日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Shaping Antimalarials: A Geometry-First Approach to PfCLK3 Covalent Inhibitors

抗疟药的调控:一种基于几何结构的PfCLK3共价抑制剂设计方法

Brettell, Skye B; Fuentes-Guerra Bustos, Carla; Sharma, Saumya; Cann, Gillian; Carruthers, Lauren V; Begen, Abbey; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Wide-field and non-invasive imaging of brain tumours with scattered light techniques

利用散射光技术对脑肿瘤进行广域无创成像

Binner, Philip; Radford, Jack; Starshynov, Ilya; Madhusudan, Mansa; Strathdee, Karen; Stevenson, Katrina; Walker, Matthew; Ciccone, Giuseppe; Tejeda, Gonzalo; Tobin, Andrew B; Vassalli, Massimo; Chalmers, Anthony J; Ekanayake, Jinendra; Faccio, Daniele

Physiological Significance of Endothelial M3 Muscarinic Receptors During Exercise

运动过程中内皮M3毒蕈碱受体的生理意义

Ackland, Gareth L; Hosford, Patrick S; Gutierrez Del Arroyo, Ana; Korsak, Alla; Machhada, Asif; Pickard, Jack; Gomez De La Torre, Genoveva Gomez; Stuckey, Daniel J; Tinker, Andrew; Tobin, Andrew B; Jeon, Jongrye; Wess, Jürgen; Gourine, Alexander V

Lysine targeting covalent inhibitors of malarial kinase PfCLK3

赖氨酸靶向共价抑制疟原虫激酶 PfCLK3 的抑制剂

Brettell, Skye B; Cann, Gillian; Begen, Abbey; Sharma, Saumya; Mahindra, Amit; Carruthers, Lauren V; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Optical, contact-free assessment of brain tissue stiffness and neurodegeneration

利用光学、非接触式方法评估脑组织硬度和神经退行性变

Binner, Philip; Starshynov, Ilya; Tejeda, Gonzalo; McFall, Aisling; Molloy, Colin; Ciccone, Giuseppe; Walker, Matthew; Vassalli, Massimo; Tobin, Andrew B; Faccio, Daniele

Targeting PfCLK3 with Covalent Inhibitors: A Novel Strategy for Malaria Treatment

利用共价抑制剂靶向 PfCLK3:一种治疗疟疾的新策略

Brettell, Skye B; Janha, Omar; Begen, Abbey; Cann, Gillian; Sharma, Saumya; Olaniyan, Niniola; Yelland, Tamas; Hole, Alison J; Alam, Benazir; Mayville, Emily; Gillespie, Ross; Capper, Michael; Fidock, David A; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Xanomeline displays concomitant orthosteric and allosteric binding modes at the M(4) mAChR

Xanomeline 在 M(4) mAChR 上表现出正构和变构结合模式。

Burger, Wessel A C; Pham, Vi; Vuckovic, Ziva; Powers, Alexander S; Mobbs, Jesse I; Laloudakis, Yianni; Glukhova, Alisa; Wootten, Denise; Tobin, Andrew B; Sexton, Patrick M; Paul, Steven M; Felder, Christian C; Danev, Radostin; Dror, Ron O; Christopoulos, Arthur; Valant, Celine; Thal, David M

Design, synthesis and evaluation of novel 2-phenyl-3-(1H-pyrazol-4-yl)pyridine positive allosteric modulators for the M(4) mAChR

设计、合成和评价新型2-苯基-3-(1H-吡唑-4-基)吡啶类M(4) mAChR正向变构调节剂

Jörg, Manuela; van der Westhuizen, Emma T; Lu, Yao; Christopher Choy, K H; Shackleford, David M; Khajehali, Elham; Tobin, Andrew B; Thal, David M; Capuano, Ben; Christopoulos, Arthur; Valant, Celine; Scammells, Peter J

A growing understanding of the role of muscarinic receptors in the molecular pathology and treatment of schizophrenia

人们对毒蕈碱受体在精神分裂症分子病理学和治疗中的作用有了越来越深入的了解

Dean, Brian; Bakker, Geor; Ueda, Hiroki R; Tobin, Andrew B; Brown, Alastair; Kanaan, Richard A A

Therapeutic validation of an orphan G protein-coupled receptor: The case of GPR84

孤儿G蛋白偶联受体的治疗验证:以GPR84为例

Marsango, Sara; Barki, Natasja; Jenkins, Laura; Tobin, Andrew B; Milligan, Graeme