日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Addressing the ADME Challenges of Compound Loss in a PDMS-Based Gut-on-Chip Microphysiological System

解决基于PDMS的肠道芯片微生理系统中化合物损失的ADME挑战

Carius, Patrick; Weinelt, Ferdinand Anton; Cantow, Chris; Holstein, Markus; Teitelbaum, Aaron M; Cui, Yunhai

The Absolute Bioavailability, Absorption, Distribution, Metabolism, and Excretion of BI 425809 Administered as an Oral Dose or an Oral Dose with an Intravenous Microtracer Dose of [(14)C]-BI 425809 in Healthy Males

健康男性口服 BI 425809 或口服联合静脉注射微量示踪剂 [(14)C]-BI 425809 后,其绝对生物利用度、吸收、分布、代谢和排泄情况

Burkard, Ute; Desch, Michael; Shatillo, Yury; Wunderlich, Glen; Mack, Salome Rebecca; Schlecker, Christina; Teitelbaum, Aaron M; Liu, Pingrong; Chan, Tom S

Novel advances in biotransformation and bioactivation research - 2020 year in review

生物转化和生物活化研究的新进展——2020年回顾

Khojasteh, S Cyrus; Argikar, Upendra A; Driscoll, James P; Heck, Carley J S; King, Lloyd; Jackson, Klarissa D; Jian, Wenying; Kalgutkar, Amit S; Miller, Grover P; Kramlinger, Valerie; Rietjens, Ivonne M C M; Teitelbaum, Aaron M; Wang, Kai; Wei, Cong

Species Differences in Microsomal Oxidation and Glucuronidation of 4-Ipomeanol: Relationship to Target Organ Toxicity

4-异戊烯醇微粒体氧化和葡萄糖醛酸化的物种差异:与靶器官毒性的关系

Parkinson, Oliver T; Teitelbaum, Aaron M; Whittington, Dale; Kelly, Edward J; Rettie, Allan E

Inhibitors of the salicylate synthase (MbtI) from Mycobacterium tuberculosis discovered by high-throughput screening

通过高通量筛选发现结核分枝杆菌水杨酸合成酶 (MbtI) 抑制剂

Vasan, Mahalakshmi; Neres, João; Williams, Jessica; Wilson, Daniel J; Teitelbaum, Aaron M; Remmel, Rory P; Aldrich, Courtney C

Natural history of experimental arterial chronic total occlusions

实验性动脉慢性完全闭塞的自然史

Jaffe, Ronen; Leung, General; Munce, Nigel R; Thind, Amandeep S; Leong-Poi, Howard; Anderson, Kevan J T; Qi, Xiuling; Trogadis, Judy; Nadler, Ariella; Shiff, Davida; Saperia, Jamie; Lockwood, Julia; Jacobs, Chaim; Qiang, Beiping; Teitelbaum, Aaron; Dick, Alexander J; Sparkes, John D; Butany, Jagdish; Wright, Graham A; Strauss, Bradley H

Efficacy of Carraguard-based microbicides in vivo despite variable in vitro activity.

尽管体外活性存在差异,但卡拉胶基杀菌剂在体内仍具有疗效

Turville Stuart G, Aravantinou Meropi, Miller Todd, Kenney Jessica, Teitelbaum Aaron, Hu Lieyu, Chudolij Anne, Zydowsky Tom M, Piatak Michael Jr, Bess Julian W Jr, Lifson Jeffrey D, Blanchard James, Gettie Agegnehu, Robbiani Melissa