Fentanyl-Type Antagonist of the μ-Opioid Receptor: Important Role of Axial Chirality in the Active Conformation
μ-阿片受体的芬太尼型拮抗剂:轴向手性在活性构象中的重要作用
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c00935
Arita, Hironobu; Tanaka, Ryoko; Kikukawa, Shuntaro; Tomizawa, Tsukasa; Sakata, Haruka; Funada, Masahiko; Tomiyama, Kenichi; Hashimoto, Masaru; Tasaka, Tomohiko; Tabata, Hidetsugu; Nakamura, Kayo; Makino, Kosho; Oshitari, Tetsuta; Natsugari, Hideaki; Takahashi, Hideyo