日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

RTK-Dependent Inducible Degradation of Mutant PI3Kα Drives GDC-0077 (Inavolisib) Efficacy

RTK依赖性诱导突变PI3Kα降解驱动GDC-0077(Inavolisib)疗效

Kyung W Song,Kyle A Edgar,Emily J Hanan,Marc Hafner,Jason Oeh,Mark Merchant,Deepak Sampath,Michelle A Nannini,Rebecca Hong,Lilian Phu,William F Forrest,Eric Stawiski,Stephen Schmidt,Nicholas Endres,Jane Guan,Jeffrey J Wallin,Jonathan Cheong,Emile G Plise,Gail D Lewis Phillips,Laurent Salphati,Timothy P Heffron,Alan G Olivero,Shiva Malek,Steven T Staben,Donald S Kirkpatrick,Anwesha Dey,Lori S Friedman

Noncovalent wild-type-sparing inhibitors of EGFR T790M

EGFR T790M 的非共价野生型保留抑制剂

Ho-June Lee, Gabriele Schaefer, Timothy P Heffron, Lily Shao, Xiaofen Ye, Steve Sideris, Shiva Malek, Emily Chan, Mark Merchant, Hank La, Savita Ubhayakar, Robert L Yauch, Valentina Pirazzoli, Katerina Politi, Jeff Settleman