日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Shifting the PPARγ conformational ensemble toward a transcriptionally repressive state improves covalent inhibitor efficacy

将PPARγ构象集合体向转录抑制状态转变可提高共价抑制剂的效力。

Arifova, Liudmyla; MacTavish, Brian S; Laughlin, Zane; Karadi Girdhar, Mithun Nag; Shang, Jinsai; Li, Min-Hsuan; Yu, Xiaoyu; Zhu, Di; Kamenecka, Theodore M; Kojetin, Douglas J

Relationships Between Circulating Lipids, Lipoproteins, and Lymphocyte Subsets in the Multi-Ethnic Study of Atherosclerosis

多民族动脉粥样硬化研究中循环脂质、脂蛋白和淋巴细胞亚群之间的关系

DeConne, Theodore M; Sitlani, Colleen M; Delaney, Joseph A; Psaty, Bruce M; Doyle, Margaret F; Otvos, James D; Feinstein, Matthew J; Olson, Nels C

Diverse high-fat diets drive multi-omic reprogramming that persists after dietary reversal

多种高脂肪饮食会驱动多组学重编程,这种重编程在饮食逆转后仍然存在。

Van Camp, Andrew G; Park, Jiwoon; Ozcelik, Elif; Eskiocak, Onur; Ozler, Kadir A; Papciak, Katie; Subhash, Santhilal; Alwaseem, Hanan; Ergin, Ilgin; Chung, Charlie; Shah, Vyom; Yueh, Brian; Fein, Miriam R; Durmaz, Ceyda; Mozsary, Chris; Kilic, Ece; Garipcan, Aybuke; Damle, Namita; Najjar, Deena; Nelson, Theodore M; Ryon, Krista A; Butler, Daniel J; Patel, Chirag J; Thaiss, Christoph A; Birsoy, Kivanc; Mason, Christopher E; Meydan, Cem; Tierney, Braden T; Beyaz, Semir

Selective Glucocorticoid Receptor Modulators of Immune Checkpoint Function

免疫检查点功能的选择性糖皮质激素受体调节剂

Kobylski, Robin R; Min, Charles K; Nwachukwu, Jerome C; Koenig, Marcel; Zhang, Haotian; Moncada, Lizbeth; Venables, Thomas T; Schell, Bin-Bin; Stein, William J; McCown, Claudia; Schumate, Justin; Bonilla, Emelie; Sobh, Amin; Romero-Toledo, Arantxa; Pipkin, Matthew E; Janiszewska, Michalina; Scampavia, Louis; Spicer, Timothy P; Licht, Jonathan D; Rogatsky, Inez; Kamenecka, Theodore M; Solt, Laura A; Nettles, Kendall W

Scalable and comprehensive mosaic variant calling using DRAGEN

使用 DRAGEN 进行可扩展且全面的嵌合变异检测

Behera, Sairam; Rossi, Massimiliano; Wang, Yina; Izydorczyk, Michal B; Tran, Duke; Dalgard, Clifton L; Kalef-Ezra, Ester; Kottapalli, Kavya; Mehta, Heer; Parnaby, Gavin; Risse-Adams, Oona Shigeno; Scholz, Sonja W; Shen, Helen; Nelson, Theodore M; Visvanath, Arun; Zheng, Xinchang; Doddapaneni, Harsha; Garcia, Thomas; Mason, Christopher E; Proukakis, Christos; Han, James; Mehio, Rami; Catreux, Severine; Sedlazeck, Fritz J

MT-125 inhibits non-muscle myosin IIA and IIB and prolongs survival in glioblastoma

MT-125抑制非肌肉肌球蛋白IIA和IIB,延长胶质母细胞瘤患者的生存期。

Rajappa S Kenchappa,Laszlo Radnai,Erica J Young,Natanael Zarco,Li Lin,Athanassios Dovas,Christian T Meyer,Ashley Haddock,Alice Hall,Katalin Toth,Peter Canoll,Naveen K H Nagaiah,Gavin Rumbaugh,Michael D Cameron,Theodore M Kamenecka,Patrick R Griffin,Courtney A Miller,Steven S Rosenfeld

MT-125 inhibits non-muscle myosin IIA and IIB and prolongs survival in glioblastoma

MT-125抑制非肌肉肌球蛋白IIA和IIB,延长胶质母细胞瘤患者的生存期。

Rajappa S Kenchappa ,Laszlo Radnai ,Erica J Young ,Natanael Zarco ,Li Lin ,Athanassios Dovas ,Christian T Meyer ,Ashley Haddock ,Alice Hall ,Katalin Toth ,Peter Canoll ,Naveen K H Nagaiah ,Gavin Rumbaugh ,Michael D Cameron ,Theodore M Kamenecka ,Patrick R Griffin ,Courtney A Miller ,Steven S Rosenfeld

Development of clinically viable non-muscle myosin II small molecule inhibitors.

开发具有临床应用价值的非肌肉肌球蛋白 II 小分子抑制剂

Radnai Laszlo, Young Erica J, Kikuti Carlos, Toth Katalin, Zhou Minghai, Hafenbreidel Madalyn, Stremel Rebecca F, Lin Li, Pasetto Paolo, Jin Xiaomin, Patel Aagam, Conlon Michael, Briggs Sherri B, Heidsieck Leïla, Sweeney H Lee, Sellers James, Krieger-Burke Teresa, Martin William H, Sisco Jay, Young Steven, Pearson Paul, Rumbaugh Gavin, Araldi Gian Luca, Duddy Steven K, Cameron Michael D, Surman Matthew, Houdusse Anne, Griffin Patrick R, Kamenecka Theodore M, Miller Courtney A

Behavioral Compared With Drug Therapy for Overactive Bladder Symptoms in Parkinson Disease: A Randomized Noninferiority Trial

帕金森病患者膀胱过度活动症的行为疗法与药物疗法比较:一项随机非劣效性试验

Vaughan, Camille P; Morley, James F; Lehosit, Jessica; McGwin, Gerald; Muirhead, Lisa; Khakharia, Anjali; Johnson, Theodore M 2nd; Evatt, Marian L; Sergent, Taressa; Burgio, Kathryn L; Markland, Alayne D

Towards a consensus atlas of human and mouse adipose tissue at single-cell resolution

构建人类和小鼠脂肪组织单细胞分辨率共识图谱

Loft, Anne; Emont, Margo P; Weinstock, Ada; Divoux, Adeline; Ghosh, Adhideb; Wagner, Allon; Hertzel, Ann V; Maniyadath, Babukrishna; Deplancke, Bart; Liu, Boxiang; Scheele, Camilla; Lumeng, Carey; Ding, Changhai; Ma, Chenkai; Wolfrum, Christian; Strieder-Barboza, Clarissa; Li, Congru; Truong, Danh D; Bernlohr, David A; Stener-Victorin, Elisabet; Kershaw, Erin E; Yeger-Lotem, Esti; Shamsi, Farnaz; Hui, Hannah X; Camara, Henrique; Zhong, Jiawei; Kalucka, Joanna; Ludwig, Joseph A; Semon, Julie A; Jalkanen, Jutta; Whytock, Katie L; Dumont, Kyle D; Sparks, Lauren M; Muir, Lindsey A; Fang, Lingzhao; Massier, Lucas; Saraiva, Luis R; Beyer, Marc D; Jeschke, Marc G; Mori, Marcelo A; Boroni, Mariana; Walsh, Martin J; Patti, Mary-Elizabeth; Lynes, Matthew D; Blüher, Matthias; Rydén, Mikael; Hamda, Natnael; Solimini, Nicole L; Mejhert, Niklas; Gao, Peng; Gupta, Rana K; Murphy, Rinki; Pirouzpanah, Saeed; Corvera, Silvia; Tang, Su'an; Das, Swapan K; Schmidt, Søren F; Zhang, Tao; Nelson, Theodore M; O'Sullivan, Timothy E; Efthymiou, Vissarion; Wang, Wenjing; Tong, Yihan; Tseng, Yu-Hua; Mandrup, Susanne; Rosen, Evan D