日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Ex vivo and in vivo HIV-1 latency reversal by "Mukungulu," a protein kinase C-activating African medicinal plant extract

非洲药用植物提取物“Mukungulu”可激活蛋白激酶C,并能逆转体外和体内HIV-1潜伏感染。

Richard, Khumoekae; Yuan, Zhe; Tang, Hsin-Yao; Goldman, Aaron R; Kuthu, Riza; Raphane, Boingotlo; Register, Emery T; Sharma, Paridhima; Ross, Brian N; Morris, Jessicamarie; Williams, David E; Cheney, Carol; Wu, Guoxin; Mounzer, Karam; Laird, Gregory M; Zuck, Paul; Andersen, Raymond J; Simonambango, Sundana; Andrae-Marobela, Kerstin; Tietjen, Ian; Montaner, Luis J

A high-throughput, microplate reader-based method to monitor in vitro HIV latency reversal in the absence of flow cytometry

一种基于高通量微孔板读数仪的方法,用于在不使用流式细胞术的情况下监测体外HIV潜伏期逆转。

Nkwelle, Chantal Emade; Stephens, Unique; Liang, Kimberly; Cassel, Joel; Salvino, Joseph M; Montaner, Luis J; Ndip, Roland N; Esemu, Seraphine N; Ntie-Kang, Fidele; Tietjen, Ian

Metabolomic Analysis and Antiviral Screening of a Marine Algae Library Yield Jobosic Acid (2,5-Dimethyltetradecanoic Acid) as a Selective Inhibitor of SARS-CoV-2.

对海洋藻类库进行代谢组学分析和抗病毒筛选,发现乔博西酸(2,5-二甲基十四烷酸)是SARS-CoV-2的选择性抑制剂

Matos-Hernández Marie L, Samples Robert, Dyer Grayce, Casimir Montán Victoria M, Morales-Colón Chris A, Salvino Joseph M, Montaner Luis J, Cassel Joel A, Messick Troy E, Tietjen Ian, Caro-Diaz Eduardo J E

Design, synthesis, and biochemical and computational screening of novel oxindole derivatives as inhibitors of Aurora A kinase and SARS-CoV-2 spike/host ACE2 interaction

设计、合成并进行生化和计算机筛选,以研究新型吲哚酮衍生物作为 Aurora A 激酶和 SARS-CoV-2 刺突蛋白/宿主 ACE2 相互作用抑制剂的活性。

Eni, Donatus B; Cassel, Joel; Namba-Nzanguim, Cyril T; Simoben, Conrad V; Tietjen, Ian; Akunuri, Ravikumar; Salvino, Joseph M; Ntie-Kang, Fidele

Corrigendum to "Discovery of lead natural products for developing pan-SARS-CoV-2 therapeutics" "Antiviral Research 209 (2023)/105484"

对“发现用于开发泛SARS-CoV-2疗法的先导天然产物”“抗病毒研究209 (2023)/105484”的更正

Perez-Vargas, Jimena; Shapira, Tirosh; Olmstead, Andrea D; Villanueva, Ivan; Thompson, Connor A H; Ennis, Siobhan; Gao, Guang; De Guzman, Joshua; Williams, David E; Wang, Meng; Chin, Aaleigha; Bautista-Sanchez, Diana; Agafitei, Olga; Levett, Paul; Xie, Xuping; Nuzzo, Genoveffa; Freire, Vitor F; Quintana-Bulla, Jairo I; Bernardi, Darlon I; Gubiani, Juliana R; Suthiphasilp, Virayu; Raksat, Achara; Meesakul, Pornphimol; Polbuppha, Isaraporn; Cheenpracha, Sarot; Jaidee, Wuttichai; Kanokmedhakul, Kwanjai; Yenjai, Chavi; Chaiyosang, Boonyanoot; Teles, Helder Lopes; Manzo, Emiliano; Fontana, Angelo; Leduc, Richard; Boudreault, Pierre-Luc; Berlinck, Roberto G S; Laphookhieo, Surat; Kanokmedhakul, Somdej; Tietjen, Ian; Cherkasov, Artem; Krajden, Mel; Nabi, Ivan Robert; Niikura, Masahiro; Shi, Pei-Yong; Andersen, Raymond J; Jean, François

Thorectidiol A Isolated from the Marine Sponge Dactylospongia elegans Disrupts Interactions of the SARS-CoV-2 Spike Receptor Binding Domain with the Host ACE2 Receptor

从海洋海绵 Dactylospongia elegans 中分离得到的 Thorectidiol A 可破坏 SARS-CoV-2 刺突蛋白受体结合域与宿主 ACE2 受体的相互作用

Williams, David E; Cassel, Joel; Zhu, Jin-Lin; Yang, Jian-Xiong; de Voogd, Nicole J; Matainaho, Teatulohi; Salvino, Joseph M; Wang, Yan Alexander; Montaner, Luis J; Tietjen, Ian; Andersen, Raymond J

Virtual Screening Identifies Chebulagic Acid as an Inhibitor of the M2(S31N) Viral Ion Channel and Influenza A Virus

虚拟筛选发现诃子酸是M2(S31N)病毒离子通道和甲型流感病毒的抑制剂

Duncan, Maggie C; Onguéné, Pascal Amoa; Kihara, Ibuki; Nebangwa, Derrick N; Naidu, Maya E; Williams, David E; Balgi, Aruna D; Andrae-Marobela, Kerstin; Roberge, Michel; Andersen, Raymond J; Niikura, Masahiro; Ntie-Kang, Fidele; Tietjen, Ian

Put a cork in it: Plugging the M2 viral ion channel to sink influenza

堵住它:堵塞 M2 病毒离子通道以阻止流感

Jalily, Pouria H; Duncan, Maggie C; Fedida, David; Wang, Jun; Tietjen, Ian

Capillasterin A, a Novel Pyrano[2,3-f]chromene from the Australian Crinoid Capillaster multiradiatus

来自澳大利亚海百合多辐射海百合(Capillaster multiradiatus)的新型吡喃并[2,3-f]色烯化合物Capillasterin A

Lum, Kah Yean; Carroll, Anthony R; Ekins, Merrick G; Read, Silven; Haq, Zahra; Tietjen, Ian; St John, James; Davis, Rohan A

Binding and Proton Blockage by Amantadine Variants of the Influenza M2(WT) and M2(S31N) Explained

金刚烷胺变体与流感病毒M2(WT)和M2(S31N)的结合及质子阻断机制详解

Tzitzoglaki, Christina; Wright, Anna; Freudenberger, Kathrin; Hoffmann, Anja; Tietjen, Ian; Stylianakis, Ioannis; Kolarov, Felix; Fedida, David; Schmidtke, Michaela; Gauglitz, Günter; Cross, Timothy A; Kolocouris, Antonios