日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

HR-MS Analysis of the Covalent Binding of Edaravone to 5-Formylpyrimidine Bases and a DNA Oligonucleotide Containing a 5-Formylcytidine Residue

利用高分辨率质谱分析依达拉奉与5-甲酰嘧啶碱基和含有5-甲酰胞苷残基的DNA寡核苷酸的共价结合

Regnault, Romain; Kouach, Mostafa; Goossens, Laurence; Thuru, Xavier; Bailly, Christian; Goossens, Jean-François

MYC dependency in GLS1 and NAMPT is a therapeutic vulnerability in multiple myeloma

GLS1 和 NAMPT 中的 MYC 依赖性是多发性骨髓瘤的治疗弱点

Lama Hasan Bou Issa, Léa Fléchon, William Laine, Aicha Ouelkdite, Silvia Gaggero, Adeline Cozzani, Remi Tilmont, Paul Chauvet, Nicolas Gower, Romanos Sklavenitis-Pistofidis, Carine Brinster, Xavier Thuru, Yasmine Touil, Bruno Quesnel, Suman Mitra, Irene M Ghobrial, Jérôme Kluza, Salomon Manier

Targeting of Tetraspanin CD81 with Monoclonal Antibodies and Small Molecules to Combat Cancers and Viral Diseases

利用单克隆抗体和小分子靶向四跨膜蛋白CD81对抗癌症和病毒性疾病

Bailly, Christian; Thuru, Xavier

Novel PD-L1-Targeted Phenyl-Pyrazolone Derivatives with Antioxidant Properties

具有抗氧化特性的新型 PD-L1 靶向苯基吡唑酮衍生物

Romain Regnault, Frédérique Klupsch, Hassiba El-Bouazzati, Romain Magnez, Raphaël Le Biannic, Natascha Leleu-Chavain, Hania Ahouari, Hervé Vezin, Régis Millet, Jean-François Goossens, Xavier Thuru, Christian Bailly

A Potential Off-Target Effect of the Wnt/β-Catenin Inhibitor KYA1797K: PD-L1 Binding and Checkpoint Inhibition.

Wnt/β-catenin抑制剂KYA1797K的潜在脱靶效应:PD-L1结合和检查点抑制

Thuru Xavier, Magnez Romain, Vergoten Gérard, Bailly Christian

IL-2 is inactivated by the acidic pH environment of tumors enabling engineering of a pH-selective mutein

IL-2 在肿瘤的酸性 pH 环境中失活,因此可以设计出 pH 选择性突变蛋白

Silvia Gaggero, Jonathan Martinez-Fabregas, Adeline Cozzani, Paul K Fyfe, Malo Leprohon, Jie Yang, F Emil Thomasen, Hauke Winkelmann, Romain Magnez, Alberto G Conti, Stephan Wilmes, Elizabeth Pohler, Manuel van Gijsel Bonnello, Xavier Thuru, Bruno Quesnel, Fabrice Soncin, Jacob Piehler, Kresten Lind

Direct interaction of TrkA/CD44v3 is essential for NGF-promoted aggressiveness of breast cancer cells

TrkA/CD44v3 的直接相互作用对于 NGF 促进乳腺癌细胞的侵袭性至关重要

Sarah Trouvilliez #, Julien Cicero #, Romain Lévêque, Léo Aubert, Cyril Corbet, Alexandre Van Outryve, Karolin Streule, Pierre-Olivier Angrand, Pamela Völkel, Romain Magnez, Guillaume Brysbaert, Caroline Mysiorek, Fabien Gosselet, Roland Bourette, Eric Adriaenssens, Xavier Thuru, Chann Lagadec, Jérô

Pyrazolones as inhibitors of immune checkpoint blocking the PD-1/PD-L1 interaction

吡唑酮类药物作为免疫检查点抑制剂阻断 PD-1/PD-L1 相互作用

Raphaël Le Biannic, Romain Magnez, Frédérique Klupsch, Natascha Leleu-Chavain, Bryan Thiroux, Morgane Tardy, Hassiba El Bouazzati, Xavier Dezitter, Nicolas Renault, Gérard Vergoten, Christian Bailly, Bruno Quesnel, Xavier Thuru, Régis Millet

A Phosphosite Mutant Approach on LRRK2 Links Phosphorylation and Dephosphorylation to Protective and Deleterious Markers, Respectively

LRRK2磷酸化位点突变方法将磷酸化和去磷酸化分别与保护性和有害性标记联系起来

Marchand, Antoine; Sarchione, Alessia; Athanasopoulos, Panagiotis S; Roy, Hélène Bauderlique-Le; Goveas, Liesel; Magnez, Romain; Drouyer, Matthieu; Emanuele, Marco; Ho, Franz Y; Liberelle, Maxime; Melnyk, Patricia; Lebègue, Nicolas; Thuru, Xavier; Nichols, R Jeremy; Greggio, Elisa; Kortholt, Arjan; Galli, Thierry; Chartier-Harlin, Marie-Christine; Taymans, Jean-Marc

Microscale Thermophoresis as a Tool to Study Protein Interactions and Their Implication in Human Diseases

利用微尺度热泳技术研究蛋白质相互作用及其在人类疾病中的作用

Magnez, Romain; Bailly, Christian; Thuru, Xavier