日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Gq activity- and β-arrestin-1 scaffolding-mediated ADGRG2/CFTR coupling are required for male fertility

更正:Gq活性和β-arrestin-1支架介导的ADGRG2/CFTR偶联是男性生育力所必需的。

Zhang, Dao-Lai; Sun, Yu-Jing; Ma, Ming-Liang; Wang, Yi-Jing; Lin, Hui; Li, Rui-Rui; Liang, Zong-Lai; Gao, Yuan; Yang, Zhao; He, Dong-Fang; Lin, Amy; Mo, Hui; Lu, Yu-Jing; Li, Mengjing; Kong, Wei; Chung, Ka Young; Yi, Fan; Li, Jian-Yuan; Qin, Ying-Ying; Li, Jingxin; Thomsen, Alex R B; Kahsai, Alem W; Chen, Zi-Jiang; Xu, Zhi-Gang; Liu, Mingyao; Li, Dali; Yu, Xiao; Sun, Jin-Peng

Endosomal chemokine receptor signalosomes regulate central mechanisms underlying cell migration.

内体趋化因子受体信号体调节细胞迁移的核心机制

Hahn Hyunggu, Daly Carole, Little John 4th, Perry-Hauser Nicole A, Flores-Espinoza Emmanuel, Inoue Asuka, Plouffe Bianca, Thomsen Alex R B

Artificial Intelligence: A New Tool for Structure-Based G Protein-Coupled Receptor Drug Discovery

人工智能:一种基于结构的G蛋白偶联受体药物发现新工具

Chung, Jason; Hahn, Hyunggu; Flores-Espinoza, Emmanuel; Thomsen, Alex R B

Small-molecule modulation of β-arrestins

小分子对β-arrestin的调控

Kahsai, Alem W; Pakharukova, Natalia; Kwon, Henry Y; Shah, Kunal S; Liang-Lin, Jason G; Del Real, Caroline T; Shim, Paul J; Lee, Mason A; Ngo, Van A; Shreiber, Bowie N; Liu, Samuel; Schwalb, Allison M; Espinoza, Emmanuel F; Thomas, Brittany N; Kunzle, Cal A; Smith, Jeffrey S; Wang, Jialu; Kim, Jihee; Zhang, Xingdong; Rockman, Howard A; Thomsen, Alex R B; Rein, Lindsay A M; Shi, Lei; Ahn, Seungkirl; Masoudi, Ali; Lefkowitz, Robert J

Plasma membrane rather than endosomal Gq signaling drives transcriptional activity by the viral chemokine receptor US28 in glioblastoma

在胶质母细胞瘤中,病毒趋化因子受体US28的转录活性是由质膜而非内体Gq信号传导驱动的。

Daly, Carole; Wright, Adam; Heukers, Raimond; McKee, Chloe M; Coll, Rebecca C; Evergren, Emma; Smit, Martine J; Thomsen, Alex R B; Plouffe, Bianca

Beneath the surface: endosomal GPCR signaling

表面之下:内体GPCR信号传导

Flores-Espinoza, Emmanuel; Thomsen, Alex R B

Label-Free Dynamic Mass Redistribution Assay To Characterize Holistic Chemokine Receptor Pharmacology in Neutrophils

无标记动态质量重分布分析法用于表征中性粒细胞中趋化因子受体的整体药理学

Thomsen, Alex R B

GPCRs and β-arrestins - an on-off relationship

GPCRs和β-arrestin——一种开关关系

Thomsen, Alex R B

Therapeutic antagonism of the neurokinin 1 receptor in endosomes provides sustained pain relief

内体中神经激肽1受体的治疗性拮抗作用可提供持续的镇痛效果

Hegron, Alan; Peach, Chloe J; Tonello, Raquel; Seemann, Philipp; Teng, Shavonne; Latorre, Rocco; Huebner, Harald; Weikert, Dorothee; Rientjes, Jeanette; Veldhuis, Nicholas A; Poole, Daniel P; Jensen, Dane D; Thomsen, Alex R B; Schmidt, Brian L; Imlach, Wendy L; Gmeiner, Peter; Bunnett, Nigel W

Emerging Role of Compartmentalized G Protein-Coupled Receptor Signaling in the Cardiovascular Field

区室化G蛋白偶联受体信号传导在心血管领域的新兴作用

Plouffe, Bianca; Thomsen, Alex R B; Irannejad, Roshanak