日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Therapeutic optimization of LIPA targeting to induce endoplasmic reticulum stress and cell death in ovarian cancer.

LIPA靶向治疗的优化,以诱导卵巢癌内质网应激和细胞死亡。

Viswanadhapalli Suryavathi, Lee Tae-Kyung, Elmore Scott, Sharma Gaurav, Gopalam Rahul, Panneerdoss Durga Meenakshi, Liu Xihui, Parra Karla, Reese Tanner, Hsieh Michael, Pratap Uday P, Yang Xue, Ebrahimi Behnam, Li Xiaonan, Neal Henry, Chen Chia-Yuan, Kassees Kara, Cervantes Christian, Baker Adriana, Subbarayalu Panneerdoss, Ramirez Paulina, Lyons Yasmin A, Lai Zhao, Chen Yidong, Boerma Joseph W, LoCoco Peter M, Clanton Nicholas A, Xu Zhenming, Rao Manjeet, Rao Tekmal Rajeshwar, Kost Edward, Sareddy Gangadhara R, Raj Ganesh V, Ahn Jung-Mo, Vadlamudi Ratna K

Lysine-specific histone demethylase 1A (KDM1A/LSD1) inhibition attenuates DNA double-strand break repair and augments the efficacy of temozolomide in glioblastoma

赖氨酸特异性组蛋白去甲基化酶1A (KDM1A/LSD1) 抑制剂可减弱DNA双链断裂修复,并增强替莫唑胺在胶质母细胞瘤中的疗效。

Alejo, Salvador; Palacios, Bridgitte E; Venkata, Prabhakar Pitta; He, Yi; Li, Wenjing; Johnson, Jessica D; Chen, Yihong; Jayamohan, Sridharan; Pratap, Uday P; Clarke, Kyra; Zou, Yi; Lv, Yingli; Weldon, Korri; Viswanadhapalli, Suryavathi; Lai, Zhao; Ye, Zhenqing; Chen, Yidong; Gilbert, Andrea R; Suzuki, Takayoshi; Tekmal, Rajeshwar R; Zhao, Weixing; Zheng, Siyuan; Vadlamudi, Ratna K; Brenner, Andrew J; Sareddy, Gangadhara R

Pharmacological inhibition of KDM1A/LSD1 enhances estrogen receptor beta-mediated tumor suppression in ovarian cancer

药理学抑制 KDM1A/LSD1 可增强雌激素受体 β 介导的卵巢癌肿瘤抑制

Prabhakar Pitta Venkata, Sridharan Jayamohan, Yi He, Salvador Alejo, Jessica D Johnson, Bridgitte E Palacios, Uday P Pratap, Yihong Chen, Zexuan Liu, Yi Zou, Zhao Lai, Takayoshi Suzuki, Suryavathi Viswanadhapalli, Susan T Weintraub, Srinath Palakurthi, Philip T Valente, Rajeshwar R Tekmal, Edward R

Preclinical Development of Brain Permeable ERβ Agonist for the Treatment of Glioblastoma

用于治疗胶质母细胞瘤的脑通透性 ERβ 激动剂的临床前开发

Uday P Pratap, Michael Tidwell, Henriette U Balinda, Nicholas A Clanton, Xue Yang, Suryavathi Viswanadhapalli, Gangadhara R Sareddy, Dong Liang, Huan Xie, Yidong Chen, Zhao Lai, Rajeshwar R Tekmal, Stanton F McHardy, Andrew J Brenner, Ratna K Vadlamudi

The LIFR Inhibitor EC359 Effectively Targets Type II Endometrial Cancer by Blocking LIF/LIFR Oncogenic Signaling

LIFR 抑制剂 EC359 通过阻断 LIF/LIFR 致癌信号有效靶向 II 型子宫内膜癌

Nicole Spencer, Alondra Lee Rodriguez Sanchez, Rahul Gopalam, Panneerdoss Subbarayalu, Daisy M Medina, Xue Yang, Paulina Ramirez, Lois Randolph, Emily Jean Aller, Bindu Santhamma, Manjeet K Rao, Rajeshwar Rao Tekmal, Hareesh B Nair, Edward R Kost, Ratna K Vadlamudi, Suryavathi Viswanadhapalli

Development and Characterization of Inducible Astrocyte-Specific Aromatase Knockout Mice

可诱导星形胶质细胞特异性芳香化酶基因敲除小鼠的开发和鉴定

Jing Wang, Uday P Pratap, Yujiao Lu, Gangadhara R Sareddy, Rajeshwar R Tekmal, Ratna K Vadlamudi, Darrell W Brann

Targeting LIPA independent of its lipase activity is a therapeutic strategy in solid tumors via induction of endoplasmic reticulum stress

靶向 LIPA(不依赖于其脂肪酶活性)是通过诱导内质网应激来治疗实体瘤的一种策略。

Xihui Liu ,Suryavathi Viswanadhapalli ,Shourya Kumar ,Tae-Kyung Lee ,Andrew Moore ,Shihong Ma ,Liping Chen ,Michael Hsieh ,Mengxing Li ,Gangadhara R Sareddy ,Karla Parra ,Eliot B Blatt ,Tanner C Reese ,Yuting Zhao ,Annabel Chang ,Hui Yan ,Zhenming Xu ,Uday P Pratap ,Zexuan Liu ,Carlos M Roggero ,Zhenqiu Tan ,Susan T Weintraub ,Yan Peng ,Rajeshwar R Tekmal ,Carlos L Arteaga ,Jennifer Lippincott-Schwartz ,Ratna K Vadlamudi ,Jung-Mo Ahn ,Ganesh V Raj

KDM1A inhibition augments the efficacy of rapamycin for the treatment of endometrial cancer

KDM1A 抑制可增强雷帕霉素治疗子宫内膜癌的疗效

Prabhakar Pitta Venkata, Yihong Chen, Salvador Alejo, Yi He, Bridgitte E Palacios, Ilanna Loeffel, Junhao Liu, Uday P Pratap, Gabrielle Gray, Sureshkumar Mulampurath Achuthan Pillai, Yi Zou, Zhao Lai, Takayoshi Suzuki, Suryavathi Viswanadhapalli, Srinath Palakurthi, Rajeshwar R Tekmal, Ratna K Vadla

Brain-derived estrogen and neural function

脑源性雌激素与神经功能

Brann, Darrell W; Lu, Yujiao; Wang, Jing; Zhang, Quanguang; Thakkar, Roshni; Sareddy, Gangadhara R; Pratap, Uday P; Tekmal, Rajeshwar R; Vadlamudi, Ratna K

SETDB1 interactions with PELP1 contributes to breast cancer endocrine therapy resistance

SETDB1 与 PELP1 的相互作用导致乳腺癌内分泌治疗耐药性

Zexuan Liu, Junhao Liu, Behnam Ebrahimi, Uday P Pratap, Yi He, Kristin A Altwegg, Weiwei Tang, Xiaonan Li, Zhao Lai, Yidong Chen, Liangfang Shen, Gangadhara R Sareddy, Suryavathi Viswanadhapalli, Rajeshwar R Tekmal, Manjeet K Rao, Ratna K Vadlamudi