日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural insights into selective small molecule activation of PKG1α

PKG1α选择性小分子激活的结构解析

Metwally, Essam; Mak, Victor; Soriano, Aileen; Zebisch, Matthias; Silvestre, H Leonardo; McEwan, Paul A; Ermakov, Grigori; Beaumont, Maribel; Tawa, Paul; Barker, John J; Yen, Rose; Patel, Akash; Lim, Yeon-Hee; Healy, David; Hanisak, Jennifer; Cheng, Alan C; Greshock, Tom; Fischmann, Thierry O

Towards Optimizing Sub-Normothermic Machine Perfusion in Fasciocutaneous Flaps: A Large Animal Study

优化筋膜皮瓣亚常温机器灌注:一项大型动物研究

Yanis Berkane, Alexandre G Lellouch, Guillaume Goudot, Austin Shamlou, Irina Filz von Reiterdank, Marion Goutard, Pierre Tawa, Paul Girard, Nicolas Bertheuil, Basak E Uygun, Mark A Randolph, Jérôme Duisit, Curtis L Cetrulo Jr, Korkut Uygun

Small molecule photocatalysis enables drug target identification via energy transfer

小分子光催化可通过能量转移实现药物靶点识别。

Trowbridge, Aaron D; Seath, Ciaran P; Rodriguez-Rivera, Frances P; Li, Beryl X; Dul, Barbara E; Schwaid, Adam G; Buksh, Benito F; Geri, Jacob B; Oakley, James V; Fadeyi, Olugbeminiyi O; Oslund, Rob C; Ryu, Keun Ah; White, Cory; Reyes-Robles, Tamara; Tawa, Paul; Parker, Dann L Jr; MacMillan, David W C

Discovery of the First Non-cGMP Mimetic Small Molecule Activators of cGMP-Dependent Protein Kinase 1 α (PKG1α)

发现首个非cGMP模拟小分子cGMP依赖性蛋白激酶1α(PKG1α)激活剂

Hanisak, Jennifer; Soriano, Aileen; Adam, Gregory C; Basso, Andrea; Bauman, David; Bell, David; Frank, Emily; O'Donnell, Gregory; Tawa, Paul; Verras, Andreas; Yu, Yang; Zhang, Lei; Seganish, W Michael

Identification of 53 compounds that block Ebola virus-like particle entry via a repurposing screen of approved drugs

通过对已批准药物进行再利用筛选,鉴定出 53 种可阻止埃博拉病毒样颗粒进入的化合物

Jennifer Kouznetsova, Wei Sun, Carles Martínez-Romero, Gregory Tawa, Paul Shinn, Catherine Z Chen, Aaron Schimmer, Philip Sanderson, John C McKew, Wei Zheng, Adolfo García-Sastre

In vitro characterization of MK-1439, a novel HIV-1 nonnucleoside reverse transcriptase inhibitor.

体外表征新型 HIV-1 非核苷类逆转录酶抑制剂 MK-1439

Lai Ming-Tain, Feng Meizhen, Falgueyret Jean-Pierre, Tawa Paul, Witmer Marc, DiStefano Daniel, Li Yuan, Burch Jason, Sachs Nancy, Lu Meiqing, Cauchon Elizabeth, Campeau Louis-Charles, Grobler Jay, Yan Youwei, Ducharme Yves, Côté Bernard, Asante-Appiah Ernest, Hazuda Daria J, Miller Michael D