日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacokinetic-pharmacodynamic-efficacy modeling of the MDM2 inhibitor brigimadlin in glioblastoma patient-derived xenografts

MDM2抑制剂brigimadlin在胶质母细胞瘤患者来源异种移植模型中的药代动力学-药效学-疗效模型

Vaubel, Rachael A; Zhang, Wenjuan; Karbhari, Nishika; Oh, Ju-Hee; Waller, Katie L; Mladek, Ann; Jain, Sonia; Burgenske, Danielle M; Decker, Paul A; Kosel, Matt L; Hu, Zeng; Ott, Lauren L; Carlson, Brett L; Bakken, Katrina K; Pasa, Tugce; Sarkaria, Nicole R; Talele, Surabhi; Eckel-Passow, Jeanette E; Sini, Patrizia; Elmquist, William F; Sarkaria, Jann N

A PARP2 active site helix melts to permit DNA damage-induced enzymatic activation

PARP2活性位点螺旋解开,从而允许DNA损伤诱导的酶激活。

Emily S Smith-Pillet ,Ramya Billur ,Marie-France Langelier ,Tanaji T Talele ,John M Pascal ,Ben E Black

The impact of therapeutic radiation on drug distribution across the blood-brain barrier in normal mouse brain and orthotopic glioblastoma tumors

治疗性辐射对正常小鼠脑组织和原位胶质母细胞瘤中药物通过血脑屏障分布的影响

Zhang, Wenjuan; Grams, Michael P; Oberoi, Rajneet K; Oh, Ju-Hee; Decker, Paul A; Sio, Terence T; Talele, Surabhi; Wilson, Zachary C; Connors, Margaret A; Bakken, Katrina K; Carlson, Brett L; Ott, Lauren L; Burgenske, Danielle M; Tryggestad, Erik J; Eckel Passow, Jeanette E; Elmquist, William F; Sarkaria, Jann N

IL-1β blockade prevents cardiotoxicity and improves the efficacy of immune checkpoint blockers and chemotherapy against pancreatic cancer in mice with obesity

IL-1β阻断可预防心脏毒性,并提高肥胖小鼠胰腺癌中免疫检查点抑制剂和化疗的疗效。

Nilesh P Talele ,Heena Kumra ,Igor L Gomes-Santos ,William W Ho ,Patrik Andersson ,Marie Siwicki ,Peigen Huang ,Dan G Duda ,Mikael J Pittet ,Dai Fukumura ,Rakesh K Jain

Preclinical Modeling of Navtemadlin Pharmacokinetics, Pharmacodynamics, and Efficacy in IDH-Wild-type Glioblastoma.

Navtemadlin 在 IDH 野生型胶质母细胞瘤中的药代动力学、药效学和疗效的临床前模型

Vaubel Rachael A, Zhang Wenjuan, Oh Ju-Hee, Mladek Ann C, Pasa Tugce I, Gantchev Jennifer K, Waller Katie L, Baquer Gerard, Stopka Sylwia A, Regan Michael S, Hossain Md Amin, Decker Paul A, Kosel Matthew L, Gupta Shiv K, Jain Sonia, Sarkaria Paige P, Hu Zeng, Ott Lauren L, Carlson Brett L, Bakken Katie K, Talele Surabhi, Zhang Wenqiu, Ligon Keith L, Lee Eudocia Q, Eckel Passow Jeanette E, Burgenske Danielle M, Agar Nathalie Y R, Elmquist William F, Sarkaria Jann N

Cell cycle regulation has shaped replication origins in budding yeast

细胞周期调控塑造了出芽酵母的复制起点。

Lim, Chew Theng; Miller, Thomas C R; Tan, Kang Wei; Talele, Saurabh; Early, Anne; East, Philip; Sánchez, Humberto; Dekker, Nynke H; Costa, Alessandro; Diffley, John F X

Structure-activity relationship studies on 2-thienylidene substituted 3-oxo-2,3-dihydrobenzofuran-7-carboxamides as poly (ADP-ribose) polymerase inhibitors

2-噻吩亚甲基取代的3-氧代-2,3-二氢苯并呋喃-7-甲酰胺作为聚(ADP-核糖)聚合酶抑制剂的构效关系研究

Salami, Abosede; Adiele, Ugochi; Coate, Griffin; Diolaiti, Morgan; Chen, Huadong; Lu, Junhao; Ashworth, Alan; Patil, Manisha; Fleishman, Joshua S; Ramaraju, Andhavaram; Patel, Akanksha; Patel, Himaxi; Patel, Ketankumar; Murakami, Megumi; Ambudkar, Suresh V; Talele, Tanaji T

Discovery of a Novel [6-6-5-5-6] Pentacyclic Tetrahydrocyclopentaphthalazinone as a Promising PARP Inhibitor Scaffold

发现一种新型[6-6-5-5-6]五环四氢环戊酞嗪酮作为有前景的PARP抑制剂骨架

Doruk, Yagmur U; Diolaiti, Morgan E; Ashworth, Alan; Talele, Tanaji T

Highly Sensitive Multiplexed Detection of Brain‐Derived Tau and Phosphorylated Tau Proteoforms with the NULISA Technology

利用NULISA技术对脑源性tau蛋白和磷酸化tau蛋白进行高灵敏度多重检测

Wang, Yi-Jun; Patel, Bhargav A; Anreddy, Nagaraju; Zhang, Yun-Kai; Zhang, Guan-Nan; Alqahtani, Saeed; Singh, Satyakam; Shukla, Suneet; Kaddoumi, Amal; Ambudkar, Suresh V; Talele, Tanaji T; Chen, Zhe-Sheng; Ma, Xiao‐Jun; Iyengar, Shweta; Deshmukh, Shalaka; Comandor, Roopa; Wang, Li; Kim, Sean; Xu, Xiaomei; Feng, Wei; Qiu, Xiaolei; Zhang, Bingqing; Luo, Yuling

Voice-based user interface for hands-free data entry and automation at workplaces

用于工作场所免提数据输入和自动化的语音用户界面

Harihar, Daiwiik; Shrivastava, Vedansh; Talele, Pratvina; Jahagirdar, Aditi