日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis, and anticancer activity of novel isocryptolepine 'aza' type acyl thiourea derivatives via combined experimental and computational approach

通过实验和计算相结合的方法设计、合成新型异隐花碱“氮杂”型酰基硫脲衍生物及其抗癌活性

Fayyaz, Ammara; Ejaz, Syeda Abida; Ahmed, Atteeque; Channar, Pervaiz Ali; Afzal, Saira; Ujan, Rabail; Saeed, Aamer; Bibi, Rifhat; Alsfouk, Bshra A; Abbas, Qamar; Sahito, Reshma; Bolte, Michael; Hökelek, Tuncer

Exploration of novel triazolo-thiadiazine hybrids of deferasirox as multi-target-directed anti-neuroinflammatory agents with structure-activity relationship (SAR): a new treatment opportunity for Alzheimer's disease.

探索新型三唑噻二嗪杂合物地拉罗司作为多靶点导向抗神经炎症药物的结构活性关系(SAR):阿尔茨海默病的新治疗机会

Shakir Syed Ahmed, Rashid Umer, Marryum, Fatima Nighat, Ejaz Syeda Abida, Fayyaz Ammara, Ullah Muhammad Zahid, Saeed Aamer, Khan Ajmal, Al Harrasi Ahmed, Mumtaz Amara

Synthesis and evaluation of thiazolyl coumarin drug conjugates as carbonic anhydrase isozyme inhibitors by using integrated invitro and insilico approaches

利用体外和计算机模拟相结合的方法合成和评价噻唑基香豆素药物偶联物作为碳酸酐酶同工酶抑制剂的活性

Ahmed, Atteeque; Kanwal, Romaisa; Channar, Pervaiz Ali; Alshahrani, Mohammad Y; Saeed, Aamer; Ejaz, Syeda Abida; Attaullah, Hafiz Muhammad; Bibi, Rifhat; Li, Chen

In silico-driven identification of potent CDK9 inhibitors through bioisosteric replacement and multi-stage virtual screening

利用生物等排体置换和多阶段虚拟筛选,通过计算机辅助方法鉴定高效 CDK9 抑制剂

Amorim, Juliana; Altamirano, Luis; de Souza, Denise Silva; Li, Chen; Ejaz, Syeda Abida; Arévalo, Juan Carpio

Exploration of newly synthesized azo-thiohydantoins as the potential alkaline phosphatase inhibitors via advanced biochemical characterization and molecular modeling approaches

通过先进的生化表征和分子建模方法探索新合成的偶氮硫代乙内酰脲作为潜在的碱性磷酸酶抑制剂

Hafiz Muhammad Attaullah, Syeda Abida Ejaz, Pervaiz Ali Channar, Aamer Saeed, Rabail Ujan, Seema Zargar, Sajid Ali Channar, Reshma Sahito, Tanveer A Wani, Qamar Abbas

Pharmacognostic Evaluation, Chemical Characterization, and Antibacterial Activity of Bassia indica (Wight) A.J. Scott

印度球孢菌(Bassia indica (Wight) AJ Scott)的药材学评价、化学表征及抗菌活性

Anjum, Fayyaz; Touqeer, Saad; Khan, Muhammad Younus; Jamil, QurratUlAin; Rida, Ayesha; Shirazi, Jafir Hussain; Ejaz, Syeda Abida; Attaullah, Hafiz Muhammad; Sarwar, Ghulam; Khan, Zaeem Hayat; Wazir, Muhammad Asif; Malik, Barizah; Aufy, Mohammed; Iqbal, Shahid Muhammad

Novel Bis-1,2,3-triazole-thiazolidinone hybrid as anticancer agents that induce apoptosis and molecular modeling study

新型双-1,2,3-三唑-噻唑烷酮杂合物作为诱导细胞凋亡的抗癌剂及其分子建模研究

Bimoussa, Abdoullah; Oubella, Ali; Alossaimi, Manal A; Aziz, Mubashir; Attaullah, Hafiz Muhammad; Ejaz, Syeda Abida; Morjani, Hamid; Auhmani, Aziz; Robert, Anthony; Riahi, Abdelkhalek; Riadi, Yassine; Ait Itto, Moulay Youssef

Identification of dimethyl 2,2'-((methylenebis(2-(2H-benzo[d][1,2,3]triazol-2-yl)-4-(2,4,4-trimethylpentan-2-yl)-6,1phenylene))bis(oxy))diacetate (TAJ4) as antagonist of NEK-Family: a future for potential drug discovery

二甲基 2,2'-((亚甲基双(2-(2H-苯并[d][1,2,3]三唑-2-基)-4-(2,4,4-三甲基戊-2-基)-6,1-亚苯基))双(氧))二乙酸酯 (TAJ4) 被鉴定为 NEK 家族拮抗剂:潜在药物发现的未来

Aziz, Mubashir; Ejaz, Syeda Abida; Channar, Pervaiz Ali; Alkhathami, Ali G; Qadri, Tahir; Hussain, Zahid; Hussaain, Mumtaz; Ujan, Rabail

Evaluation of Antiurolithiatic Effects of Moringa oleifera Lam. Leaves Extract: In-vitro, in-silico and in-vivo Approaches

辣木叶提取物抗尿路结石作用的评价:体外、计算机模拟和体内研究

Ali, Hina; Jabeen, Qaiser; Jamshed, Ayesha; Ejaz, Syeda Abida; Qadeer, Maria; Anwaar, Mariya; Rasheed, Hafiz Muhammad Farhan

Synthesis, DFT and molecular docking of novel (Z)-4-bromo-N-(4-butyl-3 (quinolin-3-yl)thiazol-2(3H)-ylidene)benzamide as elastase inhibitor

新型(Z)-4-溴-N-(4-丁基-3-(喹啉-3-基)噻唑-2(3H)-亚基)苯甲酰胺作为弹性蛋白酶抑制剂的合成、DFT计算和分子对接

Mustafa, Muhammad Naeem; Channar, Pervaiz Ali; Ejaz, Syeda Abida; Afzal, Saira; Aziz, Mubashir; Shamim, Tahira; Saeed, Aamer; Alsfouk, Aisha A; Ujan, Rabail; Abbas, Qamar; Hökelek, Tuncer