日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dyr726, a brain-penetrant inhibitor of PI3Kα, Type III receptor tyrosine kinases, and WNT signaling.

Dyr726 是一种可穿透血脑屏障的 PI3Kα、III 型受体酪氨酸激酶和 WNT 信号通路抑制剂

Tandon Vasudha, Fistrovich Alessandra, Nogales Joaquina, Ferro Febe, Rokey Samantha N, Cabel Carly, Miller Amy Dunne, Yagel Mary, Duncan Christina, Atmasidha Aditi, Sharma Ira, Wilms Gerrit, Williams Karin, Elliott Richard, Chavez Timothy, Shaw Yeng, McMahon Aidan, Ginn Sean, Basantes L Emilia, Bedard Nathan, Gokhale Vijay, Ellis Nathan, Prescott Alan R, Smith Stuart J, Rahman Ruman, Becker Walter, Read Kevin D, Chalmers Anthony J, Carragher Neil, Masson Glenn R, Montfort William, Thorne Curtis, Hulme Christopher, Banerjee Sourav

Synthesis of N-(4-chlorophenyl) substituted pyrano[2,3-c]pyrazoles enabling PKBβ/AKT2 inhibitory and in vitro anti-glioma activity.

合成 N-(4-氯苯基)取代的吡喃并[2,3-c]吡唑,使其具有 PKBβ/AKT2 抑制活性和体外抗胶质瘤活性

Vala Ruturajsinh M, Tandon Vasudha, Nicely Lynden G, Guo Luxia, Gu Yanlong, Banerjee Sourav, Patel Hitendra M

Glasgow Neuro Society 2021 Conference Proceedings

2021年格拉斯哥神经学会会议论文集

Ashraf, Mohammad; Ismahel, Hassan; Lub, Sytske; Middleton, Eilidh; Chaudhary, Attika; Gardee, Ameerah; Salloum, Laulwa Al; Szilagyi-Nagy, Eva; Wales, Rachel; Omar, Samia; Baird, Tracey Anne; O'Kane, Roddy; Holden, John; Abdelsadg, Mohamed; Burr, Pierce; Decruz, Antony Ben; Badran, Khaled; Amato-Watkins, Anthony; Alakandy, Likhith; Boardman, Rosie; Nicely, Lynden; Tandon, Vasudha; Banerjee, Sourav; Keenlyside, Andrew; Hughes, Mark; Ho, Jen Wae; Sieradzki, Jake; Phan, Elizabeth Phuong My; MacDougall, Niall John James; Bashir, Aneesah Bashir Binti Azad; Hutton, Dana L; Doley, Alexander S F; Oochit, Krishna K; Kontorinis, Georgios; Wong, Yun Yang

Emerging roles of DYRK2 in cancer

DYRK2在癌症中的新兴作用

Tandon, Vasudha; de la Vega, Laureano; Banerjee, Sourav

Inhibition of dual-specificity tyrosine phosphorylation-regulated kinase 2 perturbs 26S proteasome-addicted neoplastic progression

双特异性酪氨酸磷酸化调节激酶2的抑制会扰乱26S蛋白酶体依赖的肿瘤进展。

Banerjee, Sourav; Wei, Tiantian; Wang, Jue; Lee, Jenna J; Gutierrez, Haydee L; Chapman, Owen; Wiley, Sandra E; Mayfield, Joshua E; Tandon, Vasudha; Juarez, Edwin F; Chavez, Lukas; Liang, Ruqi; Sah, Robert L; Costello, Caitlin; Mesirov, Jill P; de la Vega, Laureano; Cooper, Kimberly L; Dixon, Jack E; Xiao, Junyu; Lei, Xiaoguang