日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Library docking for Cannabinoid-2 Receptor ligands

大麻素-2受体配体的库对接

Rachman, Moira M; Iliopoulos-Tsoutsouvas, Christos; Sacco, Michael D; Xu, Xinyu; Wu, Cheng-Guo; Santos, Emma; Glenn, Isabella S; Paris, Lu; Cahill, Michelle K; Ganapathy, Suthakar; Tummino, Tia A; Moroz, Yurii S; Radchenko, Dmytro S; Okorie, Meri; Tawfik, Vivianne; Irwin, John J; Makriyannis, Alexandros; Skiniotis, Georgios; Shoichet, Brian K

Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects.

针对副作用较小的 1 型大麻素受体激动剂的虚拟库对接

Tummino Tia A, Iliopoulos-Tsoutsouvas Christos, Braz Joao M, O'Brien Evan S, Stein Reed M, Craik Veronica, Tran Ngan K, Ganapathy Suthakar, Liu Fangyu, Shiimura Yuki, Tong Fei, Ho Thanh C, Radchenko Dmytro S, Moroz Yurii S, Rosado Sian Rodriguez, Bhardwaj Karnika, Benitez Jorge, Liu Yongfeng, Kandasamy Herthana, Normand Claire, Semache Meriem, Sabbagh Laurent, Glenn Isabella, Irwin John J, Kumar Kaavya Krishna, Makriyannis Alexandros, Basbaum Allan I, Shoichet Brian K

A Database for Large-Scale Docking and Experimental Results

大规模对接和实验结果数据库

Hall, Brendan W; Tummino, Tia A; Tang, Khanh; Mailhot, Olivier; Castanon, Mar; Irwin, John J; Shoichet, Brian K

Assessing Antibacterial Properties of Copper Oxide Nanomaterials on Gut-Relevant Bacteria In Vitro: A Multifaceted Approach

体外评估氧化铜纳米材料对肠道相关细菌的抗菌性能:一种多方面方法

Wardlaw, Tia A; Masri, Abdulkader; Brown, David M; Johnston, Helinor J

Insulin facilitates entry of calcium ions into human and murine erythrocytes via Piezo1: a newly identified mechanism with implications for type 2 diabetes.

胰岛素通过 Piezo1 促进钙离子进入人和小鼠的红细胞:这是一种新发现的机制,对 2 型糖尿病具有重要意义。

Kuck Lennart, Griffith Tia A, McNamee Antony P, Peart Jason N, Wilson John H, Sharma Ajay, Sharma Lavanya A, Robertson Kai, Du Toit Eugene F, Simmonds Michael J

The Juvenile Parkinson's Disease Mutation C212Y Impairs Mitochondrial Homeostasis in a Caenorhabditis elegans Model.

幼年帕金森病突变 C212Y 会损害秀丽隐杆线虫模型中的线粒体稳态

Spector Eyal, Michaeli Lirin, Nitzan Anat, Grobe Hanna, Axel Gabriel, Abu-Shach Ulrike Bening, Zinger Hen, Carvalho Cátia A, Zaidel-Bar Ronen, Broday Limor

Adherens junctions limit septate junction length in Drosophila midgut enterocytes but are not required for polarity.

粘着连接限制了果蝇中肠肠细胞的隔膜连接长度,但对极性并非必需

Carvalho Cátia A, Tame Mihoko A, St Johnston Daniel

Vole hunting: novel predatory and carnivorous behavior by California ground squirrels

加州地松鼠捕猎田鼠:新颖的捕食和食肉行为

Smith, Jennifer E; Ingbretson, Joey E; Miner, Mackenzie M; Oestreicher, Ella C; Podas, Mari L; Ravara, Tia A; Teles, Lupin M L; Wahl, Jada C; Todd, Lucy M; Wild, Sonja

A database for large-scale docking and experimental results

一个用于大规模对接和实验结果的数据库

Hall, Brendan W; Tummino, Tia A; Tang, Khanh; Irwin, John J; Shoichet, Brian K

AlphaFold2 structures guide prospective ligand discovery

AlphaFold2结构指导潜在配体的发现

Lyu, Jiankun; Kapolka, Nicholas; Gumpper, Ryan; Alon, Assaf; Wang, Liang; Jain, Manish K; Barros-Álvarez, Ximena; Sakamoto, Kensuke; Kim, Yoojoong; DiBerto, Jeffrey; Kim, Kuglae; Glenn, Isabella S; Tummino, Tia A; Huang, Sijie; Irwin, John J; Tarkhanova, Olga O; Moroz, Yurii; Skiniotis, Georgios; Kruse, Andrew C; Shoichet, Brian K; Roth, Bryan L