日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Divergent FOXA1 mutations drive prostate tumorigenesis and therapy-resistant cellular plasticity.

FOXA1 基因突变导致前列腺肿瘤发生和细胞耐药性

Eyunni Sanjana, Mannan Rahul, Zhang Yuping, Young Eleanor, Zhang Qiuyang, Luo Jie, Pang Matthew, Mahapatra Somnath, Tien Jean Ching-Yi, George James M, Jaber Mustapha, Hakkani Hamzah, Carson Sandra E, Todd Abigail J, Hosseini Noshad, Gondal Mahnoor, Rebernick Ryan J, Cao Xuhong, Su Fengyun, Wang Rui, Mehra Rohit, Li Jing, Cieslik Marcin, Chinnaiyan Arul M, Parolia Abhijit

Defining CDK12 as a tumor suppressor and therapeutic target in mouse models of tubo-ovarian high-grade serous carcinoma.

在输卵管卵巢高级别浆液性癌小鼠模型中,将 CDK12 定义为肿瘤抑制因子和治疗靶点

Tien Jean Ching-Yi, Zhai Yali, Wu Rong, Zhang Yuping, Chang Yu, Cheng Yunhui, Todd Abigail J, Wheeler Christina E, Li Shuqin, Mannan Rahul, Cheng Caleb, Magnuson Brian, Cruz Gabriel, Cao Yizhi, Mahapatra Somnath, Stolfi Carmine, Cao Xuhong, Su Fengyun, Wang Rui, Yang Jianzhang, Zhou Licheng, Qiao Yuanyuan, Xiao Lanbo, Cieslik Marcin, Wang Xiaoju, Wang Zhen, Chou Jonathan, Fearon Eric R, Ding Ke, Cho Kathleen R, Chinnaiyan Arul M

Discovery of YJZ5118: A Potent and Highly Selective Irreversible CDK12/13 Inhibitor with Synergistic Effects in Combination with Akt Inhibition.

YJZ5118 的发现:一种强效且高选择性的不可逆 CDK12/13 抑制剂,与 Akt 抑制剂联合使用具有协同效应

Yang Jianzhang, Chang Yu, Zhou Kaijie, Huang Weixue, Tien Jean Ching-Yi, Zhang Pujuan, Liu Wenyan, Zhou Licheng, Zhou Yang, Ren Xiaomei, Mannan Rahul, Mahapatra Somnath, Zhang Yuping, Hamadeh Rudana, Ervine Grafton, Wang Zhen, Wang George Xiaoju, Chinnaiyan Arul M, Ding Ke

An essential role for Argonaute 2 in EGFR-KRAS signaling in pancreatic cancer development

Argonaute 2 在 EGFR-KRAS 信号通路中对胰腺癌的发生发展起着至关重要的作用

Shankar, Sunita; Tien, Jean Ching-Yi; Siebenaler, Ronald F; Chugh, Seema; Dommeti, Vijaya L; Zelenka-Wang, Sylvia; Wang, Xiao-Ming; Apel, Ingrid J; Waninger, Jessica; Eyunni, Sanjana; Xu, Alice; Mody, Malay; Goodrum, Andrew; Zhang, Yuping; Tesmer, John J; Mannan, Rahul; Cao, Xuhong; Vats, Pankaj; Pitchiaya, Sethuramasundaram; Ellison, Stephanie J; Shi, Jiaqi; Kumar-Sinha, Chandan; Crawford, Howard C; Chinnaiyan, Arul M

The function of steroid receptor coactivator-1 in normal tissues and cancer

类固醇受体共激活因子-1在正常组织和癌症中的功能

Walsh, Claire A; Qin, Li; Tien, Jean Ching-Yi; Young, Leonie S; Xu, Jianming

The role of SRC-1 in murine prostate cancinogenesis is nonessential due to a possible compensation of SRC-3/AIB1 overexpression

由于SRC-3/AIB1过表达可能起到补偿作用,SRC-1在小鼠前列腺癌发生中的作用并非必需。

Tien, Jean Ching-Yi; Zhou, Suoling; Xu, Jianming

Genetic ablation of the amplified-in-breast cancer 1 inhibits spontaneous prostate cancer progression in mice

基因敲除乳腺癌扩增基因1可抑制小鼠前列腺癌的自发进展。

Chung, Arthur C-K; Zhou, Suoling; Liao, Lan; Tien, Jean Ching-Yi; Greenberg, Norman M; Xu, Jianming