日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rational design of phenyl 2,4,5-trichlorobenzenesulfonate based thiosemicarbazones as α-glucosidase and α-amylase inhibitors: integrating enzymatic evaluation and molecular modeling

基于苯基2,4,5-三氯苯磺酸酯的硫代氨基脲类化合物作为α-葡萄糖苷酶和α-淀粉酶抑制剂的合理设计:酶学评价与分子建模的整合

Noreen, Faiqa; Zaki, Magdi E A; Sadeghian, Nastaran; Tokali, Feyzi Sinan; Taslimi, Parham; Alharthy, Rima D; Şenol, Halil; Zhao, Xianliang; Çakır, Furkan; Gomha, Sobhi M; Shafiq, Zahid

Synthesis, multi-target evaluation and DFT analysis of 6-hydroxychromone derived hydrazones with carbonic anhydrase I-II/acetylcholinesterase inhibition and antioxidant activity

6-羟基色酮衍生的腙类化合物的合成、多靶点评价及DFT分析及其碳酸酐酶I-II/乙酰胆碱酯酶抑制活性和抗氧化活性

Zareen, Wajeeha; Ahmed, Nadeem; Tokali, Feyzi Sinan; Islam, Talha; Al-Rashida, Mariya; Senol, Ayşe Merve; Ulucay, Orhan; Tawfeek, Ahmed Mohamed; Taslimi, Parham; Shafiq, Zahid; Islam, Mohammad Shahidul

Synthesis and biological evaluation of 6-hydroxychromone based thiosemicarbazones as potential antidiabetic and antioxidant agents

6-羟基色酮基硫代氨基脲类化合物的合成及生物学评价:作为潜在的抗糖尿病和抗氧化剂

Zareen, Wajeeha; Ahmed, Nadeem; Siddique, Farhan; Taslimi, Parham; Khan, Muhammad Ali; Islam, Talha; Ismail, Mostafa A; Al-Rashida, Mariya; Zaki, Magdi E A; Gomha, Sobhi M; Alharthy, Rima D; Shafiq, Zahid

Synthesis, Biological Evaluation, and In Silico Characterization of Novel Imidazothiadiazole-Chalcone Hybrids as Multi-Target Enzyme Inhibitors.

新型咪唑并噻二唑-查尔酮杂合物作为多靶点酶抑制剂的合成、生物学评价和计算机表征

Alici Hakan, Topuz Senol, Demir Kadir, Taslimi Parham, Tahtaci Hakan

Synthesis, antidiabetic evaluation, and computational modeling of 3-acetyl-8-ethoxy coumarin derived hydrazones and thiosemicarbazones

3-乙酰基-8-乙氧基香豆素衍生的腙和硫代氨基脲的合成、抗糖尿病评价及计算建模

Zareen, Wajeeha; Ahmed, Nadeem; Khan, Ali Muhammad; Mali, Suraj N; Sadeghian, Nastaran; Aldawsari, Naflaa A; Taslimi, Parham; Alanazi, Abdullah K; Tahir, Muhammad; Tasleem, Mussarat; Shafiq, Zahid

Synthesis and Computational Evaluation of N‑Acetyl-Derived Schiff Bases Incorporating 1,2,4-Triazoles for Dual Inhibition of Prostate Cancer Cells and Carbonic Anhydrases

合成及计算评价含1,2,4-三唑的N-乙酰基衍生的席夫碱对前列腺癌细胞和碳酸酐酶的双重抑制作用

Medetalibeyoğlu, Hilal; Aytatlı, Abdulmelik; Manap, Sevda; Atalay, Abdurrahman; Ortaakarsu, Ahmet Buğra; Tüzün, Burak; Taslimi, Parham; Gürsoy-Kol, Özlem; Karataş, Ömer Faruk; Yüksek, Haydar

Introduction of new quinolone-2-thio-acetamide-propane hydrazide-benzimidazole derivatives as new α-glucosidase and α-amylase inhibitors

新型喹诺酮-2-硫代乙酰胺-丙烷酰肼-苯并咪唑衍生物作为新型α-葡萄糖苷酶和α-淀粉酶抑制剂的引入

Nikfar, Parisa; Karimian, Somaye; Safapoor, Sajedeh; Noori, Milad; Dastyafteh, Navid; Ghafouri, Seyedeh Niloufar; Mohammadi-Khanaposhtani, Maryam; Larijani, Bagher; Taslimi, Parham; Mahdavi, Mohammad

Synthesis, antiproliferative activity targeting lung cancer and in silico studies of hydroxypiperidine substituted thiosemicarbazones

羟基哌啶取代的硫代氨基脲的合成、针对肺癌的抗增殖活性及计算机模拟研究

Aftab, Hina; Islam, Muhammad; Şenol, Halil; Batool, Zahra; Ateşoğlu, Şeyma; Çakır, Furkan; Akbaş, Fahri; Taslimi, Parham; Alanazi, Abdullah K; Noreen, Faiqa; Shafiq, Zahid

Design, synthesis, and computational insights into 3-acetyl-8-methoxy coumarin hybrids as potential anti-alzheimer's agents

3-乙酰基-8-甲氧基香豆素杂合物作为潜在抗阿尔茨海默病药物的设计、合成和计算研究

Zareen, Wajeeha; Rafique, Maham; Ahmed, Nadeem; Khan, Muhammad Ali; Tahir, Muhammad; Mali, Suraj N; Sadeghian, Nastaran; Taslimi, Parham; Ismail, Mostafa A; Chaudhari, Somdatta Y; Khan, Ajmal; Şenol, Halil; Shafiq, Zahid

Design, synthesis, and multi-target evaluation of 4-phenyl quinoline-8-sulfonate thiosemicarbazones as potential anti-Alzheimer agents

4-苯基喹啉-8-磺酸硫代氨基脲类化合物的设计、合成及多靶点评价:作为潜在的抗阿尔茨海默病药物

Saeed, Rahma; Tariq, Hafiza Zara; Althobaiti, Aiysha; Sadeghian, Nastaran; Taslimi, Parham; Al-Rashida, Mariya; Islam, Talha; Thabet, Hamdy Khamees; Aftab, Hina; Şenol, Halil; Ameen, Mubashir; Li, Jing; Shafiq, Zahid