日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

G.AI.A: An Integrated Machine-Learning Platform for Predicting Bioaccumulation and Ecotoxicity of Pharmaceuticals

G.AI.A:用于预测药物生物累积性和生态毒性的集成机器学习平台

Tsoukas, Evangelos; Papadourakis, Michail; Chontzopoulou, Eleni; Vythoulkas, Spyridon; Didachos, Christos; Cavouras, Dionisis; Zoumpoulakis, Panagiotis; Matsoukas, Minos-Timotheos

Design of Small Non-Peptidic Ligands That Alter Heteromerization between Cannabinoid CB(1) and Serotonin 5HT(2A) Receptors

设计能够改变大麻素 CB(1) 和血清素 5HT(2A) 受体之间异源异构化的小型非肽类配体

Matsoukas, Minos-Timotheos; Ciruela-Jardí, Marc; Gallo, Maria; Ferre, Sergi; Andreu, David; Casadó, Vicent; Pardo, Leonardo; Moreno, Estefanía

Influence of a Th17-Inducing Cytokine Milieu on Phenotypical and Functional Properties of Regulatory T Cells in Chronic Inflammatory Arthritis

Th17诱导细胞因子环境对慢性炎症性关节炎中调节性T细胞表型和功能特性的影响

Schwarz, Tobias; Almanzar, Giovanni; Wulfheide, Marie; Woidich, Robert; Holzer, Marie-Therese; Christoforou, Timotheos; Karle, Leonie; Radtke, David; Brauneiser, Franziska; Haaf, Thomas; Potabattula, Ramya; Ortega, Gabriela; Lesch, Klaus-Peter; Schäfer, Arne; Benoit, Sandrine; Schmieder, Astrid; Goebeler, Matthias; Schmalzing, Marc; Feuchtenberger, Martin; Prelog, Martina

Pharmacological Characterization of the Novel CRF1 Receptor Antagonist, Thiazolo[4,5-d] Pyrimidine Analog, M43

新型 CRF1 受体拮抗剂噻唑并[4,5-d]嘧啶类似物 M43 的药理学表征

Giatro, Spyridon Marios; Komontachakis, George; Kalantidou, Aikaterini; Lesgidou, Nastazia; Karageorgos, Vlasios; Teleb, Mohamed; Islam, Md Rabiul; Mavromoustakos, Thomas; Fahmy, Hesham; Venihaki, Maria; Matsoukas, Minos-Timotheos; Liapakis, George

Natural Compounds for Bone Remodeling: A Computational and Experimental Approach Targeting Bone Metabolism-Related Proteins

用于骨骼重塑的天然化合物:一种靶向骨代谢相关蛋白的计算和实验方法

Loukas, Alexandros-Timotheos; Papadourakis, Michail; Panagiotopoulos, Vasilis; Zarmpala, Apostolia; Chontzopoulou, Eleni; Christodoulou, Stephanos; Katsila, Theodora; Zoumpoulakis, Panagiotis; Matsoukas, Minos-Timotheos

Structural Features Influencing the Bioactive Conformation of Angiotensin II and Angiotensin A: Relationship between Receptor Desensitization, Addiction, and the Blood-Brain Barrier

影响血管紧张素 II 和血管紧张素 A 生物活性构象的结构特征:受体脱敏、成瘾和血脑屏障之间的关系

Graham J Moore, Harry Ridway, Laura Kate Gadanec, Vasso Apostolopoulos, Anthony Zulli, Jordan Swiderski, Konstantinos Kelaidonis, Veroniki P Vidali, Minos-Timotheos Matsoukas, Christos T Chasapis, John M Matsoukas0

Structural and Functional Insights into CRF Peptides and Their Receptors

CRF肽及其受体的结构和功能研究

Matsoukas, Minos-Timotheos; Panagiotopoulos, Vasilis; Karageorgos, Vlasios; Chrousos, George P; Venihaki, Maria; Liapakis, George

W254 in furin functions as a molecular gate promoting anti-viral drug binding: Elucidation of putative drug tunneling and docking by non-equilibrium molecular dynamics

弗林蛋白酶中的W254作为分子门控促进抗病毒药物结合:通过非平衡分子动力学阐明假定的药物隧道和对接机制

Ridgway, Harry; Orbell, John D; Matsoukas, Minos-Timotheos; Kelaidonis, Konstantinos; Moore, Graham J; Tsiodras, Sotiris; Gorgoulis, Vasilis G; Chasapis, Christos T; Apostolopoulos, Vasso; Matsoukas, John M

Periostin is overexpressed, correlated with fibrosis and differs among grades of cardiomyocyte hypertrophy in myectomy tissue of patients with hypertrophic cardiomyopathy

肥厚型心肌病患者心肌切除组织中骨膜蛋白过度表达,与纤维化相关,且在心肌细胞肥大程度之间存在差异

Nikolaos S Ioakeimidis, Antonios Pitsis, Thomas Zegkos, Dimitrios Ntelios, Timotheos Kelpis, Theodora Papamitsou, Despoina Parcharidou, Thomas Gossios, Georgios Efthimiadis, Soultana Meditskou

A Robust Machine Learning Framework Built Upon Molecular Representations Predicts CYP450 Inhibition: Toward Precision in Drug Repurposing

基于分子表征的稳健机器学习框架预测CYP450抑制:迈向精准药物再利用

Ouzounis, Sotiris; Panagiotopoulos, Vasilis; Bafiti, Vivi; Zoumpoulakis, Panagiotis; Cavouras, Dionisis; Kalatzis, Ioannis; Matsoukas, Minos-Timotheos; Katsila, Theodora