(1aR,5aR)1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (MK-1903): a potent GPR109a agonist that lowers free fatty acids in humans
(1aR,5aR)1a,3,5,5a-四氢-1H-2,3-二氮杂-环丙基[a]戊二烯-4-羧酸 (MK-1903):一种有效的 GPR109a 激动剂,可降低人类体内的游离脂肪酸
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm2010964
P Douglas Boatman, Brett Lauring, Thomas O Schrader, Michelle Kasem, Benjamin R Johnson, Philip Skinner, Jae-Kyu Jung, Jerry Xu, Martin C Cherrier, Peter J Webb, Graeme Semple, Carleton R Sage, Jens Knudsen, Ruoping Chen, Wen-Lin Luo, Luzelena Caro, Josee Cote, Eseng Lai, John Wagner, Andrew K Tagga