日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mapping the Subtype-Specific PARP1 ADP-ribosylated Proteome in Breast Cancer Cells.

绘制乳腺癌细胞中亚型特异性 PARP1 ADP 核糖基化蛋白质组图谱。

Koul Sneh, Kwon Minjung, Tapadar Poulami, Dai Yangyang, Nandu Tulip, Huang Dan, Camacho Cristel V, Kraus W Lee

Small-molecule disruption of androgen receptor-dependent chromatin clusters

小分子对雄激素受体依赖性染色质簇的破坏作用

Kohrt, Sarah E; Novak, Emily J; Tapadar, Subhashish; Wu, Bocheng; Strope, Jonathan; Asante, Yaw; Kim, Hyunmin; Chang, Matthew S; Gurdak, Douglas; Khalil, Athar; Rood, Michael; Raftery, Eric; Stavreva, Diana; Nguyen, Holly M; Brown, Lisha G; Ramser, Maddy; Peer, Cody; Meyers, Warren M; Aboreden, Nicholas; Chakravortee, Maharshi; Sallari, Richard; Nelson, Peter S; Kelly, Kathleen K; Graham, Thomas G W; Darzacq, Xavier; Figg, William D; Oyelere, Adegboyega K; Corey, Eva; Adelaiye-Ogala, Remi; Gryder, Berkley E

A Novel Liver Cancer-Selective Histone Deacetylase Inhibitor Is Effective against Hepatocellular Carcinoma and Induces Durable Responses with Immunotherapy

一种新型肝癌选择性组蛋白去乙酰化酶抑制剂对肝细胞癌有效,并能诱导持久的免疫治疗反应。

Wu, Bocheng; Tapadar, Subhasish; Ruan, Zhiping; Sun, Carrie Q; Arnold, Rebecca S; Johnston, Alexis; Olugbami, Jeremiah O; Arunsi, Uche; Gaul, David A; Petros, John A; Kobayashi, Tatsuya; Duda, Dan G; Oyelere, Adegboyega K

Development and validation of a sensitive LC-MS/MS assay of GT-14, a novel Gα(i)2 inhibitor, in rat plasma, and its application in pharmacokinetic study

建立并验证了一种灵敏的液相色谱-串联质谱(LC-MS/MS)检测方法,用于测定大鼠血浆中新型Gα(i)2抑制剂GT-14的浓度,并将其应用于药代动力学研究。

Sarkar, Mahua; Ma, Jing; Tapadar, Subhasish; Caggia, Silvia; Oyelere, Adegboyega K; Khan, Shafiq A; Xie, Huan

Antiandrogen-Equipped Histone Deacetylase Inhibitors Selectively Inhibit Androgen Receptor (AR) and AR-Splice Variant (AR-SV) in Castration-Resistant Prostate Cancer (CRPC)

抗雄激素组蛋白去乙酰化酶抑制剂选择性抑制去势抵抗性前列腺癌 (CRPC) 中的雄激素受体 (AR) 和 AR 剪接变体 (AR-SV)

Balaji Chandrasekaran, Subhasish Tapadar, Bocheng Wu, Uttara Saran, Ashish Tyagi, Alexis Johnston, David A Gaul, Adegboyega K Oyelere, Chendil Damodaran

A machine learning-based approach to determine infection status in recipients of BBV152 (Covaxin) whole-virion inactivated SARS-CoV-2 vaccine for serological surveys

一种基于机器学习的方法,用于确定 BBV152(Covaxin)全病毒灭活 SARS-CoV-2 疫苗接种者的感染状态,以进行血清学调查

Singh, Prateek; Ujjainiya, Rajat; Prakash, Satyartha; Naushin, Salwa; Sardana, Viren; Bhatheja, Nitin; Singh, Ajay Pratap; Barman, Joydeb; Kumar, Kartik; Gayali, Saurabh; Khan, Raju; Rawat, Birendra Singh; Tallapaka, Karthik Bharadwaj; Anumalla, Mahesh; Lahiri, Amit; Kar, Susanta; Bhosale, Vivek; Srivastava, Mrigank; Mugale, Madhav Nilakanth; Pandey, C P; Khan, Shaziya; Katiyar, Shivani; Raj, Desh; Ishteyaque, Sharmeen; Khanka, Sonu; Rani, Ankita; Promila; Sharma, Jyotsna; Seth, Anuradha; Dutta, Mukul; Saurabh, Nishant; Veerapandian, Murugan; Venkatachalam, Ganesh; Bansal, Deepak; Gupta, Dinesh; Halami, Prakash M; Peddha, Muthukumar Serva; Veeranna, Ravindra P; Pal, Anirban; Singh, Ranvijay Kumar; Anandasadagopan, Suresh Kumar; Karuppanan, Parimala; Rahman, Syed Nasar; Selvakumar, Gopika; Venkatesan, Subramanian; Karmakar, Malay Kumar; Sardana, Harish Kumar; Kothari, Anamika; Parihar, Devendra Singh; Thakur, Anupma; Saifi, Anas; Gupta, Naman; Singh, Yogita; Reddu, Ritu; Gautam, Rizul; Mishra, Anuj; Mishra, Avinash; Gogeri, Iranna; Rayasam, Geethavani; Padwad, Yogendra; Patial, Vikram; Hallan, Vipin; Singh, Damanpreet; Tirpude, Narendra; Chakrabarti, Partha; Maity, Sujay Krishna; Ganguly, Dipyaman; Sistla, Ramakrishna; Balthu, Narender Kumar; A, Kiran Kumar; Ranjith, Siva; Kumar, B Vijay; Jamwal, Piyush Singh; Wali, Anshu; Ahmed, Sajad; Chouhan, Rekha; Gandhi, Sumit G; Sharma, Nancy; Rai, Garima; Irshad, Faisal; Jamwal, Vijay Lakshmi; Paddar, Masroor Ahmad; Khan, Sameer Ullah; Malik, Fayaz; Ghosh, Debashish; Thakkar, Ghanshyam; Barik, S K; Tripathi, Prabhanshu; Satija, Yatendra Kumar; Mohanty, Sneha; Khan, Md Tauseef; Subudhi, Umakanta; Sen, Pradip; Kumar, Rashmi; Bhardwaj, Anshu; Gupta, Pawan; Sharma, Deepak; Tuli, Amit; Ray Chaudhuri, Saumya; Krishnamurthi, Srinivasan; Prakash, L; Rao, Ch V; Singh, B N; Chaurasiya, Arvindkumar; Chaurasiyar, Meera; Bhadange, Mayuri; Likhitkar, Bhagyashree; Mohite, Sharada; Patil, Yogita; Kulkarni, Mahesh; Joshi, Rakesh; Pandya, Vaibhav; Mahajan, Sachin; Patil, Amita; Samson, Rachel; Vare, Tejas; Dharne, Mahesh; Giri, Ashok; Mahajan, Sachin; Paranjape, Shilpa; Sastry, G Narahari; Kalita, Jatin; Phukan, Tridip; Manna, Prasenjit; Romi, Wahengbam; Bharali, Pankaj; Ozah, Dibyajyoti; Sahu, Ravi Kumar; Dutta, Prachurjya; Singh, Moirangthem Goutam; Gogoi, Gayatri; Tapadar, Yasmin Begam; Babu, Elapavalooru Vssk; Sukumaran, Rajeev K; Nair, Aishwarya R; Puthiyamadam, Anoop; Valappil, Prajeesh Kooloth; Pillai Prasannakumari, Adrash Velayudhan; Chodankar, Kalpana; Damare, Samir; Agrawal, Ved Varun; Chaudhary, Kumardeep; Agrawal, Anurag; Sengupta, Shantanu; Dash, Debasis

Presence of Bromotyrosine Alkaloids in Marine Sponges Is Independent of Metabolomic and Microbiome Architectures

海洋海绵中溴酪氨酸生物碱的存在与代谢组和微生物组结构无关

Mohanty, Ipsita; Tapadar, Subhasish; Moore, Samuel G; Biggs, Jason S; Freeman, Christopher J; Gaul, David A; Garg, Neha; Agarwal, Vinayak

TBK1 regulates regeneration of pancreatic β-cells

TBK1 调节胰腺 β 细胞的再生

Yun-Fang Jia, Subbiah Jeeva, Jin Xu, Carrie Jo Heppelmann, Jin Sung Jang, Michael Q Slama, Subhasish Tapadar, Adegboyega K Oyelere, Sang-Moo Kang, Aleksey V Matveyenko, Quinn P Peterson, Chong Hyun Shin

Small Molecule Inhibitors Targeting Gαi2 Protein Attenuate Migration of Cancer Cells

针对 Gαi2 蛋白的小分子抑制剂可减弱癌细胞的迁移

Silvia Caggia, Subhasish Tapadar, Bocheng Wu, Smrruthi V Venugopal, Autumn S Garrett, Aditi Kumar, Janae S Stiffend, John S Davis, Adegboyega K Oyelere, Shafiq A Khan

Liver-Targeting Class I Selective Histone Deacetylase Inhibitors Potently Suppress Hepatocellular Tumor Growth as Standalone Agents

以肝脏为靶点的 I 类选择性组蛋白去乙酰化酶抑制剂作为独立药物可有效抑制肝细胞肿瘤生长

Subhasish Tapadar, Shaghayegh Fathi, Bocheng Wu, Carrie Q Sun, Idris Raji, Samuel G Moore, Rebecca S Arnold, David A Gaul, John A Petros, Adegboyega K Oyelere