Histone deacetylase activators: N-acetylthioureas serve as highly potent and isozyme selective activators for human histone deacetylase-8 on a fluorescent substrate
组蛋白去乙酰化酶激活剂:N-乙酰硫脲类化合物是高效且具有同工酶选择性的组蛋白去乙酰化酶-8激活剂,该激活剂作用于荧光底物上。
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2011.07.080
Singh, Raushan K; Mandal, Tanmay; Balsubramanian, Narayanaganesh; Viaene, Tajae; Leedahl, Travis; Sule, Nitesh; Cook, Gregory; Srivastava, D K