日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Ester Prodrug NLRP3 Inflammasome Inhibitor NT-0796 is Brain Active due to Activation by Local Expression of Carboxylesterase-1

酯类前药 NLRP3 炎症小体抑制剂 NT-0796 因羧酸酯酶-1 的局部表达而被激活,从而具有脑活性。

Digby, Zsofia; Diamond, Christine; Wescott, Heather; Smolak, Pam; Thornton, Peter; Lindsay, Nicola; Gabel, Christopher A; Clarke, Nicholas; Watt, Alan P

Efficacy of MEDI0618, a pH-dependent monoclonal antibody targeting PAR2, in preclinical models of migraine.

MEDI0618 是一种 pH 依赖性单克隆抗体,靶向 PAR2,在偏头痛的临床前模型中疗效

Kopruszinski Caroline M, Linley John E, Thornton Peter, Walker Alison S, Newton Philip, Podichetty Sadhana, Ruparel Radhey Hemendra, Moreira de Souza Luiz Henrique, Navratilova Edita, Meno-Tetang Guy, Gurrell Ian, Dodick David W, Dobson Claire, Chessell Tharani, Porreca Frank, Chessell Iain

Anti-Neuroinflammatory and Anti-Inflammatory Effects of the NLRP3 Inhibitor NT-0796 in Subjects with Parkinson's Disease

NLRP3抑制剂NT-0796在帕金森病患者中的抗神经炎症和抗炎作用

Clarke, Nicholas; Thornton, Peter; Reader, Valérie; Lindsay, Nicola; Digby, Zsofia; Mullen, Bianca; Gorman, Michelle; Jacobson, Eric; Langdon, Grant; Johnstone, Hilary; Wheeler, Alistair; Watt, Alan P

A high resolution, gridded product for vapor pressure deficit using Daymet

使用 Daymet 生成高分辨率网格化蒸汽压亏缺产品

Corak, Nicholas K; Thornton, Peter E; Lowman, Lauren E L

Profile of NT-0527, a brain penetrant NLRP3 Inflammasome inhibitor suitable as an in vivo tool compound for neuroinflammatory disorders.

NT-0527 是一种可穿透血脑屏障的 NLRP3 炎症小体抑制剂,适用于作为神经炎症性疾病的体内治疗药物

Harrison David, Billinton Andy, Bock Mark G, Clarke Nicholas P, Digby Zsofia, Gabel Christopher A, Lindsay Nicola, Reader Valérie, Scanlon Jane, Smolak Pamela, Thornton Peter, Wescott Heather, Watt Alan P

The NLRP3 inhibitor NT-0796 enhances and sustains GLP-1R agonist-mediated weight loss in a murine diet-induced obesity model

NLRP3抑制剂NT-0796可增强并维持GLP-1R激动剂介导的小鼠饮食诱导肥胖模型中的体重减轻。

Thornton, Peter; Reader, Valérie; Digby, Zsofia; Doedens, John; Lindsay, Nicola; Clarke, Nicholas; Watt, Alan P

Thermal, water, and land cover factors led to contrasting urban and rural vegetation resilience to extreme hot months

温度、水文和土地覆盖因素导致城市和乡村植被对极端高温月份的适应能力存在差异。

Wang, Yaoping; Mao, Jiafu; Brelsford, Christa M; Ricciuto, Daniel M; Yuan, Fengming; Shi, Xiaoying; Rastogi, Deeksha; Mayes, Melanie M; Kao, Shih-Chieh; Warren, Jeffrey M; Griffiths, Natalie A; Cheng, Xinghua; Weston, David J; Zhou, Yuyu; Gu, Lianhong; Thornton, Peter E

Quantifying the drivers and predictability of seasonal changes in African fire

量化非洲火灾季节性变化的驱动因素和可预测性

Yu, Yan; Mao, Jiafu; Thornton, Peter E; Notaro, Michael; Wullschleger, Stan D; Shi, Xiaoying; Hoffman, Forrest M; Wang, Yaoping

Representing the function and sensitivity of coastal interfaces in Earth system models

在地球系统模型中表征海岸界面的功能和敏感性

Ward, Nicholas D; Megonigal, J Patrick; Bond-Lamberty, Ben; Bailey, Vanessa L; Butman, David; Canuel, Elizabeth A; Diefenderfer, Heida; Ganju, Neil K; Goñi, Miguel A; Graham, Emily B; Hopkinson, Charles S; Khangaonkar, Tarang; Langley, J Adam; McDowell, Nate G; Myers-Pigg, Allison N; Neumann, Rebecca B; Osburn, Christopher L; Price, René M; Rowland, Joel; Sengupta, Aditi; Simard, Marc; Thornton, Peter E; Tzortziou, Maria; Vargas, Rodrigo; Weisenhorn, Pamela B; Windham-Myers, Lisamarie

Alder Distribution and Expansion Across a Tundra Hillslope: Implications for Local N Cycling

赤杨在苔原山坡上的分布和扩张:对局部氮循环的影响

Salmon, Verity G; Breen, Amy L; Kumar, Jitendra; Lara, Mark J; Thornton, Peter E; Wullschleger, Stan D; Iversen, Colleen M