日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Flexible fluorine-thiol displacement stapled peptides with enhanced membrane penetration for the estrogen receptor/coactivator interaction

柔性氟硫醇置换交联肽,具有增强的膜穿透性,可用于雌激素受体/辅激活因子相互作用

Robert Maloney ,Samuel L Junod ,Kyla M Hagen ,Todd Lewis ,Changfeng Cheng ,Femil J Shajan ,Mi Zhao ,Terry W Moore ,Thu H Truong ,Weidong Yang ,Rongsheng E Wang

Structure-Activity Relationships of the Antimicrobial Peptide Natural Product Apidaecin

抗菌肽天然产物Apidaecin的构效关系

Kornelia J Skowron, Chetana Baliga, Tatum Johnson, Kyle M Kremiller, Alexandra Castroverde, Trevor T Dean, A'Lester C Allen, Ana M Lopez-Hernandez, Elena V Aleksandrova, Dorota Klepacki, Alexander S Mankin, Yury S Polikanov, Terry W Moore

Labeling of a mutant estrogen receptor with an Affimer in a breast cancer cell line

在乳腺癌细胞系中用 Affimer 标记突变雌激素受体

Pin Ren, Christian Tiede, Sean W Fanning, Thomas Adams, Valerie Speirs, Erik R Nelson, Changfeng Cheng, Terry W Moore, Geoffrey L Greene, Darren Tomlinson, Paul R Selvin

Detection of thermal shift in cellular Keap1 by protein-protein interaction inhibitors using immunoblot- and fluorescence microplate-based assays

使用免疫印迹和荧光微孔板法检测蛋白质-蛋白质相互作用抑制剂对细胞 Keap1 的热变化

Sharadha Dayalan Naidu, Dina Dikovskaya, Terry W Moore, Albena T Dinkova-Kostova

Molecular basis for the disruption of Keap1-Nrf2 interaction via Hinge & Latch mechanism

通过铰链和闩锁机制破坏 Keap1-Nrf2 相互作用的分子基础

Yuta Horie #, Takafumi Suzuki #, Jin Inoue #, Tatsuro Iso, Geoffrey Wells, Terry W Moore, Tsunehiro Mizushima, Albena T Dinkova-Kostova, Takuma Kasai, Takashi Kamei, Seizo Koshiba, Masayuki Yamamoto6

The isoquinoline PRL-295 increases the thermostability of Keap1 and disrupts its interaction with Nrf2

异喹啉 PRL-295 可提高 Keap1 的热稳定性并破坏其与 Nrf2 的相互作用

Sharadha Dayalan Naidu, Takafumi Suzuki, Dina Dikovskaya, Elena V Knatko, Maureen Higgins, Miu Sato, Miroslav Novak, José A Villegas, Terry W Moore, Masayuki Yamamoto, Albena T Dinkova-Kostova

Isoquinoline Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-Derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability

具有高代谢稳定性的异喹啉类 ECH 相关蛋白 1-核因子(红细胞衍生 2)样 2 (KEAP1-NRF2) 抑制剂

Phillip R Lazzara, Brian P David, Aparna Ankireddy, Benjamin G Richardson, Katherine Dye, Kiira M Ratia, Sekhar P Reddy, Terry W Moore

SAR Study on Estrogen Receptor α/β Activity of (Iso)flavonoids: Importance of Prenylation, C-Ring (Un)Saturation, and Hydroxyl Substituents

(异)黄酮类化合物雌激素受体 α/β 活性的 SAR 研究:异戊烯化、C 环(不)饱和和羟基取代基的重要性

Obinna C Mbachu, Caitlin Howell, Charlotte Simmler, Gonzalo R Malca Garcia, Kornelia J Skowron, Huali Dong, Sarah G Ellis, Ryan T Hitzman, Atieh Hajirahimkhan, Shao-Nong Chen, Dejan Nikolic, Terry W Moore, Günter Vollmer, Guido F Pauli, Judy L Bolton, Birgit M Dietz

Replacement of a Naphthalene Scaffold in Kelch-like ECH-Associated Protein 1 (KEAP1)/Nuclear Factor (Erythroid-derived 2)-like 2 (NRF2) Inhibitors

凯尔奇样 ECH 相关蛋白 1 (KEAP1)/核因子(红细胞衍生 2)样 2 (NRF2) 抑制剂中萘支架的替换

Benjamin G Richardson, Atul D Jain, Haranatha R Potteti, Phillip R Lazzara, Brian P David, Chandra R Tamatam, Ewelina Choma, Kornelia Skowron, Katherine Dye, Zamia Siddiqui, Yue-Ting Wang, Aleksej Krunic, Sekhar P Reddy, Terry W Moore

A Cell-Permeable Stapled Peptide Inhibitor of the Estrogen Receptor/Coactivator Interaction

雌激素受体/辅激活因子相互作用的细胞通透性钉合肽抑制剂

Thomas E Speltz, Jeanne M Danes, Joshua D Stender, Jonna Frasor, Terry W Moore