日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Idler Compounds: A Simple Protocol for Openly Sharing Fridge Contents for Cross-Screening

闲置化合物:一种用于交叉筛查的开放式共享冰箱内容物的简单协议

Isaksson, Rebecka; Carter, Eve M; Hind, Charlotte K; Sutton, J Mark; Rudgyard, Hazel; Roberts, Adam H; Moon, Christopher W; Wang, Yinuo; Codony, Sandra; Martínez, Antón L; Bacon, Joanna; Todd, Matthew H

Identification of spirodioxolane nsP2 helicase inhibitors with antialphaviral activity

鉴定具有抗甲病毒活性的螺二氧戊环nsP2解旋酶抑制剂

Oh, Hans J; Sears, John D; Ramalingam, Bose Muthu; Saleem, Rahman Shah Zaib; Davis-Gilbert, Zachary W; Hossain, Mohammed Anwar; Moorman, Stella R; Ohja, Durbadal; Martinez, Sabian A; Burdick, Jane E; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Todd, Matthew H; Willson, Timothy M

Adsorption and Sensing Behavior of Pristine, P‐Doped, and Al‐Doped Boron Nitride Nanosheets Toward Toxic Hydrogen Fluoride Gas: Insights from Density Functional Theory Analysis

原始、磷掺杂和铝掺杂氮化硼纳米片对有毒氟化氢气体的吸附和传感行为:基于密度泛函理论分析的见解

Wong, Joseph K-H; Ast, Sandra; Yu, Mingfeng; Flehr, Roman; Counsell, Andrew J; Turner, Peter; Crisologo, Patrick; Todd, Matthew H; Rutledge, Peter J; Al‐Akhras, Ala'a; Ghazzy, Asma; Zakaraya, Zainab; S. Shraim, Ala'a; A. Sibai, Obada; Alsabbagh, Laila; Taher, Deeb; Siddique, Nihal; Daymond, Rashek Dewan; Fahim, Md Hasan Shahria; Golder, Utso Jyoti; Roy, Debashis; Roman, Abdullah Al; Ahmed, Mohammad Tanvir

Structure-activity relationships of fenarimol analogues with potent in vitro and in vivo activity against Madurella mycetomatis, the main causative agent of mycetoma

芬那利莫类似物具有强效的体外和体内抗马杜拉菌(足菌肿的主要致病菌)活性,并对其构效关系进行了研究。

Duong, Hung Phat; Melechov, Dmitrij; Lim, Wilson; Ma, Jingyi; Scroggie, Kymberley R; Rajendra, Luxsika; Perry, Benjamin; Cruz, Luiza R; Saleem, Rahman Shah Zaib; Rutledge, Peter J; Motion, Alice; van de Sande, Wendy W J; Todd, Matthew H

Structure-Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis

一系列咪唑并吡啶类化合物的结构-性质优化及其在内脏利什曼病中的应用

Dichiara, Maria; Simpson, Quillon J; Quotadamo, Antonio; Jalani, Hitesh B; Huang, Anson X; Millard, Caroline C; Klug, Dana M; Tse, Edwin G; Todd, Matthew H; Silva, Daniel Gedder; da Silva Emery, Flavio; Carlson, J Eric; Zheng, Shao-Liang; Vleminckx, Margot; Matheeussen, An; Caljon, Guy; Pollastri, Michael P; Sjö, Peter; Perry, Benjamin; Ferrins, Lori

Target 2035 - an update on private sector contributions

2035年目标——私营部门贡献的最新情况

Ackloo, Suzanne; Antolin, Albert A; Bartolome, Jose Manuel; Beck, Hartmut; Bullock, Alex; Betz, Ulrich A K; Böttcher, Jark; Brown, Peter J; Chaturvedi, Menorca; Crisp, Alisa; Daniels, Danette; Dreher, Jan; Edfeldt, Kristina; Edwards, Aled M; Egner, Ursula; Elkins, Jon; Fischer, Christian; Glendorf, Tine; Goldberg, Steven; Hartung, Ingo V; Hillisch, Alexander; Homan, Evert; Knapp, Stefan; Köster, Markus; Krämer, Oliver; Llaveria, Josep; Lessel, Uta; Lindemann, Sven; Linderoth, Lars; Matsui, Hisanori; Michel, Maurice; Montel, Florian; Mueller-Fahrnow, Anke; Müller, Susanne; Owen, Dafydd R; Saikatendu, Kumar Singh; Santhakumar, Vijayaratnam; Sanderson, Wendy; Scholten, Cora; Schapira, Matthieu; Sharma, Sujata; Shireman, Brock; Sundström, Michael; Todd, Matthew H; Tredup, Claudia; Venable, Jennifer; Willson, Timothy M; Arrowsmith, Cheryl H

Reaction hijacking inhibition of Plasmodium falciparum asparagine tRNA synthetase

恶性疟原虫天冬酰胺tRNA合成酶的反应劫持抑制

Xie, Stanley C; Wang, Yinuo; Morton, Craig J; Metcalfe, Riley D; Dogovski, Con; Pasaje, Charisse Flerida A; Dunn, Elyse; Luth, Madeline R; Kumpornsin, Krittikorn; Istvan, Eva S; Park, Joon Sung; Fairhurst, Kate J; Ketprasit, Nutpakal; Yeo, Tomas; Yildirim, Okan; Bhebhe, Mathamsanqa N; Klug, Dana M; Rutledge, Peter J; Godoy, Luiz C; Dey, Sumanta; De Souza, Mariana Laureano; Siqueira-Neto, Jair L; Du, Yawei; Puhalovich, Tanya; Amini, Mona; Shami, Gerry; Loesbanluechai, Duangkamon; Nie, Shuai; Williamson, Nicholas; Jana, Gouranga P; Maity, Bikash C; Thomson, Patrick; Foley, Thomas; Tan, Derek S; Niles, Jacquin C; Han, Byung Woo; Goldberg, Daniel E; Burrows, Jeremy; Fidock, David A; Lee, Marcus C S; Winzeler, Elizabeth A; Griffin, Michael D W; Todd, Matthew H; Tilley, Leann

CACHE (Critical Assessment of Computational Hit-finding Experiments): A public-private partnership benchmarking initiative to enable the development of computational methods for hit-finding

CACHE(计算命中发现实验的关键评估):一项公私合作的基准测试计划,旨在促进命中发现计算方法的发展。

Ackloo, Suzanne; Al-Awar, Rima; Amaro, Rommie E; Arrowsmith, Cheryl H; Azevedo, Hatylas; Batey, Robert A; Bengio, Yoshua; Betz, Ulrich A K; Bologa, Cristian G; Chodera, John D; Cornell, Wendy D; Dunham, Ian; Ecker, Gerhard F; Edfeldt, Kristina; Edwards, Aled M; Gilson, Michael K; Gordijo, Claudia R; Hessler, Gerhard; Hillisch, Alexander; Hogner, Anders; Irwin, John J; Jansen, Johanna M; Kuhn, Daniel; Leach, Andrew R; Lee, Alpha A; Lessel, Uta; Morgan, Maxwell R; Moult, John; Muegge, Ingo; Oprea, Tudor I; Perry, Benjamin G; Riley, Patrick; Rousseaux, Sophie A L; Saikatendu, Kumar Singh; Santhakumar, Vijayaratnam; Schapira, Matthieu; Scholten, Cora; Todd, Matthew H; Vedadi, Masoud; Volkamer, Andrea; Willson, Timothy M

Target 2035 - update on the quest for a probe for every protein

2035年目标——为每种蛋白质寻找探针的最新进展

Müller, Susanne; Ackloo, Suzanne; Al Chawaf, Arij; Al-Lazikani, Bissan; Antolin, Albert; Baell, Jonathan B; Beck, Hartmut; Beedie, Shaunna; Betz, Ulrich A K; Bezerra, Gustavo Arruda; Brennan, Paul E; Brown, David; Brown, Peter J; Bullock, Alex N; Carter, Adrian J; Chaikuad, Apirat; Chaineau, Mathilde; Ciulli, Alessio; Collins, Ian; Dreher, Jan; Drewry, David; Edfeldt, Kristina; Edwards, Aled M; Egner, Ursula; Frye, Stephen V; Fuchs, Stephen M; Hall, Matthew D; Hartung, Ingo V; Hillisch, Alexander; Hitchcock, Stephen H; Homan, Evert; Kannan, Natarajan; Kiefer, James R; Knapp, Stefan; Kostic, Milka; Kubicek, Stefan; Leach, Andrew R; Lindemann, Sven; Marsden, Brian D; Matsui, Hisanori; Meier, Jordan L; Merk, Daniel; Michel, Maurice; Morgan, Maxwell R; Mueller-Fahrnow, Anke; Owen, Dafydd R; Perry, Benjamin G; Rosenberg, Saul H; Saikatendu, Kumar Singh; Schapira, Matthieu; Scholten, Cora; Sharma, Sujata; Simeonov, Anton; Sundström, Michael; Superti-Furga, Giulio; Todd, Matthew H; Tredup, Claudia; Vedadi, Masoud; von Delft, Frank; Willson, Timothy M; Winter, Georg E; Workman, Paul; Arrowsmith, Cheryl H

There is no market for new antibiotics: this allows an open approach to research and development

新抗生素没有市场:这使得研发可以采取开放的态度。

Klug, Dana M; Idiris, Fahima I M; Blaskovich, Mark A T; von Delft, Frank; Dowson, Christopher G; Kirchhelle, Claas; Roberts, Adam P; Singer, Andrew C; Todd, Matthew H