日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Microglial-Targeted GCPII Inhibition Reverses Neurocognitive Impairment and Synaptic Loss After EcoHIV Infection.

靶向小胶质细胞的 GCPII 抑制可逆转 EcoHIV 感染后的神经认知障碍和突触丢失。

Zheng Yuxin, Huang Meixiang, Maragakis R Michael, Pietri Peter, Su Yu, Alt Jesse, Tenora Lukáš, Liyanage Wathsala, Wu Ying, Thomas Mary-Anne, Kannan Rangaramanujam M, Zhu Xiaolei, Rais Rana, Slusher Barbara S

A Star-PEGylation Strategy to Improve Testosterone Pharmacokinetics

星形聚乙二醇化策略改善睾酮药代动力学

Lee, Chae Bin; Tenora, Lukáš; Zhang, Ruoning; Ranjit, Arina; Markowski, Mark C; Slusher, Barbara S; Rais, Rana

Inhibition of microglial glutaminase alleviates chronic stress-induced neurobehavioral and cognitive deficits

抑制小胶质细胞谷氨酰胺酶可缓解慢性应激引起的神经行为和认知缺陷

Huang, Meixiang; Li, Yannan; Thomas, Ajit G; Sharma, Anjali; Liyanage, Wathsala; Tichý, Tomáš; Tenora, Lukáš; Su, Yu; Ha, Jisu; Hin, Niyada; Obayashi, Mizuho; Majer, Pavel; Kannan, Rangaramanujam M; Tsukamoto, Takashi; Ursini, Gianluca; Rais, Rana; Slusher, Barbara S; Zhu, Xiaolei

Pharmacokinetic Evaluation of Neutral Sphinghomyelinase2 (nSMase2) Inhibitor Prodrugs in Mice and Dogs

中性鞘磷脂酶2 (nSMase2) 抑制剂前药在小鼠和犬体内的药代动力学评价

Ranjit, Arina; Lee, Chae Bin; Tenora, Lukáš; Mettu, Vijaya Saradhi; Pal, Arindom; Alt, Jesse; Slusher, Barbara S; Rais, Rana

A gut-restricted glutamate carboxypeptidase II inhibitor reduces monocytic inflammation and improves preclinical colitis

肠道特异性谷氨酸羧肽酶II抑制剂可减轻单核细胞炎症并改善临床前结肠炎

Diane E Peters ,Lauren D Norris ,Lukáš Tenora ,Ivan Šnajdr ,András K Ponti ,Xiaolei Zhu ,Shinji Sakamoto ,Vijayabhaskar Veeravalli ,Manisha Pradhan ,Jesse Alt ,Ajit G Thomas ,Pavel Majer ,Rana Rais ,Christine McDonald ,Barbara S Slusher

Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery

发现基于叔丁酯的 6-重氮-5-氧代-l-正亮氨酸前药,用于增强代谢稳定性和肿瘤递送

Kateřina Novotná, Lukáš Tenora, Eva Prchalová, James Paule, Jesse Alt, Vijay Veeravalli, Jenny Lam, Ying Wu, Ivan Šnajdr, Sadakatali Gori, Vijaya Saradhi Mettu, Takashi Tsukamoto, Pavel Majer, Barbara S Slusher, Rana Rais

Microglial-Targeted nSMase2 Inhibitor Fails to Reduce Tau Propagation in PS19 Mice

靶向小胶质细胞的nSMase2抑制剂未能减少PS19小鼠体内Tau蛋白的扩散

Meixiang Huang ,Carolyn Tallon ,Xiaolei Zhu ,Kaitlyn D J Huizar ,Silvia Picciolini ,Ajit G Thomas ,Lukas Tenora ,Wathsala Liyanage ,Francesca Rodà ,Alice Gualerzi ,Rangaramanujam M Kannan ,Marzia Bedoni ,Rana Rais ,Barbara S Slusher

The combination of immunotherapy and a glutamine metabolism inhibitor represents an effective therapeutic strategy for advanced and metastatic murine pancreatic adenocarcinoma

免疫疗法与谷氨酰胺代谢抑制剂的联合应用是治疗晚期和转移性小鼠胰腺腺癌的有效策略。

Frejlachova, Andrea; Lencova, Radka; Venhauerova, Anna; Skalickova, Marketa; Uher, Ondrej; Caisova, Veronika; Majer, Pavel; Tenora, Lukas; Hansen, Per; Chmelar, Jindrich; Kopecky, Jan; Zhuang, Zhengping; Pacak, Karel; Zenka, Jan

Discovery of DRP-104, a tumor-targeted metabolic inhibitor prodrug

发现肿瘤靶向代谢抑制剂前药DRP-104

Rais, Rana; Lemberg, Kathryn M; Tenora, Lukáš; Arwood, Matthew L; Pal, Arindom; Alt, Jesse; Wu, Ying; Lam, Jenny; Aguilar, Joanna Marie H; Zhao, Liang; Peters, Diane E; Tallon, Carolyn; Pandey, Rajeev; Thomas, Ajit G; Dash, Ranjeet P; Seiwert, Tanguy; Majer, Pavel; Leone, Robert D; Powell, Jonathan D; Slusher, Barbara S

Global Impact of the COVID-19 Pandemic on Cerebral Venous Thrombosis and Mortality

COVID-19 大流行对脑静脉血栓形成和死亡率的全球影响

Nguyen, Thanh N; Qureshi, Muhammad M; Klein, Piers; Yamagami, Hiroshi; Abdalkader, Mohamad; Mikulik, Robert; Sathya, Anvitha; Mansour, Ossama Yassin; Czlonkowska, Anna; Lo, Hannah; Field, Thalia S; Charidimou, Andreas; Banerjee, Soma; Yaghi, Shadi; Siegler, James E; Sedova, Petra; Kwan, Joseph; de Sousa, Diana Aguiar; Demeestere, Jelle; Inoa, Violiza; Omran, Setareh Salehi; Zhang, Liqun; Michel, Patrik; Strambo, Davide; Marto, João Pedro; Nogueira, Raul G; Kristoffersen, Espen Saxhaug; Tsivgoulis, Georgios; Lereis, Virginia Pujol; Ma, Alice; Enzinger, Christian; Gattringer, Thomas; Rahman, Aminur; Bonnet, Thomas; Ligot, Noémie; De Raedt, Sylvie; Lemmens, Robin; Vanacker, Peter; Vandervorst, Fenne; Conforto, Adriana Bastos; Hidalgo, Raquel C T; Mora Cuervo, Daissy Liliana; de Oliveira Neves, Luciana; Lameirinhas da Silva, Isabelle; Martíns, Rodrigo Targa; Rebello, Letícia C; Santiago, Igor Bessa; Sakelarova, Teodora; Kalpachki, Rosen; Alexiev, Filip; Cora, Elena Adela; Kelly, Michael E; Peeling, Lissa; Pikula, Aleksandra; Chen, Hui-Sheng; Chen, Yimin; Yang, Shuiquan; Roje Bedekovic, Marina; Čabal, Martin; Tenora, Dusan; Fibrich, Petr; Dušek, Pavel; Hlaváčová, Helena; Hrabanovska, Emanuela; Jurák, Lubomír; Kadlčíková, Jana; Karpowicz, Igor; Klečka, Lukáš; Kovář, Martin; Neumann, Jiří; Paloušková, Hana; Reiser, Martin; Rohan, Vladimir; Šimůnek, Libor; Skoda, Ondreij; Škorňa, Miroslav; Šrámek, Martin; Drenck, Nicolas; Sobh, Khalid; Lesaine, Emilie; Sabben, Candice; Reiner, Peggy; Rouanet, Francois; Strbian, Daniel; Boskamp, Stefan; Mbroh, Joshua; Nagel, Simon; Rosenkranz, Michael; Poli, Sven; Thomalla, Götz; Karapanayiotides, Theodoros; Koutroulou, Ioanna; Kargiotis, Odysseas; Palaiodimou, Lina; Barrientos Guerra, José Dominguo; Huded, Vikram; Nagendra, Shashank; Prajapati, Chintan; Sylaja, P N; Sani, Achmad Firdaus; Ghoreishi, Abdoreza; Farhoudi, Mehdi; Sadeghi Hokmabadi, Elyar; Hashemilar, Mazyar; Sabetay, Sergiu Ionut; Rahal, Fadi; Acampa, Maurizio; Adami, Alessandro; Longoni, Marco; Ornello, Raffaele; Renieri, Leonardo; Romoli, Michele; Sacco, Simona; Salmaggi, Andrea; Sangalli, Davide; Zini, Andrea; Sakai, Kenichiro; Fukuda, Hiroki; Fujita, Kyohei; Imamura, Hirotoshi; Kosuke, Miyake; Sakaguchi, Manabu; Sonoda, Kazutaka; Matsumaru, Yuji; Ohara, Nobuyuki; Shindo, Seigo; Takenobu, Yohei; Yoshimoto, Takeshi; Toyoda, Kazunori; Uwatoko, Takeshi; Sakai, Nobuyuki; Yamamoto, Nobuaki; Yamamoto, Ryoo; Yazawa, Yukako; Sugiura, Yuri; Baek, Jang-Hyun; Lee, Si Baek; Seo, Kwon-Duk; Sohn, Sung-Il; Lee, Jin Soo; Arsovska, Anita Ante; Chieh, Chan Yong; Wan Zaidi, Wan Asyraf; Wan Yahya, Wan Nur Nafisah; Gongora-Rivera, Fernando; Martinez-Marino, Manuel; Infante-Valenzuela, Adrian; Dippel, Diederik; van Dam-Nolen, Dianne H K; Wu, Teddy Y; Punter, Martin; Adebayo, Tajudeen Temitayo; Bello, Abiodun H; Sunmonu, Taofiki Ajao; Wahab, Kolawole Wasiu; Sundseth, Antje; Al Hashmi, Amal M; Ahmad, Saima; Rashid, Umair; Rodriguez-Kadota, Liliana; Vences, Miguel Ángel; Yalung, Patrick Matic; Dy, Jon Stewart Hao; Brola, Waldemar; Dębiec, Aleksander; Dorobek, Malgorzata; Karlinski, Michal Adam; Labuz-Roszak, Beata M; Lasek-Bal, Anetta; Sienkiewicz-Jarosz, Halina; Staszewski, Jacek; Sobolewski, Piotr; Wiącek, Marcin; Zielinska-Turek, Justyna; Araújo, André Pinho; Rocha, Mariana; Castro, Pedro; Ferreira, Patricia; Nunes, Ana Paiva; Fonseca, Luísa; Pinho E Melo, Teresa; Rodrigues, Miguel; Silva, M Luis; Ciopleias, Bogdan; Dimitriade, Adela; Falup-Pecurariu, Cristian; Hamid, May Adel; Venketasubramanian, Narayanaswamy; Krastev, Georgi; Haring, Jozef; Ayo-Martin, Oscar; Hernandez-Fernandez, Francisco; Blasco, Jordi; Rodríguez-Vázquez, Alejandro; Cruz-Culebras, Antonio; Moniche, Francisco; Montaner, Joan; Perez-Sanchez, Soledad; García Sánchez, María Jesús; Guillán Rodríguez, Marta; Bernava, Gianmarco; Bolognese, Manuel; Carrera, Emmanuel; Churojana, Anchalee; Aykac, Ozlem; Özdemir, Atilla Özcan; Bajrami, Arsida; Senadim, Songul; Hussain, Syed I; John, Seby; Krishnan, Kailash; Lenthall, Robert; Asif, Kaiz S; Below, Kristine; Biller, Jose; Chen, Michael; Chebl, Alex; Colasurdo, Marco; Czap, Alexandra; de Havenon, Adam H; Dharmadhikari, Sushrut; Eskey, Clifford J; Farooqui, Mudassir; Feske, Steven K; Goyal, Nitin; Grimmett, Kasey B; Guzik, Amy K; Haussen, Diogo C; Hovingh, Majesta; Jillela, Dinesh; Kan, Peter T; Khatri, Rakesh; Khoury, Naim N; Kiley, Nicole L; Kolikonda, Murali K; Lara, Stephanie; Li, Grace; Linfante, Italo; Loochtan, Aaron I; Lopez, Carlos D; Lycan, Sarah; Male, Shailesh S; Nahab, Fadi; Maali, Laith; Masoud, Hesham E; Min, Jiangyong; Orgeta-Gutierrez, Santiago; Mohamed, Ghada A; Mohammaden, Mahmoud; Nalleballe, Krishna; Radaideh, Yazan; Ramakrishnan, Pankajavalli; Rayo-Taranto, Bliss; Rojas-Soto, Diana M; Ruland, Sean; Simpkins, Alexis N; Sheth, Sunil A; Starosciak, Amy K; Tarlov, Nicholas E; Taylor, Robert A; Voetsch, Barbara; Zhang, Linda; Duong, Hai Quang; Dao, Viet-Phuong; Le, Huynh Vu; Pham, Thong Nhu; Ton, Mai Duy; Tran, Anh Duc; Zaidat, Osama O; Machi, Paolo; Dirren, Elisabeth; Rodríguez Fernández, Claudio; Escartín López, Jorge; Fernández Ferro, Jose Carlos; Mohammadzadeh, Niloofar; Suryadevara, Neil C; de la Cruz Fernández, Beatriz; Bessa, Filipe; Jancar, Nina; Brady, Megan; Scozzari, Dawn