日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Relieving DYRK1A repression of MKL1 confers an adult-like phenotype to human infantile megakaryocytes

解除 DYRK1A 对 MKL1 的抑制可使人类婴儿巨核细胞呈现成人样表型

Kamaleldin E Elagib, Ashton Brock, Cara M Clementelli, Goar Mosoyan, Lorrie L Delehanty, Ranjit K Sahu, Alexandra Pacheco-Benichou, Corinne Fruit, Thierry Besson, Stephan W Morris, Koji Eto, Chintan Jobaliya, Deborah L French, Paul Gadue, Sandeep Singh, Xinrui Shi, Fujun Qin, Robert Cornelison, Hui

Therapeutic antibody glycosylation impacts antigen recognition and immunogenicity

治疗性抗体糖基化影响抗原识别和免疫原性

Babette Wolf, Mateusz Piksa, Isabelle Beley, Agnes Patoux, Thierry Besson, Valerie Cordier, Bernd Voedisch, Patrick Schindler, Daniela Stöllner, Ludovic Perrot, Stephan von Gunten, Dominique Brees, Michael Kammüller

Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core

直接获取具有简单二氢喹啉核心的新型双重 DYRK1A/CLK1 抑制剂

Mihaela-Liliana Ţînţaş, Ludovic Peauger, Florent Alix, Cyril Papamicaël, Thierry Besson, Jana Sopková-de Oliveira Santos, Vincent Gembus, Vincent Levacher

DYRK1A regulates B cell acute lymphoblastic leukemia through phosphorylation of FOXO1 and STAT3

DYRK1A 通过 FOXO1 和 STAT3 的磷酸化来调节 B 细胞急性淋巴细胞白血病

Rahul S Bhansali, Malini Rammohan, Paul Lee, Anouchka P Laurent, Qiang Wen, Praveen Suraneni, Bon Ham Yip, Yi-Chien Tsai, Silvia Jenni, Beat Bornhauser, Aurélie Siret, Corinne Fruit, Alexandra Pacheco-Benichou, Ethan Harris, Thierry Besson, Benjamin J Thompson, Young Ah Goo, Nobuko Hijiya, Maria Vil

Microwave-Assisted Synthesis of Potential Bioactive Benzo-, Pyrido- or Pyrazino-thieno[3,2- d]pyrimidin-4-amine Analogs of MPC-6827

微波辅助合成具有潜在生物活性的苯并、吡啶并或吡嗪并噻吩并[3,2- d]嘧啶-4-胺类 MPC-6827 类似物

Yvonnick Loidreau, Marie-Renée Nourrisson, Corinne Fruit, Cécile Corbière, Pascal Marchand, Thierry Besson

Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4- f]quinazolin-9(8 H)-one, a Promising Inhibitor of DYRK1A

8-环丙基-2-(吡啶-3-基)噻唑并[5,4- f]喹唑啉-9(8 H)-酮(一种有前途的 DYRK1A 抑制剂)的生物学特性

Corinne Fruit, Florence Couly, Rahul Bhansali, Malini Rammohan, Mattias F Lindberg, John D Crispino, Laurent Meijer, Thierry Besson

Polymeric nanocapsules prevent oxidation of core-loaded molecules: evidence based on the effects of docosahexaenoic acid and neuroprostane on breast cancer cells proliferation.

聚合物纳米胶囊可防止核心负载分子的氧化:基于二十二碳六烯酸和神经前列腺素对乳腺癌细胞增殖的影响的证据

Roy Jérôme, Oliveira Liliam Teixeira, Oger Camille, Galano Jean-Marie, Bultel-Poncé Valerie, Richard Sylvain, Guimaraes Andrea Grabe, Vilela José Mário Carneiro, Andrade Margareth Spangler, Durand Thierry, Besson Pierre, Mosqueira Vanessa Carla Furtado, Le Guennec Jean-Yves

DYRK1A controls the transition from proliferation to quiescence during lymphoid development by destabilizing Cyclin D3

DYRK1A 通过破坏 Cyclin D3 来控制淋巴发育过程中从增殖到静止的转变

Benjamin J Thompson, Rahul Bhansali, Lauren Diebold, Daniel E Cook, Lindsay Stolzenburg, Anne-Sophie Casagrande, Thierry Besson, Bertrand Leblond, Laurent Désiré, Sébastien Malinge, John D Crispino