Structure-Guided Design and Synthesis of a Pyridazinone Series of Trypanosoma cruzi Proteasome Inhibitors
基于结构的锥虫蛋白酶体抑制剂哒嗪酮系列的设计与合成
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.3c00582
Thomas, Michael G; McGonagle, Kate; Rowland, Paul; Robinson, David A; Dodd, Peter G; Camino-Díaz, Isabel; Campbell, Lorna; Cantizani, Juan; Castañeda, Pablo; Conn, Daniel; Craggs, Peter D; Edwards, Darren; Ferguson, Liam; Fosberry, Andrew; Frame, Laura; Goswami, Panchali; Hu, Xiao; Korczynska, Justyna; MacLean, Lorna; Martin, Julio; Mutter, Nicole; Osuna-Cabello, Maria; Paterson, Christy; Peña, Imanol; Pinto, Erika G; Pont, Caterina; Riley, Jennifer; Shishikura, Yoko; Simeons, Frederick R C; Stojanovski, Laste; Thomas, John; Wrobel, Karolina; Young, Robert J; Zmuda, Filip; Zuccotto, Fabio; Read, Kevin D; Gilbert, Ian H; Marco, Maria; Miles, Timothy J; Manzano, Pilar; De Rycker, Manu