日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacophore Modeling of Janus Kinase Inhibitors: Tools for Drug Discovery and Exposition Prediction

Janus激酶抑制剂的药效团模型:药物发现和暴露预测的工具

Fischer, Florian; Temml, Veronika; Schuster, Daniela

Microtubule inhibition as a proposed mechanism for the anthelmintic effect of phytochemicals isolated from Cicerbita alpina.

微管抑制是高山鹰嘴豆中分离出的植物化学物质发挥驱虫作用的一种可能机制

Horgan Mark James, Sigg Ines, Poulopoulou Ioanna, Rodriguez-Mejias Francisco J, Albertini Eva, Fusani Pietro, Fischer Florian, Martinidou Eftychia, Schuster Daniela, Martens Stefan, Dürr Pidder Jansen, Gauly Matthias, Stuppner Hermann, Weiss Alexander, Temml Veronika, Siewert Bianka

Identification of Novel β-Tubulin Inhibitors Using a Combined In Silico/ In Vitro Approach

使用计算机模拟/体外实验相结合的方法鉴定新型 β-微管蛋白抑制剂

Mark James Horgan, Lukas Zell, Bianka Siewert, Hermann Stuppner, Daniela Schuster, Veronika Temml

Highly potent and selective 5-lipoxygenase inhibition by new, simple heteroaryl-substituted catechols for treatment of inflammation

通过新的、简单的杂芳基取代的儿茶酚高效、选择性地抑制 5-脂氧合酶以治疗炎症

Verena Krauth, Ferdinando Bruno, Simona Pace, Paul M Jordan, Veronika Temml, Maria Preziosa Romano, Haroon Khan, Daniela Schuster, Antonietta Rossi, Rosanna Filosa, Oliver Werz

Dopamine Receptor Ligand Selectivity-An In Silico/In Vitro Insight

多巴胺受体配体选择性-计算机模拟/体外洞察

Lukas Zell, Alina Bretl, Veronika Temml, Daniela Schuster

Synthesis and structure-activity relationships for some novel diflapolin derivatives with benzimidazole subunit

一些新型苯并咪唑亚基二甲胺衍生物的合成及构效关系

Lisa Vieider, Eva Zoeller, Erik Romp, Martin Schoenthaler, Victor Hernández-Olmos, Veronika Temml, Thomas Hasenoehrl, Daniela Schuster, Oliver Werz, Ulrike Garscha, Barbara Matuszczak

Identification of Novel Dopamine D2 Receptor Ligands-A Combined In Silico/In Vitro Approach

新型多巴胺 D2 受体配体的鉴定-计算机/体外联合方法

Lukas Zell, Constanze Lainer, Jakub Kollár, Veronika Temml, Daniela Schuster

Analogues of Natural Chalcones as Efficient Inhibitors of AKR1C3

天然查尔酮类似物作为AKR1C3的有效抑制剂

Möller, Gabriele; Temml, Veronika; Cala Peralta, Antonio; Gruet, Océane; Richomme, Pascal; Séraphin, Denis; Viault, Guillaume; Kraus, Luisa; Huber-Cantonati, Petra; Schopfhauser, Elisabeth; Pachmayr, Johanna; Tokarz, Janina; Schuster, Daniela; Helesbeux, Jean-Jacques; Dyar, Kenneth Allen

From Vietnamese plants to a biflavonoid that relieves inflammation by triggering the lipid mediator class switch to resolution

从越南植物到一种通过触发脂质介质类别转换来缓解炎症的双黄酮类化合物,最终促成炎症消退。

Tran Thi Van Anh ,Alilou Mostafa ,Zhigang Rao ,Simona Pace ,Stefan Schwaiger ,Christian Kretzer ,Veronika Temml ,Carsten Giesel ,Paul M Jordan ,Rossella Bilancia ,Christina Weinigel ,Silke Rummler ,Birgit Waltenberger ,Tran Hung ,Antonietta Rossi ,Hermann Stuppner ,Oliver Werz ,Andreas Koeberle

Exploration of Long-Chain Vitamin E Metabolites for the Discovery of a Highly Potent, Orally Effective, and Metabolically Stable 5-LOX Inhibitor that Limits Inflammation

探索长链维生素 E 代谢物,以发现一种高效、口服有效、代谢稳定的 5-LOX 抑制剂,以限制炎症

Konstantin Neukirch, Khaled Alsabil, Chau-Phi Dinh, Rossella Bilancia, Martin Raasch, Alexia Ville, Ida Cerqua, Guillaume Viault, Dimitri Bréard, Simona Pace, Veronika Temml, Elena Brunner, Paul M Jordan, Marta C Marques, Konstantin Loeser, André Gollowitzer, Stephan Permann, Jana Gerstmeier, Stefan