp Margaret, Vitte Pierre-Alain, Ardissone Vittoria, Ferrandi Chiara, Perrin Dominique, Rommel Christian, Hooft van Huijsduijnen Rob