日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Non-covalent Ligand Reveals Biased Agonism of the TRPA1 Ion Channel

非共价配体揭示 TRPA1 离子通道的偏向激动作用

Chang Liu, Rebecca Reese, Simon Vu, Lionel Rougé, Shannon D Shields, Satoko Kakiuchi-Kiyota, Huifen Chen, Kevin Johnson, Yu Patrick Shi, Tania Chernov-Rogan, Demi Maria Zabala Greiner, Pawan Bir Kohli, David Hackos, Bobby Brillantes, Christine Tam, Tianbo Li, Jianyong Wang, Brian Safina, Steve Magnu

A TRPA1 inhibitor suppresses neurogenic inflammation and airway contraction for asthma treatment

TRPA1 抑制剂可抑制神经源性炎症和气道收缩,用于治疗哮喘

Alessia Balestrini, Victory Joseph, Michelle Dourado, Rebecca M Reese, Shannon D Shields, Lionel Rougé, Daniel D Bravo, Tania Chernov-Rogan, Cary D Austin, Huifen Chen, Lan Wang, Elisia Villemure, Daniel G M Shore, Vishal A Verma, Baihua Hu, Yong Chen, Laurie Leong, Chris Bjornson, Kathy Hötzel, Alv

Mechanism-specific assay design facilitates the discovery of Nav1.7-selective inhibitors

机制特异性检测设计有助于发现 Nav1.7 选择性抑制剂

Tania Chernov-Rogan, Tianbo Li, Gang Lu, Henry Verschoof, Kuldip Khakh, Steven W Jones, Maureen H Beresini, Chang Liu, Daniel F Ortwine, Steven J McKerrall, David H Hackos, Daniel Sutherlin, Charles J Cohen, Jun Chen

High-throughput electrophysiological assays for voltage gated ion channels using SyncroPatch 768PE

使用 SyncroPatch 768PE 对电压门控离子通道进行高通量电生理检测

Tianbo Li, Gang Lu, Eugene Y Chiang, Tania Chernov-Rogan, Jane L Grogan, Jun Chen

Antitumor activity of the glutaminase inhibitor CB-839 in triple-negative breast cancer

谷氨酰胺酶抑制剂 CB-839 对三阴性乳腺癌的抗肿瘤活性

Matt I Gross, Susan D Demo, Jennifer B Dennison, Lijing Chen, Tania Chernov-Rogan, Bindu Goyal, Julie R Janes, Guy J Laidig, Evan R Lewis, Jim Li, Andrew L Mackinnon, Francesco Parlati, Mirna L M Rodriguez, Peter J Shwonek, Eric B Sjogren, Timothy F Stanton, Taotao Wang, Jinfu Yang, Frances Zhao, Ma