日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemoproteomics validates selective targeting of Plasmodium M1 alanyl aminopeptidase as an antimalarial strategy

化学蛋白质组学验证了选择性靶向疟原虫 M1 丙氨酰氨基肽酶作为抗疟策略

Carlo Giannangelo #, Matthew P Challis #, Ghizal Siddiqui, Rebecca Edgar, Tess R Malcolm, Chaille T Webb, Nyssa Drinkwater, Natalie Vinh, Christopher Macraild, Natalie Counihan, Sandra Duffy, Sergio Wittlin, Shane M Devine, Vicky M Avery, Tania De Koning-Ward, Peter Scammells, Sheena McGowan, Darren

On-target, dual aminopeptidase inhibition provides cross-species antimalarial activity

靶向双氨基肽酶抑制提供跨物种抗疟活性

Rebecca C S Edgar, Tess R Malcolm, Ghizal Siddiqui, Carlo Giannangelo, Natalie A Counihan, Matthew Challis, Sandra Duffy, Mrittika Chowdhury, Jutta Marfurt, Madeline Dans, Grennady Wirjanata, Rintis Noviyanti, Kajal Daware, Chathura D Suraweera, Ric N Price, Sergio Wittlin, Vicky M Avery, Nyssa Drin

Experimental infection of ringtail possums (Pseudocheirus peregrinus) with Mycobacterium ulcerans, the agent of Buruli ulcer

用溃疡分枝杆菌(布鲁里溃疡的病原体)对环尾负鼠(Pseudocheirus peregrinus)进行实验性感染

Blasdell, Kim R; Ploeg, Richard J; Hobbs, Emma C; Muhi, Stephen; Riddell, Sarah J; Cunneen, Alexandra; Kelly, Michael L; Maynard, Kate; Malcolm, Tess R; Islam, Md Tanjir; Boyd, Victoria; Stinear, Timothy P; Pidot, Sacha J; Athan, Eugene; O'Brien, Daniel P

Physiological and perceptual responses of wearing a dryrobe for rewarming after passive cold-water immersion in men

男性被动冷水浸泡后穿着干式保暖服进行复温的生理和感知反应

Read, Dale B; Flood, Tess R; Harwood, Amy E; Dos'Santos, Thomas; Weakley, Jonathon J S; Evans, Gethin H

High-throughput experimentation for discovery of biodegradable polyesters

用于发现可生物降解聚酯的高通量实验

Fransen, Katharina A; Av-Ron, Sarah H M; Buchanan, Tess R; Walsh, Dylan J; Rota, Dechen T; Van Note, Lana; Olsen, Bradley D

Human Tim8a, Tim8b and Tim13 are auxiliary assembly factors of mature Complex IV

人类的Tim8a、Tim8b和Tim13是成熟复合物IV的辅助组装因子。

Alexander J Anderson, Jordan J Crameri, Ching-Seng Ang, Tess R Malcolm, Yilin Kang, Megan J Baker, Catherine S Palmer, Alice J Sharpe, Luke E Formosa, Katherine Ganio, Michael J Baker, Christopher A McDevitt, Michael T Ryan, Megan J Maher, Diana Stojanovski

Genetic and chemical validation of Plasmodium falciparum aminopeptidase Pf A-M17 as a drug target in the hemoglobin digestion pathway

恶性疟原虫氨基肽酶 Pf A-M17 作为血红蛋白消化途径药物靶点的遗传和化学验证

Rebecca C S Edgar, Ghizal Siddiqui, Katheryn Hjerrild, Tess R Malcolm, Natalie B Vinh, Chaille T Webb, Clare Holmes, Christopher A MacRaild, Hope C Chernih, Willy W Suen, Natalie A Counihan, Darren J Creek, Peter J Scammells, Sheena McGowan, Tania F de Koning-Ward

A metal ion-dependent conformational switch modulates activity of the Plasmodium M17 aminopeptidase

金属离子依赖性构象开关调节疟原虫M17氨基肽酶的活性

Chaille T Webb, Wei Yang, Blake T Riley, Brooke K Hayes, Komagal Kannan Sivaraman, Tess R Malcolm, Stephen Harrop, Sarah C Atkinson, Itamar Kass, Ashley M Buckle, Nyssa Drinkwater, Sheena McGowan

The structural basis of bacterial manganese import

细菌锰输入的结构基础

Neville, Stephanie L; Sjöhamn, Jennie; Watts, Jacinta A; MacDermott-Opeskin, Hugo; Fairweather, Stephen J; Ganio, Katherine; Carey Hulyer, Alex; McGrath, Aaron P; Hayes, Andrew J; Malcolm, Tess R; Davies, Mark R; Nomura, Norimichi; Iwata, So; O'Mara, Megan L; Maher, Megan J; McDevitt, Christopher A

Mapping the substrate specificity of the Plasmodium M1 and M17 aminopeptidases

绘制疟原虫 M1 和 M17 氨基肽酶的底物特异性图谱

Tess R Malcolm, Karolina W Swiderska, Brooke K Hayes, Chaille T Webb, Marcin Drag, Nyssa Drinkwater, Sheena McGowan