日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

OICR-41103 as a chemical probe for the DCAF1 WD40 domain.

OICR-41103 作为 DCAF1 WD40 结构域的化学探针

Kimani Serah W, Noureldin Mahmoud, Wilson Brian, Hoffer Laurent, Green Stuart R, Szewczyk Magdalena M, González-Álvarez Héctor, Mohammed Mohammed, Chan Manuel, Krausser Chiara, Li Alice Shi Ming, Hajian Taraneh, Tucker Sarah, Joshi Dhananjay, Saraon Punit, Thériault Brigitte, Kim Ji Sup, Santhakumar Vijayaratnam, Loppnau Peter, Li Yanjun, Seitova Almagul, Dong Aiping, Kiyota Taira, Hammann Tobias, Gehrtz Paul, Patel Bhashant, Rathod Vaibhavi, Vala Anand, Rout Bhimsen, Jagodra Paras, Brown Peter J, Aman Ahmed, Ramnauth Jailall, Poda Gennady, Uehling David, Arrowsmith Cheryl H, Barsyte-Lovejoy Dalia, Marcellus Richard, Ackloo Suzanne, Mamai Ahmed, Al-Awar Rima, Halabelian Levon

Chemical tools for the Gid4 subunit of the human E3 ligase C-terminal to LisH (CTLH) degradation complex

用于研究人E3连接酶C端LisH (CTLH)降解复合物Gid4亚基的化学工具

Yazdi, Aliakbar Khalili; Perveen, Sumera; Dong, Cheng; Song, Xiaosheng; Dong, Aiping; Szewczyk, Magdalena M; Calabrese, Matthew F; Casimiro-Garcia, Agustin; Chakrapani, Subramanyam; Dowling, Matthew S; Ficici, Emel; Lee, Jisun; Montgomery, Justin I; O'Connell, Thomas N; Skrzypek, Grzegorz J; Tran, Tuan P; Troutman, Matthew D; Wang, Feng; Young, Jennifer A; Min, Jinrong; Barsyte-Lovejoy, Dalia; Brown, Peter J; Santhakumar, Vijayaratnam; Arrowsmith, Cheryl H; Vedadi, Masoud; Owen, Dafydd R

Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3).

发现蛋白质精氨酸甲基转移酶 3 (PRMT3) 的强效选择性变构抑制剂

Kaniskan H Ümit, Eram Mohammad S, Zhao Kehao, Szewczyk Magdalena M, Yang Xiaobao, Schmidt Keith, Luo Xiao, Xiao Sean, Dai Miao, He Feng, Zang Irene, Lin Ying, Li Fengling, Dobrovetsky Elena, Smil David, Min Sun-Joon, Lin-Jones Jennifer, Schapira Matthieu, Atadja Peter, Li En, Barsyte-Lovejoy Dalia, Arrowsmith Cheryl H, Brown Peter J, Liu Feng, Yu Zhengtian, Vedadi Masoud, Jin Jian

LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity

LLY-283 是一种强效且选择性的精氨酸甲基转移酶 5 (PRMT5) 抑制剂,具有抗肿瘤活性。

Bonday, Zahid Q; Cortez, Guillermo S; Grogan, Michael J; Antonysamy, Stephen; Weichert, Ken; Bocchinfuso, Wayne P; Li, Fengling; Kennedy, Steven; Li, Binghui; Mader, Mary M; Arrowsmith, Cheryl H; Brown, Peter J; Eram, Mohammad S; Szewczyk, Magdalena M; Barsyte-Lovejoy, Dalia; Vedadi, Masoud; Guccione, Ernesto; Campbell, Robert M

Allosteric inhibitors of plasma membrane Ca pumps: Invention and applications of caloxins

质膜钙泵的变构抑制剂:钙氧素的发明及应用

Pande, Jyoti; Szewczyk, Magdalena M; Grover, Ashok K

Ca2+-pumps and Na2+-Ca2+-exchangers in coronary artery endothelium versus smooth muscle

冠状动脉内皮细胞与平滑肌细胞中的Ca2+泵和Na2+-Ca2+交换器

Szewczyk, Magdalena M; Davis, Kim A; Samson, Sue E; Simpson, Fiona; Rangachari, Patangi K; Grover, Ashok K