日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Drugging the intrinsically disordered transactivation domain of androgen receptor

药物靶向雄激素受体固有无序的转录激活结构域

Obst, Jon K; Banuelos, Carmen A; Jian, Kunzhong; Tien, Amy H; Shkrabak, Oleksandr A; Wang, Jun; Mawji, Nasrin R; Tam, Teresa; Vuckovic, Marija; Williams, David E; Rogalski, Jason C; Yuan, Xiaojing; Strynadka, Natalie C J; Andersen, Raymond J; Sadar, Marianne D

Treatments Targeting the Androgen Receptor and Its Splice Variants in Breast Cancer.

针对乳腺癌中雄激素受体及其剪接变体的治疗方法

Tien Amy H, Sadar Marianne D

Inhibitors of the transactivation domain of androgen receptor as a therapy for prostate cancer

雄激素受体反式激活结构域抑制剂作为前列腺癌的治疗方法

Obst, Jon K; Tien, Amy H; Setiawan, Josie C; Deneault, Lauren F; Sadar, Marianne D

Keys to unlock androgen receptor translocation

解锁雄激素受体易位的关键

Tien, Amy H; Sadar, Marianne D

Order within a Disordered Structure

无序结构中的秩序

Tien, Amy H; Sadar, Marianne D

Characterization of niphatenones that inhibit androgen receptor N-terminal domain.

对抑制雄激素受体N端结构域的尼法酮进行表征

Banuelos Carmen A, Lal Aaron, Tien Amy H, Shah Neel, Yang Yu Chi, Mawji Nasrin R, Meimetis Labros G, Park Jacob, Kunzhong Jian, Andersen Raymond J, Sadar Marianne D

An androgen receptor N-terminal domain antagonist for treating prostate cancer.

用于治疗前列腺癌的雄激素受体 N 端结构域拮抗剂

Myung Jae-Kyung, Banuelos Carmen A, Fernandez Javier Garcia, Mawji Nasrin R, Wang Jun, Tien Amy H, Yang Yu Chi, Tavakoli Iran, Haile Simon, Watt Kate, McEwan Iain J, Plymate Stephen, Andersen Raymond J, Sadar Marianne D

Spongian diterpenoids inhibit androgen receptor activity

海绵二萜类化合物抑制雄激素受体活性

Yang, Yu Chi; Meimetis, Labros G; Tien, Amy H; Mawji, Nasrin R; Carr, Gavin; Wang, Jun; Andersen, Raymond J; Sadar, Marianne D