日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oseltamivir aziridines are potent influenza neuraminidase inhibitors and imaging agents

奥司他韦氮丙啶类药物是强效的流感神经氨酸酶抑制剂和显像剂。

Vriends, Merijn B L; Moran, Elisha; Calvelo, Martín; Hansen, Thomas; Pickles, Isabelle B; Xin, Xincheng; Biezeno, Marieke; Armstrong, Zachary W B; Ferraz, Maria J; Li, Lei; Lilley, Alice; Harvey, Ruth; Filippov, Dmitri V; Liao, Qinghua; Schröder, Sybrin P; van der Marel, Gijsbert A; Artola, Marta; Aerts, Johannes M F G; Blaza, James N; Codée, Jeroen D C; Rovira, Carme; Overkleeft, Herman S; Davies, Gideon J

Selective labelling of GBA2 in cells with fluorescent β-d-arabinofuranosyl cyclitol aziridines

利用荧光标记的β-D-阿拉伯呋喃糖基环醇氮丙啶对细胞中的GBA2进行选择性标记

Su, Qin; Louwerse, Max; Lammers, Rob F; Maurits, Elmer; Janssen, Max; Boot, Rolf G; Borlandelli, Valentina; Offen, Wendy A; Linzel, Daniël; Schröder, Sybrin P; Davies, Gideon J; Overkleeft, Herman S; Artola, Marta; Aerts, Johannes M F G

Corrigendum: Xylose-Configured Cyclophellitols as Selective Inhibitors for Glucocerebrosidase

更正:木糖构型的环菲利托醇作为葡萄糖脑苷脂酶的选择性抑制剂

Su, Qin; Schröder, Sybrin P; Lelieveld, Lindsey T; Ferraz, Maria J; Verhoek, Marri; Boot, Rolf G; Overkleeft, Herman S; Aerts, Johannes M F G; Artola, Marta; Kuo, Chi-Lin

Development of Non-Hydrolysable Oligosaccharide Activity-Based Inactivators for Endoglycanases: A Case Study on α-1,6 Mannanases

基于非水解寡糖活性的内切糖苷酶灭活剂的开发:以α-1,6甘露聚糖酶为例

Schröder, Sybrin P; Offen, Wendy A; Males, Alexandra; Jin, Yi; de Boer, Casper; Enotarpi, Jacopo; Marino, Laura; van der Marel, Gijsbert A; Florea, Bogdan I; Codée, Jeroen D C; Overkleeft, Herman S; Davies, Gideon J

Correction: Glycosylated cyclophellitol-derived activity-based probes and inhibitors for cellulases

更正:糖基化环菲利醇衍生的纤维素酶活性探针和抑制剂

de Boer, Casper; McGregor, Nicholas G S; Peterse, Evert; Schröder, Sybrin P; Florea, Bogdan I; Jiang, Jianbing; Reijngoud, Jos; Ram, Arthur F J; van Wezel, Gilles P; van der Marel, Gijsbert A; Codée, Jeroen D C; Overkleeft, Herman S; Davies, Gideon J

Xylose-Configured Cyclophellitols as Selective Inhibitors for Glucocerebrosidase

木糖构型的环菲利托醇作为葡萄糖脑苷脂酶的选择性抑制剂

Su, Qin; Schröder, Sybrin P; Lelieveld, Lindsey T; Ferraz, Maria J; Verhoek, Marri; Boot, Rolf G; Overkleeft, Herman S; Aerts, Johannes M F G; Artola, Marta; Kuo, Chi-Lin

Dynamics of Ligand Binding to a Rigid Glycosidase*

配体与刚性糖苷酶结合的动力学*

Ben Bdira, Fredj; Waudby, Christopher A; Volkov, Alexander N; Schröder, Sybrin P; Ab, Eiso; Codée, Jeroen D C; Overkleeft, Hermen S; Aerts, Johannes M F G; van Ingen, Hugo; Ubbink, Marcellus

Glycosylated cyclophellitol-derived activity-based probes and inhibitors for cellulases

糖基化环菲利醇衍生的纤维素酶活性探针和抑制剂

de Boer, Casper; McGregor, Nicholas G S; Peterse, Evert; Schröder, Sybrin P; Florea, Bogdan I; Jiang, Jianbing; Reijngoud, Jos; Ram, Arthur F J; van Wezel, Gilles P; van der Marel, Gijsbert A; Codée, Jeroen D C; Overkleeft, Herman S; Davies, Gideon J

Dynamic and Functional Profiling of Xylan-Degrading Enzymes in Aspergillus Secretomes Using Activity-Based Probes

利用活性探针进行曲霉分泌组中木聚糖降解酶的动态和功能分析

Schröder, Sybrin P; de Boer, Casper; McGregor, Nicholas G S; Rowland, Rhianna J; Moroz, Olga; Blagova, Elena; Reijngoud, Jos; Arentshorst, Mark; Osborn, David; Morant, Marc D; Abbate, Eric; Stringer, Mary A; Krogh, Kristian B R M; Raich, Lluís; Rovira, Carme; Berrin, Jean-Guy; van Wezel, Gilles P; Ram, Arthur F J; Florea, Bogdan I; van der Marel, Gijsbert A; Codée, Jeroen D C; Wilson, Keith S; Wu, Liang; Davies, Gideon J; Overkleeft, Herman S

Direct Stereoselective Aziridination of Cyclohexenols with 3-Amino-2-(trifluoromethyl)quinazolin-4(3 H)-one in the Synthesis of Cyclitol Aziridine Glycosidase Inhibitors

环己烯醇与 3-氨基-2-(三氟甲基)喹唑啉-4(3H)-酮的直接立体选择性氮杂环丙烷化反应合成环己醇氮杂环丙烷糖苷酶抑制剂

Marta Artola, Shirley Wouters, Sybrin P Schröder, Casper de Boer, Yurong Chen, Rita Petracca, Adrianus M C H van den Nieuwendijk, Johannes M F G Aerts, Gijsbert A van der Marel, Jeroen D C Codée, Herman S Overkleeft