High Consistency of Structure-Based Design and X-Ray Crystallography: Design, Synthesis, Kinetic Evaluation and Crystallographic Binding Mode Determination of Biphenyl- N-acyl-β-d-Glucopyranosylamines as Glycogen Phosphorylase Inhibitors
基于结构的设计与X射线晶体学的高度一致性:联苯-N-酰基-β-d-葡萄吡喃胺作为糖原磷酸化酶抑制剂的设计、合成、动力学评估和晶体学结合模式测定
期刊:Molecules
影响因子:4.2
doi:10.3390/molecules24071322
Thomas Fischer, Symeon M Koulas, Anastasia S Tsagkarakou, Efthimios Kyriakis, George A Stravodimos, Vassiliki T Skamnaki, Panagiota G V Liggri, Spyros E Zographos, Rainer Riedl, Demetres D Leonidas1