日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Epi-Cyclophellitol Cyclosulfate, a Mechanism-Based Endoplasmic Reticulum α-Glucosidase II Inhibitor, Blocks Replication of SARS-CoV-2 and Other Coronaviruses

表环己糖醇环硫酸酯是一种基于机制的内质网 α-葡萄糖苷酶 II 抑制剂,可阻断 SARS-CoV-2 和其他冠状病毒的复制

Melissa Thaler, Tim P Ofman, Ken Kok, Jurriaan J A Heming, Elisha Moran, Isabelle Pickles, Anouk A Leijs, Adrianus M C H van den Nieuwendijk, Richard J B H N van den Berg, Gijs Ruijgrok, Zachary Armstrong, Clarisse Salgado-Benvindo, Dennis K Ninaber, Eric J Snijder, Constant A A van Boeckel, Marta A

Structure-Activity Relationship Studies of α-Ketoamides as Inhibitors of the Phospholipase A and Acyltransferase Enzyme Family

α-酮酰胺作为磷脂酶 A 和酰基转移酶家族抑制剂的构效关系研究

Juan Zhou, Elliot D Mock, Karol Al Ayed, Xinyu Di, Vasudev Kantae, Lindsey Burggraaff, Anna F Stevens, Andrea Martella, Florian Mohr, Ming Jiang, Tom van der Wel, Tiemen J Wendel, Tim P Ofman, Yvonne Tran, Nicky de Koster, Gerard J P van Westen, Thomas Hankemeier, Mario van der Stelt