日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis, and anticancer evaluation of novel pyrrole-pyrazoline/chalcone hybrids: in vitro and computational insights into EGFR inhibition

新型吡咯-吡唑啉/查尔酮杂合物的设计、合成及抗癌活性评价:体外和计算方法对EGFR抑制的深入研究

Alturki, Mansour S; Ahmed, Marwa F; Al Khzem, Abdulaziz H; Gomaa, Mohamed S; Sarafroz, Mohammad; Tawfeeq, Nada; Alharbi, Mashael M; Al Mouslem, Abdulaziz K; Aldawsari, Mohammed F; Alruwili, Wajin R; Khan, Shah Alam; El-Haggar, Radwan; Almalki, Atiah H

Structure-Based Discovery of Orthosteric Non-Peptide GLP-1R Agonists via Integrated Virtual Screening and Molecular Dynamics

基于结构的GLP-1R正构非肽类激动剂的发现:整合虚拟筛选和分子动力学模拟

Alturki, Mansour S; Alkhodier, Reem A; Gomaa, Mohamed S; Hussein, Dania A; Tawfeeq, Nada; Al Khzem, Abdulaziz H; Pottoo, Faheem H; Albugami, Shmoukh A; Aldawsari, Mohammed F; Rants'o, Thankhoe A

Repurposing FDA-Approved Agents to Develop a Prototype Helicobacter pylori Shikimate Kinase (HPSK) Inhibitor: A Computational Approach Using Virtual Screening, MM-GBSA Calculations, MD Simulations, and DFT Analysis

利用已获FDA批准的药物开发幽门螺杆菌莽草酸激酶(HPSK)抑制剂原型:一种结合虚拟筛选、MM-GBSA计算、分子动力学模拟和DFT分析的计算方法

Al Khzem, Abdulaziz H; Shoaib, Tagyedeen H; Mukhtar, Rua M; Alturki, Mansour S; Gomaa, Mohamed S; Hussein, Dania; Tawfeeq, Nada; Bano, Mohsina; Sarafroz, Mohammad; Alzahrani, Raghad; Alghamdi, Hanin; Rants'o, Thankhoe A

A Multifaceted Computational Approach to Identify PAD4 Inhibitors for the Treatment of Rheumatoid Arthritis (RA)

一种用于识别治疗类风湿性关节炎 (RA) 的 PAD4 抑制剂的多方面计算方法

Alturki, Mansour S; Gomaa, Mohamed S; Tawfeeq, Nada; Al Khzem, Abdulaziz H; Shaik, Mohsina B; Alshaikh Jafar, Murtadha; Alsamen, Mohammad; Al Nahab, Hasan; Al-Eid, Mohammad; Almutawah, Alhassan; Rants'o, Thankhoe A; Ayil, Khaled A G; Almaghrabi, Mohammed

Discovery of Non-Peptide GLP-1 Positive Allosteric Modulators from Natural Products: Virtual Screening, Molecular Dynamics, ADMET Profiling, Repurposing, and Chemical Scaffolds Identification

从天然产物中发现非肽类GLP-1正向变构调节剂:虚拟筛选、分子动力学模拟、ADMET分析、药物重定位和化学骨架鉴定

Gomaa, Mohamed S; Alturki, Mansour S; Tawfeeq, Nada; Hussein, Dania A; Pottoo, Faheem H; Al Khzem, Abdulaziz H; Sarafroz, Mohammad; Abubshait, Samar

Drug Repurposing for Cancer Treatment: A Comprehensive Review

药物再利用在癌症治疗中的应用:一项综合综述

Al Khzem, Abdulaziz H; Gomaa, Mohamed S; Alturki, Mansour S; Tawfeeq, Nada; Sarafroz, Mohammad; Alonaizi, Shareefa M; Al Faran, Alhassan; Alrumaihi, Laela Ahmed; Alansari, Fatimah Ahmed; Alghamdi, Abdullah Abbas

Treatment of a mutant KRAS lung cancer cell line with polyisoprenylated cysteinyl amide inhibitors activates the MAPK pathway, inhibits cell migration and induces apoptosis.

用聚异戊二烯化半胱氨酰胺抑制剂治疗突变型 KRAS 肺癌细胞系可激活 MAPK 通路,抑制细胞迁移并诱导细胞凋亡

Gregory Matthew D, Ofosu-Asante Kweku, Lazarte Jassy Mary S, Puente Pablo E, Tawfeeq Nada, Belony Nadine, Huang Yong, Offringa Ite A, Lamango Nazarius S

Polyisoprenylated Cysteinyl Amide Inhibitors: A Novel Approach to Controlling Cancers with Hyperactive Growth Signaling

聚异戊二烯化半胱氨酰酰胺抑制剂:控制具有过度活跃生长信号通路癌症的新方法

Lamango, Nazarius S; Nkembo, Augustine T; Ntantie, Elizabeth; Tawfeeq, Nada